2004-2005 first year review (only principles drugs have been updated; doesn’t include derm) 21...
TRANSCRIPT
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2004-2005First Year Review
(only Principles drugs have been updated; doesn’t include Derm)
April 21, 202303:57 AM
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Abciximab
Antiplatelet
Anti-GPIIb/IIIa receptor antibody
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Acetaminophen
Analgesic, Antipyretic
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Adalimumab
TNF inhibitor
Anti-TNF antibodyUsed in rheumatoid arthritis
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Adrenocorticotropin(ACTH)
Anterior pituitary hormoneAnticonvulsant
Stimulates synthesisand release of cortisol
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Alemtuzumab
Antineoplastic
Anti-CD52 antibody
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Alfentanil
OpioidGeneral anaesthetic
Intravenous anaesthetic
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Allopurinol
AntigoutAntineoplastic (supporting
agent)
Folic acid analogueXanthine oxidase inhibitor
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Amantadine
AntiviralAntiparkinson
Treatment of Influenza A Inhibits replication
at the stage of uncoatingInhibits dopamine release
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Amikacin
Aminoglycoside antibioticBactericidal protein synthesis
inhibitor
30S ribosomeFreezes initiation
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Aminocaproic acid (EACA)
Procoagulant
Inhibitor of plasminogen activation
(decreases fibrinolysis)
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Aminoglutethimide
AntineoplasticImmunosuppressive
Glucocorticoid antagonistAromatase inhibitor
(decreases steroid synthesis)
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Aminoglycosides
AntibioticsBactericidal protein synthesis
inhibitors
30S ribosomeFreeze initiation
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Amitriptyline
Tricyclic antidepressant (TCA)
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Amoxicillin
Penicillin antibioticCell wall synthesis inhibitor
Antiulcer
Amino penicillinInhibits peptidoglycan cross-
linking
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Amphetamine
Indirect sympathomimeticDrug of abuse
ADD treatmentStimulant
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Ampicillin
Penicillin antibioticCell wall synthesis inhibitor
Amino penicillinInhibits peptidoglycan cross-
linking
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Amsacrine
Antineoplastic
Miscellaneous
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Angiostatin
Antineoplastic
Angiogenesis inhibitor
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Anistreplase
Thrombolytic
Streptokinase + plasminogen
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Anti-thymocyte globulin
Immunosuppressive
Anti-T cell antibody
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Aprotinin
Procoagulant
Fibrinolytic inhibitorSerine protease inhibitor
(“serpin”)Streptokinase inhibitor
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Argatroban
Anticoagulant
Direct thrombin inhibitor
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L-asparaginase
Antineoplastic
Protein synthesis inhibitor
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Aspirin(Acetylsalicylic acid, ASA)
NSAID (acetylsalicylate)Analgesic, Anti-inflammatory
Antipyretic, Antiplatelet
Irreversible cyclooxygenase inhibitor
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Atropine
Anticholinergic
AntimuscarinicTreatment for bradycardia,
diarrhea, cholinesterase poisoning
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Azathioprine
ImmunosuppressiveAntineoplastic
Antimetabolite(“pseudofeedback inhibition” of
HGPRT and PRP)
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Azithromycin
Macrolide antibioticBacteriostatic protein synthesis
inhibitor
50S ribosome Inhibits translocation
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Aztreonam
New lactam antibiotic
Monobactam
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Baclofen
Skeletal muscle relaxantAnxiolytic
GABAB agonist
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Bacitracin
AntibioticCell wall synthesis inhibitor
Topical, not a lactam, Inhibits dephosphorylation of
bactoprenol
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Basiliximab
Immunosuppressive
Anti-CD25 (interleukin 2 receptor)
Organ transplant (antirejection)
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Benzathine penicillin G
Penicillin antibioticCell wall synthesis inhibitor
Inhibits peptidoglycan cross-linking Repository preparation
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Benztropine
AnticholinergicAntiparkinson
Muscarinic receptor antagonist
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Betamethasone
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidNot by inhalation
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Bethanecol
Cholinomimetic
Muscarinic agonistInduces defecation and
urinationBronchoconstrictor
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Bleomycin
Antineoplastic
Natural productAntibiotic
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Bivalirudin
Anticoagulant
Direct thrombin inhibitor
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Bortezomib
Antineoplastic
Proteosome inhibitor
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Bradykinin
Inflammatory mediator
Plasma, hypotension, pain
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Bromocriptine
Antiparkinson
Dopamine (D2) agonistInhibits prolactin release
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Brupropion
Second generation antidepressant
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Buprenorphine
Opioid
Partial agonist
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Buspirone
Sedative/hypnoticAnxiolytic
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Busulfan
Antineoplastic
Alkylating agent
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Butorphanol
OpioidAnalgesic
receptor partial agonistor antagonist
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C3a, C5a
Inflammatory mediators
Anaphylatoxins Low molecular weight
complement cleavage products
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Carbamazepine
Anticonvulsant
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Carbenicillin
Penicillin antibioticCell wall synthesis inhibitor
Anti-pseudomonal penicillinInhibits peptidoglycan cross-
linking
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Carbidopa
Antiparkinson
Peripheral dopa decarboxylase inhibitor
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Carmustine (BCNU)
Antineoplastic
Alkylating AgentNitrosourea
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Cefaclor
Cephalosporin antibioticCell wall synthesis inhibitor
2nd generationOral
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Cefadroxil
Cephalosporin antibioticCell wall synthesis inhibitor
1st generationOral
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Cefepime
Cephalosporin antibioticCell wall synthesis inhibitor
4th generationCSF penetration
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Cefotaxime
Cephalosporin antibioticCell wall synthesis inhibitor
3rd generationCSF penetration
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Cefoxitin
Cephalosporin antibioticCell wall synthesis inhibitor
2nd generation
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Ceftazidime
Cephalosporin antibioticCell wall synthesis inhibitor
3rd generation
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Ceftriaxone
Cephalosporin antibioticCell wall synthesis inhibitor
3rd generationCSF penetration
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Cefuroxime
Cephalosporin antibioticCell wall synthesis inhibitor
2nd generationCSF penetration
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Celecoxib
NSAIDAnti-inflammatory
Cyclooxygenase 2 (COX-2) inhibitor
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Cephalexin
Cephalosporin antibioticCell wall synthesis inhibitor
1st generationOral
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Cephalosporins
Antibiotics lactam
Cell wall synthesis inhibitorsInhibit cross-linking of
peptidoglycan
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Cephalothin
Cephalosporin antibioticCell wall synthesis inhibitor
1st generationOral
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Cetirizine
Antihistamine
H1 antagonist Non-sedating
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Chloral hydrate
Sedative/HypnoticGeneral anaesthetic
Acts on GABAA receptor complexSimilar to barbiturates
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Chloramphenicol
AntibioticBacteriostatic protein synthesis
inhibitor
50S ribosomeInhibits peptide bond formation
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Chlordiazepoxide
Sedative/hypnoticAnxiolytic
Benodiazepine Acts on GABAA receptor
complex
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Chlorpheniramine
Classical antihistamine
H1 antagonist
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Chlorpromazine
Antipsychotic
Phenothiazine
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Ciprofloxacin
Fluoroquinolone antibioticDNA replication inhibitor
Inhibits bacterial DNA gyrase
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Cisplatin
Antineoplastic
MiscellaneousCross-linking agent
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Clarithromycin
Macrolide antibioticBacteriostatic protein synthesis
inhibitor Antiulcer
50S ribosomeInhibits translocation
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Clavulanic acid
-lactamase inhibitor
Combined with antibacterials
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Clindamycin
AntibioticBacteriostatic protein synthesis
inhibitor
50S ribosomeAnaerobic infections
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Clopidogrel
Antiplatelet
ADP receptor antagonist
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Cloxacillin
Penicillin antibioticCell wall synthesis inhibitor
Penicillinase resistant penicillinInhibits peptidoglycan cross-
linking
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Clozapine
Antipsychotic
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Cobalamin(cyanocobalamin, hydroxocobalamin)
Vitamin
Treatment forvitamin B12 deficiency
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Cocaine
Indirect sympathomimeticDrug of abuse
Topical anaesthetic
StimulantLocal anaesthetic
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Codeine
OpioidAnalgesic
Weak agonist
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Cortisol (Hydrocortisone)
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroid
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Cyclophosphamide
Antineoplastic
Alkylating AgentNitrogen mustard
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Cycloserine
AntibioticCell wall synthesis inhibitor
Secondary TB drugInhibits formation of Park
nucleotide
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Cyclosporine
ImmunosuppressiveAntineoplastic
Binds cyclophilinInhibits calcineurin
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Cytarabine (AraC)
Antineoplastic
Antimetabolite
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Dacarbazine
Antineoplastic
Alkylating Agent
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Daclizumab
Immunosuppressive
Anti-CD25 (interleukin 2 receptor) antibody
Organ transplant (anti-rejection)
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Dactinomycin
Antineoplastic
Natural productAntibiotic
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Dalteparin
Anticoagulant
LMW HeparinATIII activator
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Dantrolene
Skeletal muscle relaxant
Ryanodine receptor antagonistTreatment for malignant hyperthermia
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Dapsone
Sulfone antibioticNucleic acid and
protein synthesis inhibitor
Inhibits dihydropteroate synthetase
Leprosy
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Daunorubicin
Antineoplastic
Anthracycline antibiotic Natural product
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Deprenyl/selegiline
Antiparkinson
Monoamine oxidase B inhibitor(MAO-I)
Potentiates effects of L-Dopa
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Desipramine
Tricyclic antidepressant (TCA)
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Desmopressin acetate
Synthetic analogue ofarginine vasopressin
Used in treatment of bleeding disorders
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Dexamethasone
AdrenocorticosteroidGlucocorticoidAntineoplastic
Antiemetic
Anti-inflammatory steroidNot by inhalation
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Dextromethorphan
Opioid
Antitussive
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Diazepam
Sedative/hypnoticAnxiolytic
Anticonvulsant
Benzodiazepine Acts on GABAA receptor complex
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Diflunisal
NSAIDAnalgesic, Anti-inflammatory
Antipyretic
Cyclooxygenase inhibitor
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Diphenhydramine
Classical antihistamineAntiemetic
H1 antagonist
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Diphenoxylate docusate
Antidiarrheal
Opiate
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Dipyridamole
Antiplatelet
Phosphodiesterase inhibitor(increases cAMP)
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Doxorubicin
Antineoplastic
Anthracycline antibioticNatural product
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Doxycycline
Tetracycline antibioticBacteriostatic protein synthesis
inhibitor
30S ribosomePrevents aminoacyl tRNA attachment
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Drotrecogin alfa(Activated Protein C)
Anticoagulant
Many actionsTreatment for septic shock
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Edrecolomab
Antineoplastic
Anti-17-1A antibody
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Enflurane
General anaesthetic
Inhaled anaesthetic
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Enoxaparin
Anticoagulant
LMW HeparinATIII activator
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Entacapone
Antiparkinson
Peripheral catechol-o-methyltransferase inhibitor
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Ephedra(Ma Huang)
Dietary supplement
Amphetamine-like stimulant
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Eptifibatide
Antiplatelet
GPIIb/IIIa antagonist
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Erythromycin
Macrolide antibioticBacteriostatic protein synthesis
inhibitor
50S ribosomeInhibits translocation
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Erythropoietin (EPO)
Cytokine
Primary regulator of RBC synthesis
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Etanercept
TNF inhibitor
Tumor necrosis factor receptor+ Fc portion of IgG
Used in rheumatoid arthritis
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Ethanol
Drug of abuse
Sedative
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Ethosuximide
Anticonvulsant
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Etomidate
General anaesthetic
Intravenous anaesthetic
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Etoposide
Antineoplastic
Natural productPlant alkaloid
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Fentanyl
OpioidAnalgesic
receptor agonist
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Fexofenadine
Antihistamine
H1 antagonistNon-sedating
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Flumazenil
Benzodiazepine antagonist
Acts on GABAA receptor complex
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5-Fluorouracil
Antineoplastic
AntimetaboliteThymidylate synthase inhibitor
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Fluoxetine
Antidepressant
Selective serotonin reuptake inhibitor (SSRI)
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Flurazepam
Sedative/Hypnotic
Benzodiazepine Acts on GABAA receptor
complex
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Fluorinated Quinolonesciprofloxacin, norfloxacin
AntibioticsDNA replication inhibitors
Inhibit bacterial DNA gyrase
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Folic acid
Vitamin
Treatment for folicacid deficiency
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Gefitinib
Antineoplastic
MiscellaneousTyrosine kinase inhibitor
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Gemcitabine
Antineoplastic
Antimetabolite
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Gemtuzumab
Antineoplastic
Anti-CD33 antibody
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Gentamicin
Aminoglycoside antibioticBactericidal protein synthesis
inhibitor
30S ribosome Freezes initiation
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Ginko biloba
Dietary supplement
Treatment of Alzheimer symptoms
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Glutethimide
Sedative/Hypnotic
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Haloperidol
Antipsychotic
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Halothane
General anaesthetic
Inhaled anaesthetic
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Heparin
Anticoagulant
ATIII activator
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Heroin
Drug of abuse
Opioid
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Hirudin
Anticoagulant
Direct thrombin inhibitor(DTI)
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Histamine
Inflammatory mediator
Stored in mast cells and basophils
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Hydrocortisone
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroid
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4-Hydroxycoumarin
Oral anticoagulant
Vitamin K synthesis inhibitor
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Hydroxyurea
Antineoplastic
MiscellaneousRibonucleotide reductase
inhibitor
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Hydroxyzine
Classical antihistamine
H1 antagonist
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Ibritumomab
Antineoplastic
Anti-CD20 antibody
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Ibuprofen
NSAIDAnalgesic, Anti-inflammatory
Antipyretic
Reversible cyclooxygenase inhibitor
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Imatinib
Antineoplastic
MiscellaneousTyrosine kinase inhibitor
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Imipenem/Cilastatin
New lactam antibiotic
Cilastatin inhibits akidney dipeptidase that inactivates imipenem
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Imipramine
Indirect sympathomimeticTricyclic antidepressant (TCA)
Antimicturant
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Indomethacin
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitorTocolytic
Uterine relaxant
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Infliximab
TNF inhibitor
Anti-TNF monoclonal antibodyTreatment of IBD
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Interferon alpha
Antiviral for hepatitisAntineoplastic
Cytokine
Anti-angiogenesis
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Interleukin 2
Cytokine Antineoplastic
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Interleukin 11
Cytokine Antineoplastic (supporting
agent)
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Interleukin 12
Cytokine Antineoplastic (supporting
agent)
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Irinotecan
Antineoplastic
Natural product
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Isoflurane
General anaesthetic
Inhaled anaesthetic
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Kallidin
Inflammatory mediator
Plasma, hypotension, pain
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Kava kava
Dietary supplement
Stress relief andtreatment of insomnia
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Ketamine
General anaestheticDrug of abuse
Sedative
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Ketoprofen
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
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Lepirudin
Anticoagulant
Direct thrombin inhibitor (DTI)
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Levodopa
Antiparkinson
Dopamine precursor
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Leucovorin
Antineoplastic (supporting agent)
Folic acid analogue(used in methotrexate rescue)
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Leukotriene B4 (LTB4)
Inflammatory mediator
Lipoxygenase productof arachidonate metabolism
Chemotactic
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Leukotrienes C4, D4, E4
(LTC4, LTD4, LTE4)
Inflammatory mediators
Cysteinyl leukotrienesPeptidyl leukotrienes
SRS-ALipoxygenase products ofarachidonate metabolism
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Lidocaine
Class I antiarrhythmicLocal anaesthetic
Na+ channel blocker(activated and inactivated channels)
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Linezolid
Oxazolidinone antibioticProtein synthesis inhibitor
50S ribosomal subunit
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Lithium
Antidepressant
Used to treatmanic/depressive disorder
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Lomustine (CCNU)
Antineoplastic
Alkylating AgentNitrosourea
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Loperamide
Antidiarrheal
Opiate
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Loratidine
Antihistamine
H1 antagonistNon-sedating
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Lorazepam
AnxiolyticAnticonvulsant
BenzodiazepineActs on GABAA receptor complex
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Lysergic acid diethylamide
(LSD)
Drug of abuse
Hallucinogen
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Macrolideserythromycin, azithromycin, clarithromycin
AntibioticsBacteriostatic protein synthesis
inhibitors
50S ribosome
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Marijuana
Drug of abuse
Cannabinoid
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Mechlorethamine
Antineoplastic
Alkylating AgentNitrogen mustard
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Meclofenamate
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
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Melphalan
Antineoplastic
Alkylating AgentNitrogen mustard
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Meperidine
Opioid analgesic
receptor agonist
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Mepivacaine
Local anaesthetic
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Meprobamate
Sedative/hypnoticAnxiolytic
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6-Mercaptopurine
Antineoplastic
Antimetabolite(“pseudofeedback inhibition” of
HGPRT and PRP – purine synthesis)
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Mesna
Antineoplastic (supporting agent)
Prevent hemorrhagic cystitisdue to cyclophosphamide
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Methicillin
Penicillin antibioticCell wall synthesis inhibitor
Pencillinase resistant penicillin Inhibits peptidoglycan cross-
linking
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Methotrexate
ImmunosuppressiveAntineoplastic
Folic acid antagonistDihydrofolate reductase
inhibitor
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Methylprednisolone
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidNot by inhalation
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Metronidazole
AntibioticAntiparasitic
Antiulcer
AnaerobesReduction leads to intermediates
that damage DNA
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Minocycline
Tetracycline antibioticBacteriostatic protein synthesis
inhibitor
30S ribosomePrevents aminoacyl tRNA attachment
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Mitomycin C
Antineoplastic
Natural productAntibiotic
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Metamphetamine
Drug of abuse
Stimulant
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Methadone
Opioid
receptor agonist
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Montelukast
Leukotriene inhibitor
LTR1 and LTD4 antagonistAsthma treatment
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Morphine
OpioidAnalgesic
receptor agonist
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Muromonab-CD3
Immunosuppressive
Mouse monoclonal anti-CD3 antibody
Organ transplant (anti-rejection)
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Mycophenolate
Immunosuppressive
Inhibits inosine monophosphate dehydrogenase activity
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Nalbuphine
Opioid antagonist
receptor antagonist
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Nalmefene
Opioid antagonist
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Nalorphine
Opioid antagonist
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Naloxone
Opioid antagonist
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Naltrexone
Opioid antagonist
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Naproxen
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
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Nafcillin
Penicillin antibioticCell wall synthesis inhibitor
Penicillinase resistant penicillinInhibits peptidoglycan cross-
linking
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Neomycin
Aminoglycoside antibioticBactericidal protein synthesis
inhibitor
30S ribosomeFreezes initiation
Topical
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Neostigmine
Anticholinesterase
VasodilatorTreatment for myaesthenia gravisPromotes defecation and urination
Bronchoconstrictor
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Netilmicin
Aminoglycoside antibioticBactericidal protein synthesis
inhibitor
30S ribosomeFreezes initiation
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Nicotine
CholinomimeticDrug of abuse
Nicotinic receptor agonist(skeletal muscle contraction)
StimulantSmoking cessation medication
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Nitrous oxide
General anaesthetic
Inhaled anaesthetic
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Non-steroidalAnti-inflammatory Drugs
(NSAIDs)
Analgesic, Anti-inflammatory, Antipyretic
Cyclooxygenase inhibitors
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Norfloxacin
Fluoroquinolone antibioticDNA replication inhibitor
Inhibits bacterial DNA gyrase
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Nortriptyline
Tricyclic antidepressant (TCA)
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Omalizumab
Anti-asthma
Anti-IgE antibody
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Oxacillin
Penicillin antibioticCell wall synthesis inhibitor
Pencillinase resistant penicillinInhibits peptidoglycan cross-
linking
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Oxazepam
Sedative/hypnoticAnxiolytic
BenzodiazepineActs on GABAA receptor complex
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Oxybutinin
Anticholinergic
Muscarinic receptor antagonistPrevents urination
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Oxycodone
Analgesic
Opioid agonist
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Oxytetracycline
Tetracycline antibioticBacteriostatic protein synthesis
inhibitor
30S ribosomePrevents aminoacyl tRNA attachment
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Paclitaxel
Antineoplastic
Natural productPlant alkaloid (taxane)
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Palivizumab
Antiviral
Monoclonal antibody againstthe surface of
respiratory syncytial virus
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Para-aminosalicylic acid
AntibioticNucleic acid and
protein synthesis inhibitor
Inhibits dihydropteroate synthetaseSecondary TB drug
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Paraldehyde
Sedative/Hypnotic
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Penicillins
lactam antibioticsCell wall synthesis inhibitors
Inhibit cross-linking of peptidoglycan
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Penicillin G
Penicillin antibioticCell wall synthesis inhibitor
Acid labileInhibits peptidoglycan cross-
linking
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Penicillin V
Penicillin antibioticCell wall synthesis inhibitor
More acid resistant than Penicillin G
Inhibits peptidoglycan cross-linking
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Pentazocine
Opioid analgesic
receptor partial agonist or antagonist
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Pentobarbital
Sedative/Hypnotic
Barbiturate
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Pentostatin
Antineoplastic
MiscellaneousEnzyme inhibitor
(blocks purine synthesis)
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Phencyclidine (PCP)
Drug of abuse
Hallucinogen
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Phenobarbital
Sedative/HypnoticAnticonvulsant
Barbiturate
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Phenytoin
AnticonvulsantClass I antiarrhythmic
Na+ channel blocker(inactivated channels)
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Phytonadione
Vitamin K
Warfarin antagonist
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Piperacillin
Penicillin antibioticCell wall synthesis inhibitor
Anti-pseudomonal penicillinInhibits peptidoglycan cross-
linking
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Piroxicam
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
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Platelet Activating Factor (PAF)
Inflammatory mediator
LipidHypotensive
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Polymyxin B
AntibioticDisrupts gram negative cell
membrane
Binds phosphatidylethanolamineBactericidal
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Pramipexole
Antiparkinson
Dopamine agonist (non-ergot)
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Prednisone
AdrenocorticosteroidGlucocorticoid Antineoplastic
Anti-inflammatoryNot by inhalation
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Primidone
Anticonvulsant
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Probenecid
Uricosuric
Adjunct in penicillin therapy
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Procaine
Local anaesthetic
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Procaine Penicillin G
Penicillin antibioticCell wall synthesis inhibitor
Repository preparationInhibits peptidoglycan cross-
linking
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Procarbazine
Antineoplastic
MiscellaneousProbably acts as alkylating
agent
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Promethazine
Classical antihistamineAntipsychotic
Antiemetic
H1 antagonist
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Propofol
General anaesthetic
Intravenous anaesthetic
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Prostaglandin D2 (PGD2)
Bronchoconstrictor
Cyclooxygenase product of arachidonate metabolism
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Prostaglandin E2 (PGE2)Dinoprostone (Dinoprost)
Oxytocic prostaglandinInflammatory mediator
Cyclooxygenase product of arachidonate metabolism
Uterine stimulantCervical ripener
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Prostaglandin F2 (PGF2)
Inflammatory mediator
Cyclooxygenase product of arachidonate metabolism
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Prostaglandin I2 (PGI2)
Inflammatory mediator
Inhibits platelet aggregation
Cyclooxygenase product of arachidonate metabolism
Prostacyclin
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Protamine Sulfate
Heparin antagonist
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Quinopristin/Dalfopristin
Streptogramin antibioticProtein synthesis inhibitor
50S ribosomal subunit
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Resperidone
Antipsychotic
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Rifampin
AntibioticNucleic acid synthesis inhibitor
Inhibits DNA dependent RNA polymerase
Major drug for TB
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Rituxumab
Antineoplastic
Anti-CD20 antibody
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Rofecoxib
NSAIDAnti-inflammatory
Cyclooxygenase 2 (COX-2) inhibitor
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Ropinirole
Antiparkinson
Dopamine agonist (non-ergot)
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Sargramostim(GM-CSF)
Colony stimulating factor
WBC (granulocyte and macrophage)
stimulant
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Sertraline
Antidepressant
Selective serotonin reuptake inhibitor (SSRI)
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Sildenafil
Vasodilator
Promotes erection
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Silver sulfadiazine
Sulfonamide antibioticMicrobial nucleic acid
and protein synthesis inhibitor
Inhibits dihydropteroate synthetase
Topical
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Sirolimus
Immunosuppressive
Binds FKBP, inhibits mTOR (mammalian kinase target of
rapamycin) & cell cycle progression
Rapamycin
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Spectinomycin
AntibioticBacteriostatic protein synthesis
inhibitor
30S ribosome
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St. John’s Wort
Dietary supplement
Antidepressant
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Streptokinase
Thrombolytic
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Streptomycin
Aminoglycoside antibioticBactericidal protein synthesis
inhibitor
30S ribosomeFreezes initiation
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Sufentanil
OpioidGeneral anaesthetic
Intravenous anaesthetic
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Sulfacetamide
Sulfonamide antibioticMicrobial nucleic acid
and protein synthesis inhibitor
Inhibits dihydropteroate synthetaseTopical
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Sulfadoxine
Sulfonamide antibioticMicrobial nucleic acid
and protein synthesis inhibitor
Dihydropteroate synthetase inhibitor
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Sulfamethoxazole
Sulfonamide antibioticMicrobial nucleic acid
and protein synthesis inhibitor
Inhibits dihydropteroate synthetase
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Sulfisoxazole
Sulfonamide antibioticNucleic acid and
protein synthesis inhibitor
Inhibits dihydropteroate synthetase
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Sulfonamides
AntibioticsNucleic acid and
protein synthesis inhibitors
Inhibit dihydropteroate synthetase
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Sulindac
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
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Tacrolimus
ImmunosuppressiveAntineoplastic
Binds FKBP (FK506 binding protein)
Inhibits calcineurin
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Temazepam
Sedative/Hypnotic
BenzodiazepineActs on GABAA receptor complex
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Tetracaine
Local anaesthetic
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Tetracycline
AntibioticBacteriostatic protein synthesis
inhibitor Antiulcer
30S ribosomePrevents aminoacyl tRNA attachment
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Thalidomide
AntineoplasticLeprosy treatment
Anti-angiogenicAnti-TNF
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6-Thioguanine
Antineoplastic
Antimetabolite (“pseudofeedback inhibition” of
HGPRT and PRP – purine synthesis)
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Thiopental
General anaesthetic
Ultra-short-acting barbiturate
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Thioridazine
Antipsychotic
Phenothiazine
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Thiotepa
Antineoplastic
Alkylating agent
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Thiothixene
Antipsychotic
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Thromboxane A2 (TXA2)
Autacoid
Promotes platelet aggregation Cyclooxygenase product of arachidonate metabolism
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Ticlopidine
Antiplatelet
ADP receptor antagonist
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Ticarcillin
Penicillin antibioticCell wall synthesis inhibitor
Anti-pseudomonal penicillinInhibits peptidoglycan cross-
linking
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Tissue plasminogen activators
Thrombolytics
alteplase, reteplase, tenecteplase
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Tobramycin
Aminoglycoside antibioticBactericidal protein synthesis
inhibitor
30S ribosomeFreezes initiation
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Tolterodine
Anticholinergic
Muscarinic receptor antagonistPrevents urination
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Tositumomab
Antineoplastic
Anti-CD20 antibody
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Tranylcypromine
Antidepressant
Monoamine oxidase inhibitor (MAO-I)
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Trastuzumab
Antineoplastic
Anti-HER2 antibody
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Triazolam
Sedative/Hypnotic
BenzodiazepineActs on GABAA receptor complex
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Trifluoperazine
Antipsychotic
Phenothiazine
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Trihexyphenidyl
Antiparkinson
Antimuscarinic
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Trimethoprim
AntibioticProtein and nucleic acid
synthesis inhibitor
Folic acid antagonistInhibits bacterial dihydrofolate
reductase
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Tripelennamine
Classical antihistamine
H1 antagonist
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Tumor necrosis factor
CytokineAntineoplastic
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Urokinase
Thrombolytic
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Valproic acid
Anticonvulsant
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Vancomycin
AntibioticInhibits cell wall synthesis
Not a lactam
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Vigabatrin
Anticonvulsant
Irreversible GABA aminotransferase inhibitor
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Vinblastine
Antineoplastic
Vinca alkaloidNatural product
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Vincristine
Antineoplastic
Vinca alkaloidNatural product
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Warfarin
Anticoagulant
Vitamin K synthesis inhibitor
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Zafirlukast
Leukotriene inhibitor
LTR1 and LTD4 antagonistAsthma treatment
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Zileuton
Leukotriene inhibitor
5-lipoxygenase inhibitorUsed in asthma
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Zolpidem
Sedative/Hypnotic
Non-benzodiazepine