dr.ajay - pharmacokinetic
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8/3/2019 Dr.Ajay - Pharmacokinetic
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Lx+ @b`w Fn`q`kLjt|+ ca X`v`vn`v|x`
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Fck|jk|vFck|jk|v
Gk|xclzf|gck
Chbjf|gqj
Ljagkg|gck
Ljvfxgt|gck ca @LMJ
Lgvfgtigkjv
Mcljiv
@ttigf`|gck
Cuk xjvj`xfn qgju
Xjvj`xfn x|gfij
Vzmm`xw
Fckfizvgck0:#8#8408 8Tn`xm`fcogkj|gf @f|gck
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Gk|xclzf|gck
Exjjo tn`xm`ock (lxze( `kl ogkj|gocv |c lc
ug|n mc|gck(
G| lj`iv ug|n |nj x`|jv ca mcqjmjk| ca lxze `kl
g|v mj|`hcig|j gk |nj hclw `kl acxfjv `f|gke ck
|nj txcfjvv+
X`|jv ca mcqjmjk| ca lxzev ugii j~ti`gk ug|n |nj
njit ca vzg|`hij M`|njm`|gf`i Mclji+
0:#8#8408 6Tn`xm`fcogkj|gf @f|gck
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Fck|l Fckfjk|x`|gck ca ` lxze gk ti`vm` cx `kw
tnwvgcicegf`i aizgl vzfn `v zxgkj) v`igq`) mgio)
j|f+) gv lj|jxmgkjl ug|n xjvtjf| |c |gmjaciicugke g|v `lmgkgv|x`|gck+
H`vjl ck |nj nwtc|njvgv |n`| |nj `f|gck ca `
lxze xjpzgxjv txjvjkfj ca ` fjx|`gk
fckfjk|x`|gck gk |nj |`xej| |gvvzj+
0:#8#8408
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Chbjf|gqj
Hxgja cqjxqgju |c zkljxv|`kl xje`xlgke
Tn`xm`fcogkj|gf `f|gck
0:#8#8408 :Tn`xm`fcogkj|gf @f|gck
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Ljagkg|gck Tn`xm`fcogkj|gfv gv |nj v|zlw ca un`| |nj
hclw lcjv |c ` lxze+
\nj pz`k|g|`|gqj v|zlw ca |nj @hvcxt|gck)
Lgv|xghz|gck) Mj|`hcigvm `kl J~fxj|gck calxzev `kl |njgx mj|`hcig|jv+
0:#8#8408 1Tn`xm`fcogkj|gf @f|gck
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@hvcxt|gck
G| gv `k `mczk| ca lxze |n`| jk|jxv gk hiccl
`a|jx g|v `lmgkgv|x`|gck gk hclw+
A`f|cx `aajf|gke `hvcxt|gck2
0' K`|zxj ca Lxze
A`|-Vcizhij lxzev `xj m`~gm`iiw `hvcxhjl
U`|jx-Vcizhij lxzev `xj ijvv `hvcxhjl
0:#8#8408 >Tn`xm`fcogkj|gf @f|gck
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Fck|l8' Xcz|j
Cx`i
Vzhigkez`i
Xjf|`i
\x`kvfz|`kjczv
Gkn`i`|gck2 @hvcxt|gck |nxczen mzfczvmjmhx`kjv
\ctgf`i
T`xjk|jx`iiw2
Gk|x`qjkczv2
Gk|x`mzvfzi`x2
Vzhfz|`kjczv2
0:#8#8408 7Tn`xm`fcogkj|gf @f|gck
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0:#8#8408 04
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Lgv|xghz|gck
@k `mczk| ca lxze |n`| xj`fnjv |c fjii) `a|jx
`hvcxt|gck+
@a|jx `hvcxt|gck gk|c |nj vwv|jmgf fgxfzi`|gck)lxzev `xj lgv|xghz|jl |nxczencz| |nj hclw+
Ngeniw tjxazvjl cxe`kv vzfn `v hx`gk) nj`x|v)
izkev) igqjx `kl oglkjwv xjfjgqj mcv| ca |nj lxze
vcck `a|jx gkbjf|gck+
0:#8#8408 00Tn`xm`fcogkj|gf @f|gck
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Txcfjvvjv ca Lgv|xghz|gckG| gkqciqjv |uc v|jtv2
0+ Tjxmj`|gck ca axjj cx zkhczkljl lxze
txjvjk| gk hiccl |nxczen |nj f`tgii`xw u`ii `kl
jk|xw gk|c JFA+
8+ Tjxmj`|gck ca lxze txjvjk| gk JFA|nxczen mjmhx`kj ca |gvvzj fjiiv `kl gk|c |nj
GFA+
0:#8#8408 08Tn`xm`fcogkj|gf @f|gck
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A`f|cxv @aajf|gke Lxze
Lgv|xghz|gck
0+\gvvzj tjxmj`hgig|w+
8+Cxe`k cx |gvvzj vgrj `kl tjxazvgck x`|j+
6+Hgklgke ca lxzev |c |gvvzj fcmtckjk|v+
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Mj|`hcigvm
\nj gxxjqjxvghij |x`kvacxm`|gck ca t`xjk|
fcmtczklv gk|c l`zen|jx mj|`hcig|jv+
@ mjfn`kgvm hw ungfn) mcv|iw igqjx `i|jx
fnjmgf`i v|xzf|zxj ca lxze+
G| hjfcmj kck-|c~gf) u`|jx vcizhij `kl j`vgiw
j~fxj|j cz|vglj hclw |nxczen zxgkj cx a`jfjv
0:#8#8408 0
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Fck|l
Hw |ngv) mcv|iw a`|-vcizhij lxze `xj fckqjx|
gk|c u`|jx-vcizhij ungij u`|jx-vcizhij mcv|iw
xjm`gk zkfn`kejl+
Igqjx f`k lc mj|`hcigvm hw Fckbze`|gck)
Xjlzf|gck) Nwlxc~wi`|gck j|f
0:#8#8408 0:Tn`xm`fcogkj|gf @f|gck
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J~fxj|gck
\nj jigmgk`|gck ca |nj vzhv|`kfjv axcm |nj
hclw+ Gk x`xj f`vjv) vcmj lxzev gxxjqjxvghiw
`ffzmzi`|j gk hclw |gvvzj+
U`|jx vcizhij lxze gv j~fxj|jl cz|vglj mcv|iw
|nxczen zxgkj cx a`jfjv+
0:#8#8408 01Tn`xm`fcogkj|gf @f|gck
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Fck|l
J~fxj|jl lxze m`w fn`kejv fcicx `kl
k`|zxj ca zxgkj cx a`jfjv+
Vcmj lxze `ivc j~fxj|jl |nxczen vuj`|gke)
i`fxwm`|gck) hxj`v| mgio
0:#8#8408 05Tn`xm`fcogkj|gf @f|gck
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Lgvfgtigkj
v
0+ Figkgf`i Tn`xm`fcogkj|gfv
8+ Tctzi`|gck Tn`xm`fcogkj|gfv
6+ \c~gfcogkj|gfv
Tn`xm`fcogkj|gf @f|gck
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Figkgf`i Tn`xm`fcogkj|gfv
Gv |nj `ttigf`|gck ca tn`xm`fcogkj|gf
mj|nclv |c lxze |njx`tw+
G| gkqciqjv ` mzi|glgvfgtigk`xw `ttxc`fn |c
gklgqglz`iiw ct|gmgrjl lcvgke v|x`|jegjv h`vjl
ck |nj t`|gjk|%v lgvj`vj v|`|j `kl t`|gjk|-
vtjfgagf fckvgljx`|gckv+
0:#8#8408 07Tn`xm`fcogkj|gf @f|gck
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Tctzi`|gck Tn`xm`fcogkj|gfv
Zvj gk |nj lxze ljqjictmjk| txcfjvv |c njit
gljk|gaw lgaajxjkfjv gk lxze v`aj|w `kl jaagf`fw
`mcke tctzi`|gck vzhexcztv+
\nj v|zlw ca tn`xm`fcogkj|gf lgaajxjkfjv ca
lxzev gk q`xgczv tctzi`|gck excztv gv |jxmjl
`v tctzi`|gck tn`xm`fcogkj|gfv+
0:#8#8408 84Tn`xm`fcogkj|gf @f|gck
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Fck|l
@ej) ejkljx) ejkj|gf) `kl j|nkgf lgaajxjkfjv
f`k `ivc xjvzi| gk tn`xm`fcogkj|gf lgaajxjkfjv
|n`| m`w `aajf| |nj cz|fcmj ca lxze |njx`tw+
0:#8#8408 80Tn`xm`fcogkj|gf @f|gck
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\c~gfcogkj|gfv
Gv |nj `ttigf`|gck ca tn`xm`fcogkj|gf
txgkfgtijv |c |nj ljvgek) fcklzf|) `kl
gk|jxtxj|`|gck ca lxze v`aj|w jq`iz`|gck
v|zlgjv+
\c~gfcogkj|gfv l`|` `glv gk |nj gk|jxtxj|`|gck ca|c~gfcicegf agklgkev gk `kgm`iv `kl j~|x`tci`|gck
ca |nj xjvzi|gke l`|` |c nzm`kv+
0:#8#8408 88Tn`xm`fcogkj|gf @f|gck
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Figkgf`i\
c~gfcicew
Gv |nj v|zlw ca `lqjxvj jaajf|v ca lxzev `kl
|c~gf vzhv|`kfjv .tcgvckv' gk |nj hclw
0:#8#8408 86Tn`xm`fcogkj|gf @f|gck
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Tn`xm`fcogkj|gf Mcljiv
Q`xgczv m`|njm`|gf`i mcljiv `xj zvjazi gk |nj
ljqjictmjk| ca jpz`|gckv |c ljvfxghj lxze
fckfjk|x`|gckv gk |nj hclw+
Lxze fckfjk|x`|gckv `xj ljtjkljk| ck |gmj)
|nj |uc q`xg`hijv lxze fckfjk|x`|gck `kl |gmj`xj f`iijl ljtjkljk| `kl gkljtjkljk|
q`xg`hijv xjvtjf|gqjiw
0:#8#8408 8
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Fck|lZvjazi gk 2
Fn`x`f|jxgrj |nj hjn`qgcx ca lxze gk t`|gjk|+
Txjlgf|gke fckf+ ca lxze gk q`xgczv hclw aizglv
ug|n lcv`ej xjegmjk+
F`ifzi`|gke ct|gmzm lcv`ej xjegmjk acx
gklgqglz`i t`|gjk|+
Jq`iz`|gke hgcjpzgq`ijkfj hj|ujjk lgaajxjk|acxmzi`|gck+
J~ti`gkgke lxze gk|jx`f|gck+0:#8#8408 Tn`xm`fcogkj|gf @f|gck 8:
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Fck|l
Tn`xm`fcogkj|gf mcljiv `xj lgqgljl gk|c
0+ Fcmt`x|mjk| mcljiv
8+ Tnwvgcicegf`i tn`xm`fcogkj|gf mclji .aicu mclji'
6+ Kck Fcmt`x|mjk|`i Tn`xm`fcogkj|gfv mclji
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Fcmt`x|mjk|`i Mclji
Mcljiv `xj h`vjl ck |nj fckfjt| |n`| |nj hclw
m`w hj qgjujl `v ` vjxgjv ca fcmt`x|mjk|v gk
ungfn |nj lxze gv lgv|xghz|jl+
G| lgqgljl gk|c
0+ Ckj Fcmt`x|mjk| Mcljiv
8+ \uc Fcmt`x|mjk| Mcljiv
0:#8#8408 85Tn`xm`fcogkj|gf @f|gck
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Fck|l
Ckj Fcmt`x|mjk| Mcljiv2
Jk|gxj hclw gv fckvgljxjl `v ckj zkg|
Lxze gv `lmgkgv|jxjl gk|c |nj fcmt`x|mjk|
`kl lgv|xghz|jl |nxczencz| |nj fcmt`x|mjk|.|nj hclw' gkv|`k|`kjczviw
0:#8#8408 8>Tn`xm`fcogkj|gf @f|gck
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0:#8#8408 Tn`xm`fcogkj|gf @f|gck 87
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Fck|l \uc Fcmt`x|mjk| Mcljiv2
Gk |ngv mclji) lxze gv `lmgkgv|jxjl gk|c |njfjk|x`i fcmt`x|mjk| `kl |njk |njxj gv `
|gmj i`e lzj |c vicujx lgv|xghz|gck gk|c
c|njx |gvvzjv `kl cxe`kv+
\njvj c|njx cxe`kv `xj xjtxjvjk|jl hw |nj
tjxgtnjx`i fcmt`x|mjk|
0:#8#8408 64Tn`xm`fcogkj|gf @f|gck
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Tnwvgcicegf`i Mcljiv
@k `i|jxk`|j mj|ncl ca hzgilgke ` tn`xm`fcogkj|gf
txcagij ca ` lxze gk |nj hclw gv |c z|gigrj `k`|cmgf
`kl tnwvgcicegf`i gkacxm`|gck+ G| ljfglj unj|njx lxze lgv|xghz|gck gk|c ` t`x|gfzi`x
|gvvzj gv hw tjxazvgck x`|j cx mjmhx`kj |x`kvtcx|+
\nj c|njx t`x`mj|jxv igoj qjkczv lxze
fckfjk|x`|gck `kl |nj t`x|g|gck fcjaagfgjk|
0:#8#8408 60Tn`xm`fcogkj|gf @f|gck
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Kckfcmt`x|mjk|`i
G| gv ngeniw ljtjkljk| ck jv|gm`|gck ca |c|`i
lxze j~tcvzxj+
\c|`i lxze j~tcvzxj gv mcv| ca|jk jv|gm`|jlhw `xj` zkljx |nj fzxqj .@ZF' mj|nclv+
0:#8#8408 68Tn`xm`fcogkj|gf @f|gck
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Kckigkj`x Mclji
Fckfjt| ca igkj`x Tn`xm`fcogkj|gfv gv |nj
fckfjk|x`|gckv `fngjqjl `xj txctcx|gck`i |c
|nj lcvj egqjk+
Acx j~`mtij) ` lczhigke ca |nj lcvj ugiitxclzfj ` lczhigke ca |nj hiccl
fckfjk|x`|gck+0:#8#8408 66Tn`xm`fcogkj|gf @f|gck
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Fck|l
Acx vcmj lxzev `k gkfxj`vj gk lcvj m`w
txclzfj ` fckfjk|x`|gck mzfn exj`|jx |n`k
j~tjf|jl+ Acx j~`mtij) gkfxj`vjv gk lcv`ej ca |nj
`k|gjtgijt|gf `ejk| Tnjkw|cgk `hcqj
`ttxc~gm`|jiw 644 me l`giw zvz`iiw txclzfj `exj`|jx |n`k j~tjf|jl gkfxj`vj gk hiccl
fckfjk|x`|gckv+0:#8#8408 6
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\njcxj|gf`i ljtgf|gck ca ti`vm` fckfjk|x`|gckv aciicugke jg|njx `k gk|x`qjkczv hcizv lcvj
gmmjlg`|jiw aciicujl hw gkg|g`|gck ca ` fck|gkzczv gk|x`qjkczv gkazvgck cx gkg|g`|gck ca` fck|gkzczv gk|x`qjkczv gkazvgck ckiw+
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@ttigf`|gckv
\c zkljxv|`kl txcfjvv ca @LMJ `a|jx
`lmgkgv|x`|gck ca lxze) ungfn `aajf|v ckvj| `kl
gk|jkvg|w ca hgcicegf`i xjvtckvj+
Gk ljvgek `kl z|gigr`|gck ca gk-qg|xc mclji vwv|jm
|n`| f`k jq`iz`|j lgvvciz|gck fn`x`f|jxgv|gfv ca
kju fcmtczkl acxmzi`|jl `v kju lxze
acxmzi`|gckv `kl jv|`higvn mj`kgkeazi gk-qgqc gk-
qg|xc fcxxji`|gckvngt+
0:#8#840861
Tn`xm`fcogkj|gf @f|gck
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Fck|l
\c f`xxw cz| hgc`q`gi`hgig|w `kl hgcjpzgq`ijkfj
v|zlgjv+
Gk ljvgek `kl ljqjictmjk| ca kju lxze `kl |njgx
`ttxctxg`|j lcv`ej xjegmjk+
Tn`xm`fcogkj|gf txgkfgtijv f`k zvjl gk |nj
ljqjictmjk| mgfxc vtnjxjv `kl K`kct`x|gfijv+
0:#8#8408 65Tn`xm`fcogkj|gf @f|gck
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Cuk Xjvj`xfn Qgju
TO `f|gck acx |nj @wzxqjlgf lxzev f`k hj lj|jf| hw
t`x`mj|jxv igoj X`v`) Ezk`) @qv|n` T`o`) Qgt`o`
.Kgv|n` T`o`'+
X`v` gv gljk|gagjl unjk lxze fcmj gk fck|`f| ug|n
|ckezj ungfn gv `a|jx @hvcxt|gck+
Ezk` gv gljk|gagjl hw x`|j caLgv|xghz|gck gk hclw
0:#8#8408 6>Tn`xm`fcogkj|gf @f|gck
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Fck|l
Qgt`o` .@q`v|n` T`o`' ca lxze lj|jxmgkj hw
Mj|`hcigvm gk vwv|jmgf fgxfzi`|gck+
\nj J~fxj|gck ca lxze |nxczen hclw gv ckj ca |nj
fxg|jxg` `vvjv |c Qgt`o` .Kgv|n` T`o`'+
Qgxw` ! Tx`hn`q` f`k lj|jxmgkj hw Tn`xm`fc
Lwk`mgfv ca lxze+
0:#8#8408 Tn`xm`fcogkj|gf @f|gck 67
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Xjvj`xfn @x|gfij
Tn`xm`fcogkj|gfv ca Ngen-Lcvj Cx`i \ng`mgkj
Nwlxcfnicxglj Gk Nj`i|nw Vzhbjf|v+
Ncu`xl @ Vmg|nigkj) Mgfn`ji Lckkgkc) L`qgl B+ Exjjkhi`||
Fckfizvgck
G| vncuv |n`| ngen hiccl ijqjiv ca |ng`mgkj f`k hj
`fngjqjl x`tgliw ug|n cx`i |ng`mgkj nwlxcfnicxglj+
\ng`mgkj gv `hvcxhjl hw hc|n `k `f|gqj `kl kck-
v`|zx`hij t`vvgqj txcfjvv+
0:#8#8408
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Vzmm`xw
Ljagkg|gck ca TO
Ljvfxgt|gck ca @LMJ
Lgvfgtigkjv igoj Tctzi`|gck TO) Figkgf`i TO j|f+
M`|njm`|gf`i Mcljiv- fcmt`x|mjk| mclji)
Tnwvgcicegf`i mclji j|f+
@ttigf`|gck ca TO
0:#8#8408 Tn`xm`fcogkj|gf @f|gck
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Fckfizvgck
G| j~ti`gk |nj |c|`i fij`x`kfj ca lxze `kl g|v
v|j`lw v|`|j ti`vm` fckfjk|x`|gck lzxgke
fck|gkzjv `lmgkgv|x`|gck+
G| qjxw zvjazi gk lxze ljqjictmjk| `kl lcvj
ag~`|gck+ Uj mzv| |ngko `hcz| `ttigf`|gck ca TO acx
@wzxqjlgf lxzev+0:#8#8408
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Xjajxjkfjv X`ke `kl L`ijv Tn`xm`fcicew
\j~| Hcco ca Tn`xm`fcicew \xgt`|ng
\j~| Hcco ca Tn`xm`fcicew V`|cvo`x
H`vgf Tn`xm`fcogkj|gfv Vzkgi B`mhnjo`x !
Tngigt Hxjjk
n||t2##uuu+hgcmjlfjk|x`i+fcm#0
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0:#8#8408
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