ligand p-gp inhibition (11-me-leu)-cyclosporin a 1...clanobutin 0 clebopride 0 clemastine 1...

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ligand P-gp inhibition (11-Me-Leu)-Cyclosporin A 1 1,2,3,4-Tetrahydro-1-methyl-6,7-isoquinolinediol 0 1,2,3,4-Tetrahydro-6,7-dimethoxy-isoquinoline 0 1,2,3,4-Tetrahydro-isoquinoline 0 1,3,5-Triazacycloheptane 4b 1 1,3,5-Triazacycloheptane 4c 1 1,3,5-Triazacycloheptane 5b 1 1,3,5-Triazacycloheptane 5c 1 1,3,5-Triazacycloheptane 5d 1 1,3,5-Triazacycloheptane 6b 1 1,3,5-Triazacycloheptane 6c 1 1-(3-methoxyphenyl)-N,N-dimethylmethanamine 0 1-(4-chlorbenzhydryl)piperazine 0 1-Benzyl-3-pyrroline 0 1-Benzylimidazole 0 1-Phenethylpiperidine 0 1-Phenylpiperazine 0 11-Deoxycortisol 1 14-Benzoylyohimbine 1 16-Dehydroprogesterone 1 16-Methylprogesterone 1 17-Hydroxypregnenolone 0 17-Hydroxyprogesterone 1 2,2'-Diphenylethylamine 0 2,4,6,8-Tetradiethano 0 2,4,6,8-Tetramopholin 0 2,4,6,8-Tetrapiperidy 0 2,4,6-Trimorpholinepy 0 2,4,8-Trimorpholinepy 0 2-Benzylpyridine 0 2-Chloro-10-[2-(dimethylamino)ethyl] phenothiazine 1 2-Chloro-10-[4-(dimethylamino)butyl] phenothiazine 1 2-Chloroimipramine 1 2-Oxazolidinone 0 3'-4'-Dichlorobenzamil 0 3,8-Dihydroxychlorpromazine 0 3-Methyl choroquine 1 4,8-Dipiperidyl-2,6-D 0 4,8-Dipiperidyl-2,6-M 0 4,8-Dipiperidyl-Dimet 0 4-(2-Dimethylamino)ethyl)morpholine 0 4-Androstene-3,17-dione 1 4-Hydroxytamoxifen 1 4-Hydroxytoremifene 1 4-Iodotamoxifen 1 4-beta-Phorbol 12,13-dibutyrate 1 4-beta-Phorbol 13-acetate 0 4-beta-Phorbol 13-butyrate 0 5-(N,N-hexamethylene)amiloride 0

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  • ligand P-gp inhibition

    (11-Me-Leu)-Cyclosporin A 1

    1,2,3,4-Tetrahydro-1-methyl-6,7-isoquinolinediol 0

    1,2,3,4-Tetrahydro-6,7-dimethoxy-isoquinoline 0

    1,2,3,4-Tetrahydro-isoquinoline 0

    1,3,5-Triazacycloheptane 4b 1

    1,3,5-Triazacycloheptane 4c 1

    1,3,5-Triazacycloheptane 5b 1

    1,3,5-Triazacycloheptane 5c 1

    1,3,5-Triazacycloheptane 5d 1

    1,3,5-Triazacycloheptane 6b 1

    1,3,5-Triazacycloheptane 6c 1

    1-(3-methoxyphenyl)-N,N-dimethylmethanamine 0

    1-(4-chlorbenzhydryl)piperazine 0

    1-Benzyl-3-pyrroline 0

    1-Benzylimidazole 0

    1-Phenethylpiperidine 0

    1-Phenylpiperazine 0

    11-Deoxycortisol 1

    14-Benzoylyohimbine 1

    16-Dehydroprogesterone 1

    16-Methylprogesterone 1

    17-Hydroxypregnenolone 0

    17-Hydroxyprogesterone 1

    2,2'-Diphenylethylamine 0

    2,4,6,8-Tetradiethano 0

    2,4,6,8-Tetramopholin 0

    2,4,6,8-Tetrapiperidy 0

    2,4,6-Trimorpholinepy 0

    2,4,8-Trimorpholinepy 0

    2-Benzylpyridine 0

    2-Chloro-10-[2-(dimethylamino)ethyl] phenothiazine 1

    2-Chloro-10-[4-(dimethylamino)butyl] phenothiazine 1

    2-Chloroimipramine 1

    2-Oxazolidinone 0

    3'-4'-Dichlorobenzamil 0

    3,8-Dihydroxychlorpromazine 0

    3-Methyl choroquine 1

    4,8-Dipiperidyl-2,6-D 0

    4,8-Dipiperidyl-2,6-M 0

    4,8-Dipiperidyl-Dimet 0

    4-(2-Dimethylamino)ethyl)morpholine 0

    4-Androstene-3,17-dione 1

    4-Hydroxytamoxifen 1

    4-Hydroxytoremifene 1

    4-Iodotamoxifen 1

    4-beta-Phorbol 12,13-dibutyrate 1

    4-beta-Phorbol 13-acetate 0

    4-beta-Phorbol 13-butyrate 0

    5-(N,N-hexamethylene)amiloride 0

  • 5-(N-Methyl-N-isobutyl)amiloride 0

    5-N-acetyl-8-demethylardeemin 1

    5-N-acetylardeemin 1

    5-[N-Methyl-N-(tert-butyl)]-amiloride 0

    6-Phenyl-2,4,7-pterid 0

    7,8-Dihydroxychlorpromazine 0

    7-Hydroxychlorpromazine 0

    AF-1393 1

    AG-1112 0

    AG-213 0

    AG-690 1

    AHC-52 1

    AHR 06601 1

    AHR 16462 1

    AHR-16303 1

    AN-989 1

    AY 9944 1

    Acapriazine 0

    Acebutolol 0

    Acecainide 0

    Acepromazine 1

    Aceprometazine 1

    Acetophenazine 1

    Acridine 0

    Acridone-4-carboxamide 22 1

    Acridone-4-carboxamide 23 1

    Acridone-4-carboxamide 24 1

    Acridone-4-carboxamide 28 1

    Acridone-4-carboxamide 29 1

    Acridone-4-carboxamide 30 1

    Acridone-4-carboxamide 31 1

    Acridone-4-carboxamide 32 1

    Acridone-4-carboxamide 36 1

    Acridone-4-carboxamide 39 1

    Acridone-4-carboxamide 43 1

    Acridone-4-carboxamide 44 1

    Acridone-4-carboxamide 47 1

    Acridone-4-carboxamide 48 1

    Acridone-4-carboxamide 49 1

    Acridone-4-carboxamide 50 1

    Acridone-4-carboxamide 51 1

    Acridone-4-carboxamide 52 1

    Acridone-4-carboxamide 53 1

    Acridone-4-carboxamide 54 1

    Acridone-4-carboxamide 55 1

    Acridone-4-carboxamide 59 1

    Acridone-4-carboxamide 60 1

    Acridone-4-carboxamide 61 1

    Acridone-4-carboxamide 64 1

    Acridone-4-carboxamide 65 1

  • Acridone-4-carboxamide 66 1

    Acridone-4-carboxamide 67 1

    Acridone-4-carboxamide 68 1

    Acridone-4-carboxamide 69 1

    Acridone-4-carboxamide 70 1

    Acridone-4-carboxamide 71 1

    Acridone-4-carboxamide 72 1

    Acridone-4-carboxamide 73 1

    Acridone-4-carboxamide 74 1

    Acridone-4-carboxamide 75 1

    Acridone-4-carboxamide 76 1

    Acridone-4-carboxamide 77 1

    Acridone-4-carboxamide 78 1

    Acridone-4-carboxamide 79 1

    Acridone-4-carboxamide 80 1

    Acridone-4-carboxamide 81 1

    Acridone-4-carboxamide 82 1

    Acridone-4-carboxamide 83 1

    Acridone-4-carboxamide 85 1

    Acrivastine 0

    Actinomycin D 0

    Adiphenine 0

    Aldicarb 0

    Aldoxycarb 0

    Aldrich 21430-2 1

    Almitrine 1

    Alpertine 1

    Alpha-Tocopherol 0

    Alprenolol 1

    Alverine

    Amantadine 0

    Ambodryl 0

    Amiloride 0

    Aminocarb 0

    Aminopentamide 0

    Amiodarone 1

    Amitriptyline 1

    Amlodipine 1

    Amodiaquin 0

    Amotriphene 1

    Amoxapine 1

    Amoxecaine 0

    Amperozide 1

    Amphotericin B 0

    Amprenavir 1

    Androstenedione 1

    Androsterone 1

    Antazoline 0

    Antenolol 0

    Antipyrine 0

  • Apomorphine 0

    Aprindine 1

    Ascorbic acid 0

    Asocainol 1

    Astemizole 1

    Atorvastatin (methyl ester) 1

    Atorvastatin lactone 1

    Atrazine 0

    Atropine 0

    Aureobasidin A (ABA) 1

    Azaclorazine 1

    Azaconazole 0

    Azaperone 0

    Azelastine 1

    Azidopine 1

    Azidoprocainamide methoiodide 0

    Azipramine 1

    B3-243 1

    B669 1

    B9109-012 1

    BIBW 22 1

    BW 1019W91 1

    BW 1136U89 1

    BW 1288U89 1

    BW 1351W91 1

    BW 1379W91 1

    BW 565C81 1

    Bamipine 0

    Barnidipine 1

    Befuraline 0

    Benactyzine 0

    Bencyclane 0

    Benidipine 1

    Benzathine 1

    Benzmalecene 0

    Benzofuran derivative 2a 0

    Benzofuran derivative 2c 1

    Benzofuran derivative 2d 1

    Benzofuran derivative 2e 1

    Benzofuran derivative 2f 1

    Benzquinamide 0

    Benztropine 1

    Bepridil 1

    Berberine 0

    Bevantolol 1

    Bifonazole 1

    Biperiden 0

    Biphenamine 0

    Biricodar 1

    Bisobrin 0

  • Bleomycin A2 0

    Boldine 0

    Boxidine 0

    Bromocriptine 1

    Brompheniramine 0

    Bryostatin 0

    Bucainide 1

    Buclizine 1

    Budipine

    Buflomedil 0

    Bufuralol 1

    Bunaftine 1

    Buspirone 1

    Butalamine 0

    Butaperazine 1

    Buterizine 1

    Butethamate 0

    CP-100356 1

    CP-101556 1

    CP-114416 1

    CP-114769 1

    CP-117227 1

    CP-12379 1

    CP-141938 1

    CP-147478 1

    CP-69042 1

    Calcimycin 0

    Calphostin C 1

    Captodiame

    Carbamazepine 0

    Carbaryl 0

    Carbinoxamine 1

    Carbiphene 1

    Carnitine 0

    Caroverine 1

    Carphenazine 1

    Carvedilol 1

    Carvedilol metabolite M2 0

    Carvedilol metabolite M4 0

    Carvedilol metabolite M5 0

    Catharanthine 1

    Cefoperazone 0

    Cefotetan 0

    Ceftazidime 0

    Celiprolol 0

    Cepharanthine 1

    Cephradine 0

    Cetiedil 1

    Cetrizine 0

    Chelerythrine 0

  • Chlophedianol 0

    Chloracyzine 1

    Chlorbenzoxamine 1

    Chlorcyclizine 0

    Chlorogenic acid 0

    Chloropyramine 0

    Chloroquine 0

    Chlorpheniramine 0

    Chlorphenoxamine

    Chlorproethazine 1

    Chlorpromazine 1

    Chlorprothixene 1

    Chlorzoxazone 0

    Chromonar

    Cimetidine 0

    Cinchonidine 1

    Cinepaxadil 1

    Cinepazet 0

    Cinepazic acid 0

    Cinepazide 0

    Cinnarizine 1

    Cinprazole 1

    Cinpropazide 0

    Cintriamide 0

    Cinuperone 1

    Ciprofloxacin 0

    Citalopram 0

    Citatepine 1

    Citenamide 0

    Clamoxyquin 0

    Clanobutin 0

    Clebopride 0

    Clemastine 1

    Clemizole 1

    Cletoquine 0

    Clobutinol 0

    Clocinizine 1

    Clomestrone 0

    Clomiphene 0

    Clomipramine 1

    Clonidine 0

    Clopenthixol 1

    Cloperastine 1

    Clopimozide 1

    Clopipazan 1

    Clothiapine 1

    Clothixamide 1

    Clotrimazole 1

    Colchicine 0

    Colforsin 1

  • Coralyne 0

    Corticosterone 0

    Cortisone 0

    Corynanthine 1

    Coumaphos 1

    Cryptophycin 1

    Cyclobenzaprine 1

    Cyclofenazine 1

    Cyclopeptolide(1) 0

    Cyclopeptolide(11) 0

    Cyclopeptolide(12a) 1

    Cyclopeptolide(12b) 1

    Cyclopeptolide(15a) 1

    Cyclopeptolide(15b) 1

    Cyclopeptolide(16a) 1

    Cyclopeptolide(16c) 1

    Cyclopeptolide(16h) 1

    Cyclopeptolide(18) 1

    Cyclopeptolide(19) 0

    Cyclopeptolide(2a) 1

    Cyclopeptolide(2c) 1

    Cyclopeptolide(2f) 1

    Cyclopeptolide(3a) 1

    Cyclopeptolide(3c) 1

    Cyclopeptolide(3f) 1

    Cyclopeptolide(3g) 1

    Cyclopeptolide(3h) 1

    Cyclopeptolide(3i) 1

    Cyclopeptolide(3j) 1

    Cyclopeptolide(3l) 1

    Cyclopeptolide(3n) 1

    Cyclopeptolide(4) 1

    Cyclopeptolide(7) 1

    Cyclopeptolide(8) 1

    Cyclopeptolide(9) 1

    Cyclophenazine 1

    Cyclosporin A 1

    Cyclosporin C 1

    Cyclosporin G 1

    Cypermethrin 1

    Cyproheptadine 1

    Cytochalasin A 0

    Cytochalasin C 0

    Cytochalasin D 0

    Cytochalasin E 1

    Cytochalasin H 0

    Cytochalasin J 0

    D490 1

    D525 1

    D528 0

  • D557 1

    D559 1

    D595 1

    D784 1

    D894 1

    DDE 0

    DDT 0

    DHP-014 1

    DMDP 1

    DPDPE 0

    Dagapamil 1

    Danitracen 0

    Dapiprazole 0

    Darodipine 1

    Debrisoquin 0

    Dehydroemetine 0

    Delavirdine 1

    Delfantrine 0

    Deltorphin II 0

    Denzimol 0

    Deoxycorticosterone 1

    Desethylamiodarone 1

    Desipramine 1

    Desmethoxyyangonin 1

    Desmethylazelastine 1

    Desmethylchlorpromazine 0

    Desmethylcitalopram 0

    Desmethylsertraline 1

    Devapamil 1

    Dexamethasone 0

    Dexniguldipine 1

    Dialifos 0

    Dibenzylamine 0

    Dibozan 0

    Dibucaine 1

    Dicapthon 1

    Diclofensine 0

    Didesmethylchlorpromzine 0

    Diethylaniline 0

    Diethylstilbestrol 1

    Difloxacin 0

    Difluanine 1

    Digoxin 0

    Dihydroergotamine 0

    Dihydromethysticin 1

    Dihydropyridine DP11 1

    Dihydropyridine DP5 1

    Dihydropyridine DP6 1

    Dihydropyridine DP7 1

    Dihydropyridine DP9 1

  • Dihydropyrroloquinoline series 14 0

    Dihydropyrroloquinoline series 27 1

    Diisopromine

    Dilazep 1

    Diltiazem 1

    Dimethindene 1

    Diosmetin 0

    Diosmin 0

    Diphenamid 0

    Diphenazoline 0

    Diphenidol 1

    Diphenylpyraline 1

    Disopyramide 0

    Dixyrazine 1

    Dobutamine 0

    Doconazole 1

    Domperidone 0

    Doxapram 1

    Doxazosin

    Doxepine 1

    Doxorubicin 0

    Doxylamine 0

    Drobuline 1

    Drofenine 0

    Droloxifen 0

    Droprenilamine 1

    Droproizine 0

    Duoperone 1

    EKI-785 1

    Ebastine 1

    Econazole 0

    Efonidipine 1

    Eletriptan 0

    Eltoprazine 0

    Emepronium 0

    Emetine 0

    Emopamil 1

    Enciprazine 1

    Endosulfan 1

    Enilconazole 0

    Enoxacin 0

    Epinephrine 0

    Eprazinone 1

    Eprozinol 1

    Equilenine 0

    Equilin 0

    Ergocristine 1

    Ergocryptine 1

    Ergonovine 0

    Ergotamine 1

  • Erythromycin 1

    Estradiol 0

    Estriol 0

    Estrone 0

    Etafenone 1

    Ethylbenztropine 1

    Ethylbenzylaniline 0

    Etifelmin 0

    Etodroxizine

    Etolotifene 1

    Etomidoline 1

    Etoposide 0

    Euphodendroidin A 1

    Euphodendroidin B 1

    Euphodendroidin C 1

    Euphodendroidin D 1

    Euphodendroidin E 1

    Euphodendroidin G 1

    Euphodendroidin H 1

    Euphodendroidin I 1

    Euprocin 1

    Falipamil 0

    Famciclovir 0

    Farnesyl analog AFCA 1

    Farnesyl analog AFCMA 1

    Farnesyl analog AFCME 1

    Febuverine 1

    Felodipine 1

    Fenbutrazate 1

    Fendiline 1

    Fenoctimine 0

    Fenoterol 0

    Fenoxedil 1

    Fenpipramide 0

    Fenpiverinium 0

    Fenticonazole 1

    Fenvalerate 0

    Fexofenadine 0

    Filipin 0

    Fisetin 0

    Flavonoid ID 13 1

    Flavonoid ID 21 0

    Flavonoid ID 22 0

    Flavonoid ID 23 0

    Flavonoid ID 24 0

    Flavonoid ID 37 1

    Flavonoid ID 38 0

    Fleroxacin 0

    Flesinoxan 0

    Flezelastine 1

  • Flordipine 1

    Fluanisone 1

    Fluazifop-butyl 0

    Fluconazole 0

    Flumazenil 0

    Flunarizine 1

    Fluoxetine 1

    Fluperamide 1

    Fluperlapine 1

    Fluphenazine 1

    Flurazepam 1

    Fluspirilene 1

    Fluvoxamine 1

    GF120918 1

    GGCME 1

    GW 420867 1

    Gallopamil 1

    Gamfexine 0

    Geldanamycin 1

    Geldanamycin 17-AAG 1

    Gepirone 0

    Ginsenoside Rg3 1

    Ginsenoside Rh2 1

    Glaucine 1

    Gramine 0

    Guanabenz 0

    Guanfacine 0

    H-7 0

    H-89 1

    HA-1004 0

    HDL-2722 0

    Halopemide 1

    Haloperidol 1

    Hepzidine 1

    Hexadiline 0

    Hexobendine 1

    Hexoprenaline 0

    Histapyrrodine 0

    Hoechst 33342 0

    Homochlorocyclizine 0

    Homofenazine

    Homoveratrylamine 0

    Hoquizil 0

    Hydramethylnon 1

    Hydrastine 0

    Hydrocotarnine 0

    Hydromorphone 0

    Hydroxyzine 1

    Hyperforin 0

    Idarubicin 1

  • Imatinib 1

    Imiclopazine 0

    Imipramine 1

    Imolamine 0

    Imoxiterol 0

    Indinavir 0

    Indomethacin 0

    Isoconazole 1

    Isoniazid 0

    Isopromethazine 1

    Isoxsuprine 0

    Isradipine 1

    Itraconazole

    Ivermectin Bla 1

    Jatrophane diterpene(7) 1

    Jatrophane diterpenoid(1) 1

    Jatrophane diterpenoid(10) 1

    Jatrophane diterpenoid(11) 1

    Jatrophane diterpenoid(12) 1

    Jatrophane diterpenoid(13) 1

    Jatrophane diterpenoid(14) 1

    Jatrophane diterpenoid(15) 1

    Jatrophane diterpenoid(16) 1

    Jatrophane diterpenoid(2) 1

    Jatrophane diterpenoid(3) 1

    Jatrophane diterpenoid(5) 1

    Jatrophane diterpenoid(6) 1

    Jatrophane diterpenoid(8) 1

    Jatrophane diterpenoid(9) 1

    K02 1

    Keoxifene 0

    Ketamine 0

    Ketoconazole 1

    Ketotifen 1

    LR 764 0

    LU43918 1

    LU46324 1

    LU47474 1

    LU48895 1

    LU49667 1

    LU49940 1

    LU51903 1

    LY18947 0

    LY292540 1

    LY296097 1

    LY335979 1

    LY335983 1

    LY350344 1

    Labetalol 0

    Laudanosine 1

  • Laudanosoline 0

    Lenperone 1

    Levodopa 0

    Levophacetoperane 0

    Lidocaine 0

    Lidoflazine 1

    Linadryl 1

    Lindane 0

    Lobeline 1

    Lombazole

    Loperamide 1

    Lopinavir 1

    Loratadine 1

    Lorcainide 1

    Losartan 0

    Lovastatin acid 0

    Lovastatin lactone 1

    Loxapine 1

    Luteolin 0

    Luteolin-4'-O-glucoside 0

    MA 1499 1

    MA 1509 1

    MA 1510 1

    MA 1586 1

    MA 1588 1

    MA 1598 1

    MA 1813 1

    MA 1862 0

    MA 1865 0

    MA 1880 0

    MDL 6792

    MDL-10393

    MDL8917V 1

    MDR reversal agent 15h 1

    MDR reversal agent 15i 1

    MDR reversal agent 15m 1

    MDR reversal agent 15o 1

    MDR reversal agent 15u 1

    MDR reversal agent 15x 1

    MDR reversal agent 28a 1

    MDR reversal agent 28c 1

    MDR reversal agent 35a 1

    MDR reversal agent 35d 1

    MDR reversal agent 37b 1

    MER37 1

    MK-571 0

    MM36 1

    MS-209 1

    Macbecin II 1

    Manidipine 1

  • Mannitol 0

    Maprotiline 1

    Maroxepine 0

    Mebendazole 1

    Mebeverine 1

    Meclizine 1

    Mecloxamine 0

    Medroxyprogesterone 1

    Medroxyprogesterone acetate 1

    Mefloquine 1

    Megestrol Acetate 1

    Meglitinide 0

    Memotine 0

    Mephentermine 0

    Mephenytoin 0

    Mepramidil 1

    Meprobamate 0

    Mequitazine 1

    Mesoridazine 1

    Mesuprine 0

    Metergoline 1

    Methadone 1

    Methaphenilene 0

    Methdilazine 0

    Methixene 0

    Methomyl 0

    Methotrimeprazine 1

    Methoxychlor 0

    Methoxypromazine

    Methyl Cellosolve Acetate 0

    Methylamine 0

    Methysergide 0

    Methysticin 1

    Metiapine 1

    Metoclopramide 0

    Metofenazate 1

    Metopimazine 0

    Metoprolol 0

    Metoserpate 1

    Metoxepin 1

    Mevinphos 0

    Mexilitene 0

    Mezilamine 0

    Mianserin 0

    Mibefradil 1

    Miconazole 0

    Midazolam 1

    Mifepristone (RU486) 1

    Milenperone 1

    Milipertine 1

  • Mioflazine 1

    Mirex 0

    Mitomycin C 0

    Mitoxantrone 0

    Mixidine 0

    Moclobemide 0

    Monensin 1

    Mopidamol 0

    Morin 0

    Morphine 0

    Motracetam 0

    Moxapridine 1

    N,N'-Diphenyl-p-phenylenediamine 0

    N,N'-dibenzylethylene diamine 0

    N,N-Bis(alkanol)amine aryl ester analog 21 1

    N,N-Bis(alkanol)amine aryl ester analog 5 0

    N,N-Bis(alkanol)amine aryl ester analog 6 1

    N,N-Bis(alkanol)amine aryl ester analog 8 1

    N,N-Bis(alkanol)amine aryl ester analog 9 1

    N,N-Dimethylbenzylamine 0

    N,N-bis(cyclohexanol)amine aryl ester (3) 1

    N,N-bis(cyclohexanol)amine aryl ester (4) 1

    N,N-bis-arylalkylamine derivative(1) 1

    N,N-bis-arylalkylamine derivative(2) 1

    N,N-diethylcyclohexylamine 0

    N-Benzylbenzamide 0

    N-Methyl-gallopamil 0

    N-Norlaudanosine 1

    N-Norlaudanosoline 0

    N-Phenyl-1-naphthylamine 0

    N-Phenyl-2-naphthylamine 0

    N-acetyl-daunorubicin 1

    N-acyloxy-1,4-dihydropyridine(10) 1

    N-acyloxy-1,4-dihydropyridine(5) 1

    N-acyloxy-1,4-dihydropyridine(6) 1

    N-acyloxy-1,4-dihydropyridine(7) 1

    N-acyloxy-1,4-dihydropyridine(8) 1

    N-acyloxy-1,4-dihydropyridine(9) 1

    N-desmethyl-toremifene 1

    N-desmethyl-venlafaxine 1

    N-desmethyltamoxifen 1

    N-trialkylglycine N31214C 1

    NK-101 0

    NK-106 1

    NSC 102843 1

    NSC 169647 0

    NSC 220202 1

    NSC 303594 1

    NSC 30774 1

    NSC 33128 1

  • NSC 344003 1

    NSC 359449 0

    NSC 633043 0

    NSC 633320 0

    NSC 640085 0

    NSC 648114 1

    NSC 649087 1

    NSC 665333 1

    NSC 666490 0

    NSC 667739 1

    NSC 668360 1

    NSC 673413 0

    NSC 676590 1

    NSC 676591 1

    NSC 676600 1

    NSC 676605 1

    NSC 88116 0

    NSC 88657 0

    NSC 94907 0

    Nafcillin 0

    Nafiverine 1

    Nafoxidine 1

    Naftifine 0

    Naftopidil 1

    Naftoxate 1

    Nalbuphine 0

    Naloxone 0

    Naltrexone 0

    Naltrindole 0

    Nefazodone 1

    Nelfinavir 1

    Neostigmine 0

    Nicardipine 1

    Nicergoline 1

    Nifedipine 1

    Nilprazole 1

    Niludipine 1

    Nimodipine 1

    Nisoldipine 1

    Nitrazepam 0

    Nitrendipine 1

    Nitromifene 1

    Nobiletin 1

    Nomifensine 0

    Nordazepam 0

    Norfloxacin 0

    Norfluxetine 1

    Norgallopamil 1

    Nortriptylene 1

    Norverapamil 1

  • Noscapine 1

    Nuclotixene 0

    Nylidrin 0

    O-desmethyl-venlafaxine 0

    OBF-1622 0

    OBF-1822 1

    OBF-1834 0

    OC144-093 1

    OL-57 1

    Ofloxacin 0

    Oleanolic acid 0

    Olivomycin A 0

    Omeprazole 1

    Omeprazole sulfone 0

    Omoconazole 0

    Opipramol 0

    Opromazine 1

    Orconazole

    Oxamarin 0

    Oxatomide 1

    Oxiconazole 0

    Oxolinic acid 0

    Oxprenolol 0

    Oxybutynin 1

    Oxyfedrine 0

    Oxypendyl 0

    Oxyperomide 0

    Oxypertine 1

    PAK-1 1

    PAK-200 1

    PAK-8 0

    PGP-4008 1

    Palmitoylcartinine 0

    Papaverine 0

    Paraquat 0

    Parathion-methyl 1

    Parconazole 0

    Paroxetine 1

    Pefloxacin 0

    Penfluridol 1

    Pentachlorophenol 0

    Pentazocine 1

    Peptoid 1 1

    Peptoid 2 1

    Peradoxime 1

    Perafensine 0

    Perazine

    Perhexilline 0

    Perimetazine 1

    Perlapine 1

  • Perphenazine 1

    Phenethylamine 0

    Pheniramine 0

    Phenoxazine ID 11 1

    Phenoxazine ID 12 1

    Phenoxazine ID 15 0

    Phenoxazine ID 18 1

    Phenoxazine ID 2 1

    Phenoxazine ID 3 1

    Phenoxazine ID 4 1

    Phenoxazine ID 5 1

    Phenylamil 1

    Phenyltoloxamine 0

    Phenytoin 0

    Phorbol 0

    Phosmet 0

    Physostigmine 1

    Pifarnine 1

    Piflutixol 1

    Pimethixene 1

    Pimozide 1

    Pinafide 0

    Pinoxepine 1

    Pipamperone 1

    Pipemidic Acid 0

    Piperacetazine

    Piperamide 0

    Piperdimerine A 1

    Piperine 1

    Pipoxizine 1

    Pipoxolan 0

    Pirenzepine 0

    Pirohenptine 1

    Piromidic Acid 0

    Pirprofen 0

    Pizotyline 1

    Pramiverin 0

    Pravastatin 0

    Prazosin 1

    Predifine 1

    Pregnanedione 1

    Prenoverine 0

    Prenoxidiazine 1

    Prenylamine 1

    Primaquine 0

    Primidolol 0

    Prinixic acid 0

    Pristinamycin IA 1

    Proadifen 1

    Prochlorperazine 1

  • Procyclidine 1

    Prodipine

    Progabide 1

    Progesterone 1

    Promazine 0

    Promethazine 1

    Propafenone 1

    Propafenone derivative 1b 1

    Propafenone derivative 1c 1

    Propafenone derivative 1e 1

    Propafenone derivative 1f 1

    Propafenone derivative 1g 1

    Propafenone derivative 1i 1

    Propafenone derivative 1k 1

    Propafenone derivative GP01 1

    Propafenone derivative GP02 1

    Propafenone derivative GP03 0

    Propafenone derivative GP05 1

    Propafenone derivative GP07 0

    Propafenone derivative GP10 0

    Propafenone derivative GP134 1

    Propafenone derivative GP155 1

    Propafenone derivative GP159 1

    Propafenone derivative GP163 1

    Propafenone derivative GP164 1

    Propafenone derivative GP17 0

    Propafenone derivative GP240 1

    Propafenone derivative GP29 1

    Propafenone derivative GP31 1

    Propafenone derivative GP339 1

    Propafenone derivative GP358 1

    Propafenone derivative GP359 1

    Propafenone derivative GP360 1

    Propafenone derivative GP366 1

    Propafenone derivative GP381 1

    Propafenone derivative GP388 1

    Propafenone derivative GP389 0

    Propafenone derivative GP46 0

    Propafenone derivative GP57 1

    Propafenone derivative GP62 1

    Propafenone derivative GP88 1

    Propafenone derivative GP90 1

    Propafenone derivative ID 16 1

    Propafenone derivative ID 17 1

    Propafenone derivative ID 19 1

    Propafenone derivative ID 20 1

    Propafenone derivative ID 21 1

    Propafenone derivative ID 22 1

    Propafenone derivative ID 23 1

    Propafenone derivative ID 24 1

  • Propafenone derivative ID 28 1

    Propafenone derivative ID 29 1

    Propafenone derivative ID 36 1

    Propafenone derivative ID 37 1

    Propafenone derivative ID 38 1

    Propafenone derivative ID 39 1

    Propafenone derivative ID 40 1

    Propafenone derivative ID 7b 1

    Propantheline 0

    Propenzolate 1

    Propericiazine 0

    Propiconazole 0

    Propoxur 0

    Propoxyphene 1

    Propranolol 1

    Prothipendyl 0

    Protokylol 0

    Protriptyline 1

    Proxazole 0

    Prozapine

    Purine analog ID 17 1

    Purine analog ID 18 1

    Purine analog ID 24 1

    Purine analog ID 26 1

    Purine analog ID 28 1

    Purine analog ID 3 1

    Purine analog ID 32 1

    Purine analog ID 4 1

    Purine analog ID 5 1

    Purine analog ID 7 1

    Purine analog ID 8 1

    Purine analog ID 9 1

    Puromycin 0

    Pyrathiazine 1

    Pyrilamine 0

    Quinacrine 1

    Quinazosin 0

    Quinidine 1

    Quinupramine 1

    Quipazine 0

    R40 500 1

    R41300 1

    R42164 1

    R49960

    R59022

    R6033 1

    RA-134 1

    RA-14 1

    RA-158 0

    RA-159 0

  • RA-168 1

    RA-17 0

    RA-171 1

    RA-178 1

    RA-19 1

    RA-198 0

    RA-24 1

    RA-3 0

    RA-4 0

    RA-8 1

    RA-83 0

    RE-244 1

    RE-28 1

    RE-34 0

    RE-38 1

    RE-57 1

    RE-61 1

    RE-62 1

    RE-66 0

    RXRA-160

    RXRA-642 1

    RXRA-69 1

    RXRE-104 1

    RXRE-61 0

    RXRE-62 0

    RXRE-63 1

    Racefemine 1

    Racemethorphan 0

    Ranitidine 0

    Razinodil 1

    Reboxetine 1

    Rescinnamine 1

    Reserpic acid 0

    Reserpine 1

    Revenast 1

    Reversin 121 1

    Reversin 205 1

    Rhoifolin 0

    Rifampin 1

    Rifamycin B 0

    Rifamycin SV 0

    Rilapine 1

    Risperidone 1

    Ritodrine 0

    Ritonavir 1

    Ro 4-1284 1

    Ro-04-2249 1

    Ro-04-2250 1

    Ro-04-2285 1

    Ro-04-2287 1

  • Ro-04-2359 1

    Ro-04-2360 1

    Ro-04-2669 1

    Ro11-2933 1

    Rolitetracycline 0

    Ropitoin 1

    Ropizine 1

    Roxithromycin 1

    Rythmol 1

    S 9788 1

    S-Farnesylcysteine 0

    S76 5200 1

    S78 5780

    S78 5781 1

    S79 0491 1

    S79 0671 1

    S79 1099 1

    S79 1100 1

    S79 2823 1

    S81 0337 1

    S81 0339 1

    S81 1951 1

    S83 4096 1

    S83 4163 1

    SCH66336 1

    SDZ-PSC 833 1

    SKF-16467 1

    SKF-3301

    SNC 121 0

    SPS 1768 0

    SPS 1769 1

    SPS 1770 1

    SPS 1772 1

    SPS 1773 1

    SPS 1774 1

    SPS 1775 1

    SPS 1776 1

    SPS 1777 1

    SPS 1778 1

    SPS 1779 1

    SPS 1793 1

    SPS 1835 1

    SPS 1836 0

    SPS 1837 0

    SPS 1838 1

    SPS 1839 1

    SPS 1840 1

    SPS 1841 0

    SPS 1842 1

    SPS 1843 1

  • SPS 1844 1

    SPS 1845 1

    SPS 1846 1

    SPS 1847

    SPS 1848 0

    SPS 1849 1

    SPS 1850 1

    SPS 1852 1

    SPS 1853 1

    SPS 1854 1

    SZ48 1

    Safingol 0

    Salmeterol

    Salverine 0

    Saquinavir 1

    Scopolamine 0

    Secoverine 1

    Selegiline 0

    Selparazine 1

    Sertraline 1

    Sesquiterpene(1) 1

    Sesquiterpene(11) 1

    Sesquiterpene(12) 1

    Sesquiterpene(13) 1

    Sesquiterpene(14) 1

    Sesquiterpene(8) 1

    Setastine 1

    Silybin 1

    Simetride 1

    Simvastatin acid 0

    Sirolimus 1

    Sitagliptin 0

    Solanesol 0

    Solypertine 1

    Spasmadryl 0

    Spiramide 1

    Spirilene 1

    Strophanthidin 0

    Sulconazole 0

    Sulfasalazine 0

    Sulfinpyrazone 0

    Sulforidazine 1

    Suloctidil 0

    Sumatriptan 0

    Suramin 0

    Syrosingopine 1

    T13 1

    TMB8 1

    TPP 0

    TRX-13 0

  • Tacrine 0

    Tacrolimus 1

    Talinolol 0

    Tamoxifen 1

    Tampramine 1

    Tangeretin 1

    Tefludazine 1

    Telithromycin 1

    Terbinafine 0

    Terconazole 1

    Terfenadine 1

    Terodiline 1

    Teroxalene 1

    Testosterone 1

    Tetrabenazine 0

    Tetrahydroquinoline ID 2a 1

    Tetrahydroquinoline ID 2b 1

    Tetrahydroquinoline ID 2f 1

    Tetrahydroquinoline ID 2g 1

    Tetrahydroquinoline ID 3f 1

    Tetrahydroquinoline ID 3g 1

    Tetraphenylphosphonium 0

    Thalicarpine 1

    Thenaldine 0

    Thenyldiamine 0

    Thiethylperazine 1

    Thioproperazine 1

    Thioridazine 1

    Thonzylamine 0

    Tiapamil 1

    Tiaramide 0

    Tilorone 0

    Tilozepine 1

    Tioconazole 0

    Tiodazosin 0

    Tioperidone 1

    Tiopropamine

    Tiprenolol 0

    Tipropidil 0

    Tixadil 0

    Tolamolol 0

    Tolnapersine 1

    Tolpropamine

    Tolyporphin A 1

    Toprilidine 1

    Toremifene 1

    Trazodone 1

    Tretoquinol 0

    Tri-n-butylmethylamminiun 0

    Triazine derivative ID 11 1

  • Triazine derivative ID 12 1

    Triazine derivative ID 15 1

    Triazine derivative ID 16 1

    Triazine derivative ID 17 1

    Triazine derivative ID 18 1

    Triazine derivative ID 20 1

    Triazine derivative ID 21 1

    Triazine derivative ID 22 1

    Triazine derivative ID 23 1

    Triazine derivative ID 24 1

    Triazine derivative ID 25 1

    Triazine derivative ID 26 1

    Triazine derivative ID 30 1

    Triazine derivative ID 32 1

    Triazine derivative ID 33 1

    Triazine derivative ID 34 1

    Triazine derivative ID 35 1

    Triazine derivative ID 36 1

    Triazine derivative ID 37 1

    Triazine derivative ID 38 1

    Triazine derivative ID 39 1

    Triazine derivative ID 40 1

    Triazine derivative ID 42 1

    Triazine derivative ID 44 1

    Triazine derivative ID 45 1

    Triazine derivative ID 46 1

    Triazine derivative ID 47 1

    Triazine derivative ID 54 1

    Triazine derivative ID 57 1

    Triazine derivative ID 6 1

    Triazine derivative ID 7 1

    Triazine derivative ID 8 1

    Triazine derivative ID 9 1

    Triazolam 0

    Trifluoperazine 1

    Trifluperidol 1

    Triflupromazine 1

    Triforine 0

    Trihexyphenidyl 0

    Trimazosin 0

    Trimebutine 1

    Trimeprazine 0

    Trimethoprim 0

    Trimetozine 0

    Trimipramine 1

    Triparanol 1

    Tripelennamine 0

    Triprolidine 1

    Tropirine 1

    Troxonium 0

  • Trypan blue 0

    Tryptanmine 0

    Tryptophan 0

    Tubulzole 0

    U-69593 0

    U10520A 1

    U11555A 0

    U18666A 1

    UCB-26166 1

    UCB-26359 1

    UCB-J028 0

    UCB-L172 1

    UCB-N101 1

    Urapidil 0

    Valinomycin 1

    Vancomycin 0

    Venlafaxine 0

    Verapamil 1

    Verapamil analogue(19) 1

    Verapamil analogue(2) 1

    Verapamil analogue(25) 1

    Verapamil analogue(29) 1

    Verapamil analogue(4) 1

    Verapamil analogue(5) 1

    Vetrabutine 1

    Vinblastine 1

    Vinclozolin 0

    Vincristine 0

    Vindoline 1

    Vitamin A palmitate 0

    W-12 0

    W-13 0

    W-7 0

    W2795 0

    W8-032 1

    Warfarin 0

    XR9051 1

    XR9576 1

    Xenthiorate 0

    Zimeldine 0

    Zipeprol 1

    Zolamine 0

    Zolertine 0

    Zolmitriptan 0

    Zoloperone 0

    Zolpidem 1

    Zomepirac 0

    cis-Flupentixol 1

    cis-Thiothixene 1

    o-Nitropehenyl N,N-dimethylcarbamate 0

  • tRA96023 1

    1-P-gp inhibitor

    0-P-gp non-inhibitor