ligand p-gp inhibition (11-me-leu)-cyclosporin a 1...clanobutin 0 clebopride 0 clemastine 1...
TRANSCRIPT
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ligand P-gp inhibition
(11-Me-Leu)-Cyclosporin A 1
1,2,3,4-Tetrahydro-1-methyl-6,7-isoquinolinediol 0
1,2,3,4-Tetrahydro-6,7-dimethoxy-isoquinoline 0
1,2,3,4-Tetrahydro-isoquinoline 0
1,3,5-Triazacycloheptane 4b 1
1,3,5-Triazacycloheptane 4c 1
1,3,5-Triazacycloheptane 5b 1
1,3,5-Triazacycloheptane 5c 1
1,3,5-Triazacycloheptane 5d 1
1,3,5-Triazacycloheptane 6b 1
1,3,5-Triazacycloheptane 6c 1
1-(3-methoxyphenyl)-N,N-dimethylmethanamine 0
1-(4-chlorbenzhydryl)piperazine 0
1-Benzyl-3-pyrroline 0
1-Benzylimidazole 0
1-Phenethylpiperidine 0
1-Phenylpiperazine 0
11-Deoxycortisol 1
14-Benzoylyohimbine 1
16-Dehydroprogesterone 1
16-Methylprogesterone 1
17-Hydroxypregnenolone 0
17-Hydroxyprogesterone 1
2,2'-Diphenylethylamine 0
2,4,6,8-Tetradiethano 0
2,4,6,8-Tetramopholin 0
2,4,6,8-Tetrapiperidy 0
2,4,6-Trimorpholinepy 0
2,4,8-Trimorpholinepy 0
2-Benzylpyridine 0
2-Chloro-10-[2-(dimethylamino)ethyl] phenothiazine 1
2-Chloro-10-[4-(dimethylamino)butyl] phenothiazine 1
2-Chloroimipramine 1
2-Oxazolidinone 0
3'-4'-Dichlorobenzamil 0
3,8-Dihydroxychlorpromazine 0
3-Methyl choroquine 1
4,8-Dipiperidyl-2,6-D 0
4,8-Dipiperidyl-2,6-M 0
4,8-Dipiperidyl-Dimet 0
4-(2-Dimethylamino)ethyl)morpholine 0
4-Androstene-3,17-dione 1
4-Hydroxytamoxifen 1
4-Hydroxytoremifene 1
4-Iodotamoxifen 1
4-beta-Phorbol 12,13-dibutyrate 1
4-beta-Phorbol 13-acetate 0
4-beta-Phorbol 13-butyrate 0
5-(N,N-hexamethylene)amiloride 0
-
5-(N-Methyl-N-isobutyl)amiloride 0
5-N-acetyl-8-demethylardeemin 1
5-N-acetylardeemin 1
5-[N-Methyl-N-(tert-butyl)]-amiloride 0
6-Phenyl-2,4,7-pterid 0
7,8-Dihydroxychlorpromazine 0
7-Hydroxychlorpromazine 0
AF-1393 1
AG-1112 0
AG-213 0
AG-690 1
AHC-52 1
AHR 06601 1
AHR 16462 1
AHR-16303 1
AN-989 1
AY 9944 1
Acapriazine 0
Acebutolol 0
Acecainide 0
Acepromazine 1
Aceprometazine 1
Acetophenazine 1
Acridine 0
Acridone-4-carboxamide 22 1
Acridone-4-carboxamide 23 1
Acridone-4-carboxamide 24 1
Acridone-4-carboxamide 28 1
Acridone-4-carboxamide 29 1
Acridone-4-carboxamide 30 1
Acridone-4-carboxamide 31 1
Acridone-4-carboxamide 32 1
Acridone-4-carboxamide 36 1
Acridone-4-carboxamide 39 1
Acridone-4-carboxamide 43 1
Acridone-4-carboxamide 44 1
Acridone-4-carboxamide 47 1
Acridone-4-carboxamide 48 1
Acridone-4-carboxamide 49 1
Acridone-4-carboxamide 50 1
Acridone-4-carboxamide 51 1
Acridone-4-carboxamide 52 1
Acridone-4-carboxamide 53 1
Acridone-4-carboxamide 54 1
Acridone-4-carboxamide 55 1
Acridone-4-carboxamide 59 1
Acridone-4-carboxamide 60 1
Acridone-4-carboxamide 61 1
Acridone-4-carboxamide 64 1
Acridone-4-carboxamide 65 1
-
Acridone-4-carboxamide 66 1
Acridone-4-carboxamide 67 1
Acridone-4-carboxamide 68 1
Acridone-4-carboxamide 69 1
Acridone-4-carboxamide 70 1
Acridone-4-carboxamide 71 1
Acridone-4-carboxamide 72 1
Acridone-4-carboxamide 73 1
Acridone-4-carboxamide 74 1
Acridone-4-carboxamide 75 1
Acridone-4-carboxamide 76 1
Acridone-4-carboxamide 77 1
Acridone-4-carboxamide 78 1
Acridone-4-carboxamide 79 1
Acridone-4-carboxamide 80 1
Acridone-4-carboxamide 81 1
Acridone-4-carboxamide 82 1
Acridone-4-carboxamide 83 1
Acridone-4-carboxamide 85 1
Acrivastine 0
Actinomycin D 0
Adiphenine 0
Aldicarb 0
Aldoxycarb 0
Aldrich 21430-2 1
Almitrine 1
Alpertine 1
Alpha-Tocopherol 0
Alprenolol 1
Alverine
Amantadine 0
Ambodryl 0
Amiloride 0
Aminocarb 0
Aminopentamide 0
Amiodarone 1
Amitriptyline 1
Amlodipine 1
Amodiaquin 0
Amotriphene 1
Amoxapine 1
Amoxecaine 0
Amperozide 1
Amphotericin B 0
Amprenavir 1
Androstenedione 1
Androsterone 1
Antazoline 0
Antenolol 0
Antipyrine 0
-
Apomorphine 0
Aprindine 1
Ascorbic acid 0
Asocainol 1
Astemizole 1
Atorvastatin (methyl ester) 1
Atorvastatin lactone 1
Atrazine 0
Atropine 0
Aureobasidin A (ABA) 1
Azaclorazine 1
Azaconazole 0
Azaperone 0
Azelastine 1
Azidopine 1
Azidoprocainamide methoiodide 0
Azipramine 1
B3-243 1
B669 1
B9109-012 1
BIBW 22 1
BW 1019W91 1
BW 1136U89 1
BW 1288U89 1
BW 1351W91 1
BW 1379W91 1
BW 565C81 1
Bamipine 0
Barnidipine 1
Befuraline 0
Benactyzine 0
Bencyclane 0
Benidipine 1
Benzathine 1
Benzmalecene 0
Benzofuran derivative 2a 0
Benzofuran derivative 2c 1
Benzofuran derivative 2d 1
Benzofuran derivative 2e 1
Benzofuran derivative 2f 1
Benzquinamide 0
Benztropine 1
Bepridil 1
Berberine 0
Bevantolol 1
Bifonazole 1
Biperiden 0
Biphenamine 0
Biricodar 1
Bisobrin 0
-
Bleomycin A2 0
Boldine 0
Boxidine 0
Bromocriptine 1
Brompheniramine 0
Bryostatin 0
Bucainide 1
Buclizine 1
Budipine
Buflomedil 0
Bufuralol 1
Bunaftine 1
Buspirone 1
Butalamine 0
Butaperazine 1
Buterizine 1
Butethamate 0
CP-100356 1
CP-101556 1
CP-114416 1
CP-114769 1
CP-117227 1
CP-12379 1
CP-141938 1
CP-147478 1
CP-69042 1
Calcimycin 0
Calphostin C 1
Captodiame
Carbamazepine 0
Carbaryl 0
Carbinoxamine 1
Carbiphene 1
Carnitine 0
Caroverine 1
Carphenazine 1
Carvedilol 1
Carvedilol metabolite M2 0
Carvedilol metabolite M4 0
Carvedilol metabolite M5 0
Catharanthine 1
Cefoperazone 0
Cefotetan 0
Ceftazidime 0
Celiprolol 0
Cepharanthine 1
Cephradine 0
Cetiedil 1
Cetrizine 0
Chelerythrine 0
-
Chlophedianol 0
Chloracyzine 1
Chlorbenzoxamine 1
Chlorcyclizine 0
Chlorogenic acid 0
Chloropyramine 0
Chloroquine 0
Chlorpheniramine 0
Chlorphenoxamine
Chlorproethazine 1
Chlorpromazine 1
Chlorprothixene 1
Chlorzoxazone 0
Chromonar
Cimetidine 0
Cinchonidine 1
Cinepaxadil 1
Cinepazet 0
Cinepazic acid 0
Cinepazide 0
Cinnarizine 1
Cinprazole 1
Cinpropazide 0
Cintriamide 0
Cinuperone 1
Ciprofloxacin 0
Citalopram 0
Citatepine 1
Citenamide 0
Clamoxyquin 0
Clanobutin 0
Clebopride 0
Clemastine 1
Clemizole 1
Cletoquine 0
Clobutinol 0
Clocinizine 1
Clomestrone 0
Clomiphene 0
Clomipramine 1
Clonidine 0
Clopenthixol 1
Cloperastine 1
Clopimozide 1
Clopipazan 1
Clothiapine 1
Clothixamide 1
Clotrimazole 1
Colchicine 0
Colforsin 1
-
Coralyne 0
Corticosterone 0
Cortisone 0
Corynanthine 1
Coumaphos 1
Cryptophycin 1
Cyclobenzaprine 1
Cyclofenazine 1
Cyclopeptolide(1) 0
Cyclopeptolide(11) 0
Cyclopeptolide(12a) 1
Cyclopeptolide(12b) 1
Cyclopeptolide(15a) 1
Cyclopeptolide(15b) 1
Cyclopeptolide(16a) 1
Cyclopeptolide(16c) 1
Cyclopeptolide(16h) 1
Cyclopeptolide(18) 1
Cyclopeptolide(19) 0
Cyclopeptolide(2a) 1
Cyclopeptolide(2c) 1
Cyclopeptolide(2f) 1
Cyclopeptolide(3a) 1
Cyclopeptolide(3c) 1
Cyclopeptolide(3f) 1
Cyclopeptolide(3g) 1
Cyclopeptolide(3h) 1
Cyclopeptolide(3i) 1
Cyclopeptolide(3j) 1
Cyclopeptolide(3l) 1
Cyclopeptolide(3n) 1
Cyclopeptolide(4) 1
Cyclopeptolide(7) 1
Cyclopeptolide(8) 1
Cyclopeptolide(9) 1
Cyclophenazine 1
Cyclosporin A 1
Cyclosporin C 1
Cyclosporin G 1
Cypermethrin 1
Cyproheptadine 1
Cytochalasin A 0
Cytochalasin C 0
Cytochalasin D 0
Cytochalasin E 1
Cytochalasin H 0
Cytochalasin J 0
D490 1
D525 1
D528 0
-
D557 1
D559 1
D595 1
D784 1
D894 1
DDE 0
DDT 0
DHP-014 1
DMDP 1
DPDPE 0
Dagapamil 1
Danitracen 0
Dapiprazole 0
Darodipine 1
Debrisoquin 0
Dehydroemetine 0
Delavirdine 1
Delfantrine 0
Deltorphin II 0
Denzimol 0
Deoxycorticosterone 1
Desethylamiodarone 1
Desipramine 1
Desmethoxyyangonin 1
Desmethylazelastine 1
Desmethylchlorpromazine 0
Desmethylcitalopram 0
Desmethylsertraline 1
Devapamil 1
Dexamethasone 0
Dexniguldipine 1
Dialifos 0
Dibenzylamine 0
Dibozan 0
Dibucaine 1
Dicapthon 1
Diclofensine 0
Didesmethylchlorpromzine 0
Diethylaniline 0
Diethylstilbestrol 1
Difloxacin 0
Difluanine 1
Digoxin 0
Dihydroergotamine 0
Dihydromethysticin 1
Dihydropyridine DP11 1
Dihydropyridine DP5 1
Dihydropyridine DP6 1
Dihydropyridine DP7 1
Dihydropyridine DP9 1
-
Dihydropyrroloquinoline series 14 0
Dihydropyrroloquinoline series 27 1
Diisopromine
Dilazep 1
Diltiazem 1
Dimethindene 1
Diosmetin 0
Diosmin 0
Diphenamid 0
Diphenazoline 0
Diphenidol 1
Diphenylpyraline 1
Disopyramide 0
Dixyrazine 1
Dobutamine 0
Doconazole 1
Domperidone 0
Doxapram 1
Doxazosin
Doxepine 1
Doxorubicin 0
Doxylamine 0
Drobuline 1
Drofenine 0
Droloxifen 0
Droprenilamine 1
Droproizine 0
Duoperone 1
EKI-785 1
Ebastine 1
Econazole 0
Efonidipine 1
Eletriptan 0
Eltoprazine 0
Emepronium 0
Emetine 0
Emopamil 1
Enciprazine 1
Endosulfan 1
Enilconazole 0
Enoxacin 0
Epinephrine 0
Eprazinone 1
Eprozinol 1
Equilenine 0
Equilin 0
Ergocristine 1
Ergocryptine 1
Ergonovine 0
Ergotamine 1
-
Erythromycin 1
Estradiol 0
Estriol 0
Estrone 0
Etafenone 1
Ethylbenztropine 1
Ethylbenzylaniline 0
Etifelmin 0
Etodroxizine
Etolotifene 1
Etomidoline 1
Etoposide 0
Euphodendroidin A 1
Euphodendroidin B 1
Euphodendroidin C 1
Euphodendroidin D 1
Euphodendroidin E 1
Euphodendroidin G 1
Euphodendroidin H 1
Euphodendroidin I 1
Euprocin 1
Falipamil 0
Famciclovir 0
Farnesyl analog AFCA 1
Farnesyl analog AFCMA 1
Farnesyl analog AFCME 1
Febuverine 1
Felodipine 1
Fenbutrazate 1
Fendiline 1
Fenoctimine 0
Fenoterol 0
Fenoxedil 1
Fenpipramide 0
Fenpiverinium 0
Fenticonazole 1
Fenvalerate 0
Fexofenadine 0
Filipin 0
Fisetin 0
Flavonoid ID 13 1
Flavonoid ID 21 0
Flavonoid ID 22 0
Flavonoid ID 23 0
Flavonoid ID 24 0
Flavonoid ID 37 1
Flavonoid ID 38 0
Fleroxacin 0
Flesinoxan 0
Flezelastine 1
-
Flordipine 1
Fluanisone 1
Fluazifop-butyl 0
Fluconazole 0
Flumazenil 0
Flunarizine 1
Fluoxetine 1
Fluperamide 1
Fluperlapine 1
Fluphenazine 1
Flurazepam 1
Fluspirilene 1
Fluvoxamine 1
GF120918 1
GGCME 1
GW 420867 1
Gallopamil 1
Gamfexine 0
Geldanamycin 1
Geldanamycin 17-AAG 1
Gepirone 0
Ginsenoside Rg3 1
Ginsenoside Rh2 1
Glaucine 1
Gramine 0
Guanabenz 0
Guanfacine 0
H-7 0
H-89 1
HA-1004 0
HDL-2722 0
Halopemide 1
Haloperidol 1
Hepzidine 1
Hexadiline 0
Hexobendine 1
Hexoprenaline 0
Histapyrrodine 0
Hoechst 33342 0
Homochlorocyclizine 0
Homofenazine
Homoveratrylamine 0
Hoquizil 0
Hydramethylnon 1
Hydrastine 0
Hydrocotarnine 0
Hydromorphone 0
Hydroxyzine 1
Hyperforin 0
Idarubicin 1
-
Imatinib 1
Imiclopazine 0
Imipramine 1
Imolamine 0
Imoxiterol 0
Indinavir 0
Indomethacin 0
Isoconazole 1
Isoniazid 0
Isopromethazine 1
Isoxsuprine 0
Isradipine 1
Itraconazole
Ivermectin Bla 1
Jatrophane diterpene(7) 1
Jatrophane diterpenoid(1) 1
Jatrophane diterpenoid(10) 1
Jatrophane diterpenoid(11) 1
Jatrophane diterpenoid(12) 1
Jatrophane diterpenoid(13) 1
Jatrophane diterpenoid(14) 1
Jatrophane diterpenoid(15) 1
Jatrophane diterpenoid(16) 1
Jatrophane diterpenoid(2) 1
Jatrophane diterpenoid(3) 1
Jatrophane diterpenoid(5) 1
Jatrophane diterpenoid(6) 1
Jatrophane diterpenoid(8) 1
Jatrophane diterpenoid(9) 1
K02 1
Keoxifene 0
Ketamine 0
Ketoconazole 1
Ketotifen 1
LR 764 0
LU43918 1
LU46324 1
LU47474 1
LU48895 1
LU49667 1
LU49940 1
LU51903 1
LY18947 0
LY292540 1
LY296097 1
LY335979 1
LY335983 1
LY350344 1
Labetalol 0
Laudanosine 1
-
Laudanosoline 0
Lenperone 1
Levodopa 0
Levophacetoperane 0
Lidocaine 0
Lidoflazine 1
Linadryl 1
Lindane 0
Lobeline 1
Lombazole
Loperamide 1
Lopinavir 1
Loratadine 1
Lorcainide 1
Losartan 0
Lovastatin acid 0
Lovastatin lactone 1
Loxapine 1
Luteolin 0
Luteolin-4'-O-glucoside 0
MA 1499 1
MA 1509 1
MA 1510 1
MA 1586 1
MA 1588 1
MA 1598 1
MA 1813 1
MA 1862 0
MA 1865 0
MA 1880 0
MDL 6792
MDL-10393
MDL8917V 1
MDR reversal agent 15h 1
MDR reversal agent 15i 1
MDR reversal agent 15m 1
MDR reversal agent 15o 1
MDR reversal agent 15u 1
MDR reversal agent 15x 1
MDR reversal agent 28a 1
MDR reversal agent 28c 1
MDR reversal agent 35a 1
MDR reversal agent 35d 1
MDR reversal agent 37b 1
MER37 1
MK-571 0
MM36 1
MS-209 1
Macbecin II 1
Manidipine 1
-
Mannitol 0
Maprotiline 1
Maroxepine 0
Mebendazole 1
Mebeverine 1
Meclizine 1
Mecloxamine 0
Medroxyprogesterone 1
Medroxyprogesterone acetate 1
Mefloquine 1
Megestrol Acetate 1
Meglitinide 0
Memotine 0
Mephentermine 0
Mephenytoin 0
Mepramidil 1
Meprobamate 0
Mequitazine 1
Mesoridazine 1
Mesuprine 0
Metergoline 1
Methadone 1
Methaphenilene 0
Methdilazine 0
Methixene 0
Methomyl 0
Methotrimeprazine 1
Methoxychlor 0
Methoxypromazine
Methyl Cellosolve Acetate 0
Methylamine 0
Methysergide 0
Methysticin 1
Metiapine 1
Metoclopramide 0
Metofenazate 1
Metopimazine 0
Metoprolol 0
Metoserpate 1
Metoxepin 1
Mevinphos 0
Mexilitene 0
Mezilamine 0
Mianserin 0
Mibefradil 1
Miconazole 0
Midazolam 1
Mifepristone (RU486) 1
Milenperone 1
Milipertine 1
-
Mioflazine 1
Mirex 0
Mitomycin C 0
Mitoxantrone 0
Mixidine 0
Moclobemide 0
Monensin 1
Mopidamol 0
Morin 0
Morphine 0
Motracetam 0
Moxapridine 1
N,N'-Diphenyl-p-phenylenediamine 0
N,N'-dibenzylethylene diamine 0
N,N-Bis(alkanol)amine aryl ester analog 21 1
N,N-Bis(alkanol)amine aryl ester analog 5 0
N,N-Bis(alkanol)amine aryl ester analog 6 1
N,N-Bis(alkanol)amine aryl ester analog 8 1
N,N-Bis(alkanol)amine aryl ester analog 9 1
N,N-Dimethylbenzylamine 0
N,N-bis(cyclohexanol)amine aryl ester (3) 1
N,N-bis(cyclohexanol)amine aryl ester (4) 1
N,N-bis-arylalkylamine derivative(1) 1
N,N-bis-arylalkylamine derivative(2) 1
N,N-diethylcyclohexylamine 0
N-Benzylbenzamide 0
N-Methyl-gallopamil 0
N-Norlaudanosine 1
N-Norlaudanosoline 0
N-Phenyl-1-naphthylamine 0
N-Phenyl-2-naphthylamine 0
N-acetyl-daunorubicin 1
N-acyloxy-1,4-dihydropyridine(10) 1
N-acyloxy-1,4-dihydropyridine(5) 1
N-acyloxy-1,4-dihydropyridine(6) 1
N-acyloxy-1,4-dihydropyridine(7) 1
N-acyloxy-1,4-dihydropyridine(8) 1
N-acyloxy-1,4-dihydropyridine(9) 1
N-desmethyl-toremifene 1
N-desmethyl-venlafaxine 1
N-desmethyltamoxifen 1
N-trialkylglycine N31214C 1
NK-101 0
NK-106 1
NSC 102843 1
NSC 169647 0
NSC 220202 1
NSC 303594 1
NSC 30774 1
NSC 33128 1
-
NSC 344003 1
NSC 359449 0
NSC 633043 0
NSC 633320 0
NSC 640085 0
NSC 648114 1
NSC 649087 1
NSC 665333 1
NSC 666490 0
NSC 667739 1
NSC 668360 1
NSC 673413 0
NSC 676590 1
NSC 676591 1
NSC 676600 1
NSC 676605 1
NSC 88116 0
NSC 88657 0
NSC 94907 0
Nafcillin 0
Nafiverine 1
Nafoxidine 1
Naftifine 0
Naftopidil 1
Naftoxate 1
Nalbuphine 0
Naloxone 0
Naltrexone 0
Naltrindole 0
Nefazodone 1
Nelfinavir 1
Neostigmine 0
Nicardipine 1
Nicergoline 1
Nifedipine 1
Nilprazole 1
Niludipine 1
Nimodipine 1
Nisoldipine 1
Nitrazepam 0
Nitrendipine 1
Nitromifene 1
Nobiletin 1
Nomifensine 0
Nordazepam 0
Norfloxacin 0
Norfluxetine 1
Norgallopamil 1
Nortriptylene 1
Norverapamil 1
-
Noscapine 1
Nuclotixene 0
Nylidrin 0
O-desmethyl-venlafaxine 0
OBF-1622 0
OBF-1822 1
OBF-1834 0
OC144-093 1
OL-57 1
Ofloxacin 0
Oleanolic acid 0
Olivomycin A 0
Omeprazole 1
Omeprazole sulfone 0
Omoconazole 0
Opipramol 0
Opromazine 1
Orconazole
Oxamarin 0
Oxatomide 1
Oxiconazole 0
Oxolinic acid 0
Oxprenolol 0
Oxybutynin 1
Oxyfedrine 0
Oxypendyl 0
Oxyperomide 0
Oxypertine 1
PAK-1 1
PAK-200 1
PAK-8 0
PGP-4008 1
Palmitoylcartinine 0
Papaverine 0
Paraquat 0
Parathion-methyl 1
Parconazole 0
Paroxetine 1
Pefloxacin 0
Penfluridol 1
Pentachlorophenol 0
Pentazocine 1
Peptoid 1 1
Peptoid 2 1
Peradoxime 1
Perafensine 0
Perazine
Perhexilline 0
Perimetazine 1
Perlapine 1
-
Perphenazine 1
Phenethylamine 0
Pheniramine 0
Phenoxazine ID 11 1
Phenoxazine ID 12 1
Phenoxazine ID 15 0
Phenoxazine ID 18 1
Phenoxazine ID 2 1
Phenoxazine ID 3 1
Phenoxazine ID 4 1
Phenoxazine ID 5 1
Phenylamil 1
Phenyltoloxamine 0
Phenytoin 0
Phorbol 0
Phosmet 0
Physostigmine 1
Pifarnine 1
Piflutixol 1
Pimethixene 1
Pimozide 1
Pinafide 0
Pinoxepine 1
Pipamperone 1
Pipemidic Acid 0
Piperacetazine
Piperamide 0
Piperdimerine A 1
Piperine 1
Pipoxizine 1
Pipoxolan 0
Pirenzepine 0
Pirohenptine 1
Piromidic Acid 0
Pirprofen 0
Pizotyline 1
Pramiverin 0
Pravastatin 0
Prazosin 1
Predifine 1
Pregnanedione 1
Prenoverine 0
Prenoxidiazine 1
Prenylamine 1
Primaquine 0
Primidolol 0
Prinixic acid 0
Pristinamycin IA 1
Proadifen 1
Prochlorperazine 1
-
Procyclidine 1
Prodipine
Progabide 1
Progesterone 1
Promazine 0
Promethazine 1
Propafenone 1
Propafenone derivative 1b 1
Propafenone derivative 1c 1
Propafenone derivative 1e 1
Propafenone derivative 1f 1
Propafenone derivative 1g 1
Propafenone derivative 1i 1
Propafenone derivative 1k 1
Propafenone derivative GP01 1
Propafenone derivative GP02 1
Propafenone derivative GP03 0
Propafenone derivative GP05 1
Propafenone derivative GP07 0
Propafenone derivative GP10 0
Propafenone derivative GP134 1
Propafenone derivative GP155 1
Propafenone derivative GP159 1
Propafenone derivative GP163 1
Propafenone derivative GP164 1
Propafenone derivative GP17 0
Propafenone derivative GP240 1
Propafenone derivative GP29 1
Propafenone derivative GP31 1
Propafenone derivative GP339 1
Propafenone derivative GP358 1
Propafenone derivative GP359 1
Propafenone derivative GP360 1
Propafenone derivative GP366 1
Propafenone derivative GP381 1
Propafenone derivative GP388 1
Propafenone derivative GP389 0
Propafenone derivative GP46 0
Propafenone derivative GP57 1
Propafenone derivative GP62 1
Propafenone derivative GP88 1
Propafenone derivative GP90 1
Propafenone derivative ID 16 1
Propafenone derivative ID 17 1
Propafenone derivative ID 19 1
Propafenone derivative ID 20 1
Propafenone derivative ID 21 1
Propafenone derivative ID 22 1
Propafenone derivative ID 23 1
Propafenone derivative ID 24 1
-
Propafenone derivative ID 28 1
Propafenone derivative ID 29 1
Propafenone derivative ID 36 1
Propafenone derivative ID 37 1
Propafenone derivative ID 38 1
Propafenone derivative ID 39 1
Propafenone derivative ID 40 1
Propafenone derivative ID 7b 1
Propantheline 0
Propenzolate 1
Propericiazine 0
Propiconazole 0
Propoxur 0
Propoxyphene 1
Propranolol 1
Prothipendyl 0
Protokylol 0
Protriptyline 1
Proxazole 0
Prozapine
Purine analog ID 17 1
Purine analog ID 18 1
Purine analog ID 24 1
Purine analog ID 26 1
Purine analog ID 28 1
Purine analog ID 3 1
Purine analog ID 32 1
Purine analog ID 4 1
Purine analog ID 5 1
Purine analog ID 7 1
Purine analog ID 8 1
Purine analog ID 9 1
Puromycin 0
Pyrathiazine 1
Pyrilamine 0
Quinacrine 1
Quinazosin 0
Quinidine 1
Quinupramine 1
Quipazine 0
R40 500 1
R41300 1
R42164 1
R49960
R59022
R6033 1
RA-134 1
RA-14 1
RA-158 0
RA-159 0
-
RA-168 1
RA-17 0
RA-171 1
RA-178 1
RA-19 1
RA-198 0
RA-24 1
RA-3 0
RA-4 0
RA-8 1
RA-83 0
RE-244 1
RE-28 1
RE-34 0
RE-38 1
RE-57 1
RE-61 1
RE-62 1
RE-66 0
RXRA-160
RXRA-642 1
RXRA-69 1
RXRE-104 1
RXRE-61 0
RXRE-62 0
RXRE-63 1
Racefemine 1
Racemethorphan 0
Ranitidine 0
Razinodil 1
Reboxetine 1
Rescinnamine 1
Reserpic acid 0
Reserpine 1
Revenast 1
Reversin 121 1
Reversin 205 1
Rhoifolin 0
Rifampin 1
Rifamycin B 0
Rifamycin SV 0
Rilapine 1
Risperidone 1
Ritodrine 0
Ritonavir 1
Ro 4-1284 1
Ro-04-2249 1
Ro-04-2250 1
Ro-04-2285 1
Ro-04-2287 1
-
Ro-04-2359 1
Ro-04-2360 1
Ro-04-2669 1
Ro11-2933 1
Rolitetracycline 0
Ropitoin 1
Ropizine 1
Roxithromycin 1
Rythmol 1
S 9788 1
S-Farnesylcysteine 0
S76 5200 1
S78 5780
S78 5781 1
S79 0491 1
S79 0671 1
S79 1099 1
S79 1100 1
S79 2823 1
S81 0337 1
S81 0339 1
S81 1951 1
S83 4096 1
S83 4163 1
SCH66336 1
SDZ-PSC 833 1
SKF-16467 1
SKF-3301
SNC 121 0
SPS 1768 0
SPS 1769 1
SPS 1770 1
SPS 1772 1
SPS 1773 1
SPS 1774 1
SPS 1775 1
SPS 1776 1
SPS 1777 1
SPS 1778 1
SPS 1779 1
SPS 1793 1
SPS 1835 1
SPS 1836 0
SPS 1837 0
SPS 1838 1
SPS 1839 1
SPS 1840 1
SPS 1841 0
SPS 1842 1
SPS 1843 1
-
SPS 1844 1
SPS 1845 1
SPS 1846 1
SPS 1847
SPS 1848 0
SPS 1849 1
SPS 1850 1
SPS 1852 1
SPS 1853 1
SPS 1854 1
SZ48 1
Safingol 0
Salmeterol
Salverine 0
Saquinavir 1
Scopolamine 0
Secoverine 1
Selegiline 0
Selparazine 1
Sertraline 1
Sesquiterpene(1) 1
Sesquiterpene(11) 1
Sesquiterpene(12) 1
Sesquiterpene(13) 1
Sesquiterpene(14) 1
Sesquiterpene(8) 1
Setastine 1
Silybin 1
Simetride 1
Simvastatin acid 0
Sirolimus 1
Sitagliptin 0
Solanesol 0
Solypertine 1
Spasmadryl 0
Spiramide 1
Spirilene 1
Strophanthidin 0
Sulconazole 0
Sulfasalazine 0
Sulfinpyrazone 0
Sulforidazine 1
Suloctidil 0
Sumatriptan 0
Suramin 0
Syrosingopine 1
T13 1
TMB8 1
TPP 0
TRX-13 0
-
Tacrine 0
Tacrolimus 1
Talinolol 0
Tamoxifen 1
Tampramine 1
Tangeretin 1
Tefludazine 1
Telithromycin 1
Terbinafine 0
Terconazole 1
Terfenadine 1
Terodiline 1
Teroxalene 1
Testosterone 1
Tetrabenazine 0
Tetrahydroquinoline ID 2a 1
Tetrahydroquinoline ID 2b 1
Tetrahydroquinoline ID 2f 1
Tetrahydroquinoline ID 2g 1
Tetrahydroquinoline ID 3f 1
Tetrahydroquinoline ID 3g 1
Tetraphenylphosphonium 0
Thalicarpine 1
Thenaldine 0
Thenyldiamine 0
Thiethylperazine 1
Thioproperazine 1
Thioridazine 1
Thonzylamine 0
Tiapamil 1
Tiaramide 0
Tilorone 0
Tilozepine 1
Tioconazole 0
Tiodazosin 0
Tioperidone 1
Tiopropamine
Tiprenolol 0
Tipropidil 0
Tixadil 0
Tolamolol 0
Tolnapersine 1
Tolpropamine
Tolyporphin A 1
Toprilidine 1
Toremifene 1
Trazodone 1
Tretoquinol 0
Tri-n-butylmethylamminiun 0
Triazine derivative ID 11 1
-
Triazine derivative ID 12 1
Triazine derivative ID 15 1
Triazine derivative ID 16 1
Triazine derivative ID 17 1
Triazine derivative ID 18 1
Triazine derivative ID 20 1
Triazine derivative ID 21 1
Triazine derivative ID 22 1
Triazine derivative ID 23 1
Triazine derivative ID 24 1
Triazine derivative ID 25 1
Triazine derivative ID 26 1
Triazine derivative ID 30 1
Triazine derivative ID 32 1
Triazine derivative ID 33 1
Triazine derivative ID 34 1
Triazine derivative ID 35 1
Triazine derivative ID 36 1
Triazine derivative ID 37 1
Triazine derivative ID 38 1
Triazine derivative ID 39 1
Triazine derivative ID 40 1
Triazine derivative ID 42 1
Triazine derivative ID 44 1
Triazine derivative ID 45 1
Triazine derivative ID 46 1
Triazine derivative ID 47 1
Triazine derivative ID 54 1
Triazine derivative ID 57 1
Triazine derivative ID 6 1
Triazine derivative ID 7 1
Triazine derivative ID 8 1
Triazine derivative ID 9 1
Triazolam 0
Trifluoperazine 1
Trifluperidol 1
Triflupromazine 1
Triforine 0
Trihexyphenidyl 0
Trimazosin 0
Trimebutine 1
Trimeprazine 0
Trimethoprim 0
Trimetozine 0
Trimipramine 1
Triparanol 1
Tripelennamine 0
Triprolidine 1
Tropirine 1
Troxonium 0
-
Trypan blue 0
Tryptanmine 0
Tryptophan 0
Tubulzole 0
U-69593 0
U10520A 1
U11555A 0
U18666A 1
UCB-26166 1
UCB-26359 1
UCB-J028 0
UCB-L172 1
UCB-N101 1
Urapidil 0
Valinomycin 1
Vancomycin 0
Venlafaxine 0
Verapamil 1
Verapamil analogue(19) 1
Verapamil analogue(2) 1
Verapamil analogue(25) 1
Verapamil analogue(29) 1
Verapamil analogue(4) 1
Verapamil analogue(5) 1
Vetrabutine 1
Vinblastine 1
Vinclozolin 0
Vincristine 0
Vindoline 1
Vitamin A palmitate 0
W-12 0
W-13 0
W-7 0
W2795 0
W8-032 1
Warfarin 0
XR9051 1
XR9576 1
Xenthiorate 0
Zimeldine 0
Zipeprol 1
Zolamine 0
Zolertine 0
Zolmitriptan 0
Zoloperone 0
Zolpidem 1
Zomepirac 0
cis-Flupentixol 1
cis-Thiothixene 1
o-Nitropehenyl N,N-dimethylcarbamate 0
-
tRA96023 1
1-P-gp inhibitor
0-P-gp non-inhibitor