one-pot synthesis of new heterocycles: 2,4-disubstituted...

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2003 Fused pyrimidine derivatives Fused pyrimidine derivatives R 0515 One-Pot Synthesis of New Heterocycles: 2,4-Disubstituted 6,7-Dihydro-5H-ben- zo[6,7]cyclohepta[1,2-d]pyrimidines. — The pharmacologically interesting title compounds are directly obtained from condensation of benzosuberone (I) with various nitriles in the presence of triflic anhydride. — (HERRERA, A.; MARTINEZ-ALVAREZ*, R.; CHIOUA, R.; CHIOUA, M.; Tetrahedron Lett. 44 (2003) 10, 2149-2151; Dep. Quim. Org., Fac. Cienc. Quim., Univ. Complutense, E-28040 Madrid, Spain; Eng.) — Mais 22- 158

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2003 Fused pyrimidine derivatives

Fused pyrimidine derivativesR 0515 One-Pot Synthesis of New Heterocycles: 2,4-Disubstituted 6,7-Dihydro-5H-ben-

zo[6,7]cyclohepta[1,2-d]pyrimidines. — The pharmacologically interesting titlecompounds are directly obtained from condensation of benzosuberone (I) with variousnitriles in the presence of triflic anhydride. — (HERRERA, A.;MARTINEZ-ALVAREZ*, R.; CHIOUA, R.; CHIOUA, M.; Tetrahedron Lett. 44(2003) 10, 2149-2151; Dep. Quim. Org., Fac. Cienc. Quim., Univ. Complutense,E-28040 Madrid, Spain; Eng.) — Mais

22- 158