scheduling actions controlled substances regulated chemicals
TRANSCRIPT
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U.S. Department of Justice Drug Enforcement Administration Diversion Control Division Drug & Chemical Evaluation Section
Lists of:
Scheduling Actions
Controlled Substances
Regulated Chemicals
March 2018
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Foreword The first three sections of this booklet list the names of the substances which are described in the Code of Federal
Regulations (CFR) as well as some of those which generate frequent inquiries. The substances are first arranged
alphabetically, then by Drug Enforcement Administration (DEA) drug code number, and finally by Controlled Substances
Act (21 U.S.C. 801 et seq.) (CSA) schedule.
These lists describe the basic or parent chemical and do not describe the salts, isomers, salts of isomers, esters,
ethers, and derivatives which may be controlled substances. These are not comprehensive lists so please note that a
substance need not be listed as a controlled substance to be treated as a scheduled substance for criminal prosecution.
The Other Names column, provides some examples of alternate names for certain compounds, and in some
instances provides examples of positional isomers. If outside parties want to ensure that a compound is not
considered a scheduled substance or listed chemical, they should write the DEA, Drug and Chemical Evaluation
Section (DRE), Diversion Control Division, 8701 Morrissette Drive, Springfield, Virginia 22152, for an official
determination.
A substance (not included on these lists) may also be regulated as a controlled substance analogue. A controlled
substance analogue is a substance which is intended for human consumption, is structurally substantially similar to a schedule
I or schedule II substance, is pharmacologically substantially similar to a schedule I or schedule II substance, or is
represented as being similar to a schedule I or schedule II substance and is not an approved medication in the United States.
See 21 U.S.C. 802(32)(A) for the definition of a controlled substance analogue and 21 U.S.C. 813 for the schedule.
The next two sections of this booklet list the Federal Register notices through which the DEA has directed substances
to be added, deleted or transferred between schedules of the CSA. The scheduling changes are listed first in alphabetical
order by substance and then in chronological order by effective date. With the exception of anabolic steroids, section 812 of
the CSA lists only those substances which were controlled in 1970 when the law was enacted. Since then, over 200
substances have been added, removed, or transferred from one schedule to another. The current official list of controlled
substances can be found in section 1308 of the most recent issue of Title 21 Code of Federal Regulations Part 1300 to end (21
CFR 1308) and the final rules which have been published in the Federal Register subsequent to the issuance of the CFR.
The CFR and the Federal Register are available on the U.S. Government Printing Office web site at
https://www.gpo.gov/fdsys/. This information is accessible, also, on the Diversion Control Divisions website at
https://www.deadiversion.usdoj.gov/.
The last section of this booklet identifies the List I and List II chemicals. Certain commercial transactions
involving these chemicals are regulated by the CSA. See 21 CFR 1309, 1310 and 1313 for details.
These lists are intended as general references and are not comprehensive listings of all controlled substances and
regulated chemicals.
Drug and Chemical Evaluation Section Diversion Control Division
Drug Enforcement Administration
Telephone: 202-307-7183 FAX: 202-353-1263
March 2018
http:https://www.deadiversion.usdoj.govhttps://www.gpo.gov/fdsys
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Abbreviations
2C-B = 4-Bromo-2,5-dimethoxyphenethylamine
2C-T-7 = 2,5-Dimethoxy-4(n)-propylthiophenethylamine
BZP = N-Benzylpiperazine
DMT = Dimethyltryptamine
DOM = 4-Methyl-2,5-dimethoxyamphetamine
GBL = Gamma butyrolactone
GHB = Gamma hydroxybutyric acid, gamma hydroxybutyrate, 4-hydroxybutanoic acid, sodium oxybate
LAAM = Levo-alphacetylmethadol
LSD = Lysergic acid diethylamide, lysergide
MDA = 3,4-Methylenedioxyamphetamine
MDE = 3,4-Methylenedioxy-N-ethylamphetamine
MDMA = 3,4-Methylenedioxymethamphetamine
MPPP = 1-Methyl-4-phenyl-4-propionoxypiperidine
P2P = Phenyl-2-propanone, phenylacetone
PCC = 1-Piperidinocyclohexanecarbonitrile
PCE = N-Ethyl-1-phenylcyclohexylamine
PCH = 1-Phenylcyclohexylamine
PCP = 1-(1-Phenylcyclohexyl)piperidine, phencyclidine
PEPAP = 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine
PHP = 1-(1-Phenylcyclohexyl)pyrrolidine
SPA = (-)-1-Dimethylamino-1,2-diphenylethane
TCP = 1-[1-(2-Thienyl)cyclohexyl]piperidine
TCPy = 1-[1-(2-Thienyl)cyclohexyl]pyrrolidine
THC = Tetrahydrocannabinols
THG = Tetrahydrogestrinone
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Scheduling Actions A
lphabetical Order
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Scheduling Actions
- Alphabetical Order -
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
(1-PENTYL-1H-INDOL-3-YL)(2,2,3,3- 05-16-13 78 FR 28735 5/16/2013 I TETRAMETHYLCYCLOPROPYL)METHANONE (UR-144)*
[1-(5-FLUOROPENTYL)-1H-INDAZOL-3- 01-30-15 80 FR 5042 1/30/2015 I YL](NAPHTHALEN-1-YL)METHANONE (THJ-2201)*
[1-(5-FLUORO-PENTYL)1H-INDOL-3-YL](2,2,3,3- 05-16-13 78 FR 28735 5/16/2013 I TETRAMETHYLCYCLOPROPYL)METHANONE(5-FLUORO-UR-144, XLR11)*
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) 09-08-03 03-18-04 69 FR 12794 3/19/2004 I --> 0
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) * 09-20-02 67 FR 59161 9/20/2002 I
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) ** 09-10-03 68 FR 53289 9/20/2003 I
1-[1-(2-THIENYL)CYCLOHEXYL]PYRROLIDINE 03-20-89 07-06-89 54 FR 28414 7/6/1989 I
19-NOR-4,9(10)-ANDROSTADIENEDIONE (estra-4,9(10)-diene- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III 3,17-dione)
2-(4-BROMO-2,5-DIMETHOXYPHENYL)-N-(2- 11-15-13 78 FR 68716 11/15/2013 I METHOXYBENZYL) ETHANAMINE (25B-NBOMe)*
2-(4-CHLORO-2,5-DIMETHOXYPHENYL)-N-(2- 11-15-13 78 FR 68716 11/15/2013 I METHOXYBENZYL) ETHANAMINE (25C-NBOMe)*
2-(4-IODO-2,5-DIMETHOXYPHENYL)-N-(2-METHOXYBENZYL) 11-15-13 78 FR 68716 11/15/2013 I ETHANAMINE (25I-NBOMe)*
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-08-03 03-18-04 69 FR 12794 3/18/2004 I T-7)
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-20-02 67 FR 59163 9/20/2002 I T-7) *
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-10-03 68 FR 53289 9/20/2003 I T-7) **
2,5-DIMETHOXY-4-ETHYLAMPHETAMINE (DOET) 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
2,5-DIMETHOXYAMPHETAMINE (DMA) 05-31-73 09-21-73 38 FR 26447 9/21/1973 I
3,4-DICHLORO-N-[(1- 04-14-16 81 FR 22023 5/15/2016 I DIMETHYLAMINO)CYCLOHEXYLMETHYL]BENZAMIDE) (AH-7921)
3,4-DICHLORO-N-[2-(DIMETHYLAMINO)CYCLOHEXYL]-N- 11-14-16 81 FR 79389 11/14/2016 I METHYLBENZAMIDE (U-47700)*
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE* 10-15-87 52 FR 38225 10/15/1987 I
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE** 10-13-88 53 FR 40061 10/13/1988 I
3,4-METHYLENEDIOXY-N-METHYLCATHINONE 10-21-11 04-12-13 78 FR 21818 4/12/2013 I (METHYLONE)
3,4-METHYLENEDIOXY-N-METHYLCATHINONE 10-21-11 76 FR 65371 10/21/2011 I (METHYLONE)*
3,4-METHYLENEDIOXYPYROVALERONE (MDPV)* 10-21-11 76 FR 65371 10/21/2011 I
3-FLUORO-N-METHYLCATHINONE (3-FMC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
3-FLUORO-N-METHYLCATHINONE (3-FMC)* 03-07-14 79 FR 12938 3/7/2014 I
Scheduling Actions - Alphabetical Order
01-Mar-18 Page 1 of 10
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SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
3-FLUORO-N-METHYLCATHINONE (3-FMC)** 03-04-16 81 FR 11429 3/4/2016 I
3-METHYLFENTANYL 04-24-86 09-22-86 51 FR 33592 9/22/1986 I
3-METHYLFENTANYL* 03-25-85 50 FR 11690 4/25/1985 I
3-METHYLFENTANYL** 04-24-86 51 FR 15474 4/25/1986 I
3-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
3-METHYLTHIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
3-METHYLTHIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
4-ANILINO-N-PHENETHYL-4-PIPERIDINE (ANPP) 04-09-08 06-29-10 75 FR 37296 8/30/2010 II
4-BROMO-2,5-DIMETHOXYAMPHETAMINE 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE 12-20-94 06-02-95 60 FR 28718 6/2/1995 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE* 01-06-94 59 FR 00671 1/6/1994 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE** 12-21-94 59 FR 65710 1/6/1995 I
4-FLUORO-N-METHYLCATHINONE (4-FMC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
4-FLUORO-N-METHYLCATHINONE (4-FMC)* 03-07-14 79 FR 12938 3/7/2014 I
4-FLUORO-N-METHYLCATHINONE (4-FMC)** 03-04-16 81 FR 11429 3/4/2016 I
4-METHOXYAMPHETAMINE (PMA) 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-04-16 03-01-17 82 FR 12171 3/1/2017 I MePPP)
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-07-14 79 FR 12938 3/7/2014 I MePPP)*
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-04-16 81 FR 11429 3/4/2016 I MePPP)**
4-METHYLAMINOREX 10-14-88 04-13-89 54 FR 14799 4/13/1989 I
4-METHYLAMINOREX* 10-15-87 52 FR 38225 10/15/1987 I
4-METHYLAMINOREX** 10-13-88 53 FR 40061 10/13/1988 I
4-METHYL-N-ETHYLCATHINONE (4-MEC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
4-METHYL-N-ETHYLCATHINONE (4-MEC)* 03-07-14 79 FR 12938 3/7/2014 I
4-METHYL-N-ETHYLCATHINONE (4-MEC)** 03-04-16 81 FR 11429 3/4/2016 I
4-METHYL-N-METHYLCATHINONE (MEPHEDRONE)* 10-21-11 76 FR 65371 10/21/2011 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) 09-29-04 69 FR 58050 9/29/2004 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) * 04-04-03 68 FR 16427 4/4/2003 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) 04-01-04 69 FR 17034 4/1/2004 I **
5-METHOXY-N,N-DIMETHYLTRYPTAMINE 08-21-09 12-20-10 75 FR 79296 1/19/2011 I
ACETYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 06-07-17 82 FR 26349 6/7/2017 I PHENYLACETAMIDE)
ACETYL FENTANYL* (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 07-17-15 80 FR 42381 7/17/2015 I PHENYLACETAMIDE)
ACETYL-ALPHA-METHYLFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
ACETYL-ALPHA-METHYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
ACETYL-ALPHA-METHYLFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
ACRYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 07-14-17 82 FR 32453 7/14/2017 I PHENYLACRYLAMIDE)*
ALFAXALONE (5-PREGNAN-3-OL-11,20-DIONE) 03-25-13 02-27-14 79 FR 10985 3/31/2014 IV
Scheduling Actions - Alphabetical Order
01-Mar-18 Page 2 of 10
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FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
ALFENTANIL 04-17-86 01-23-87 52 FR 2516 1/23/1987 I -> II
ALFENTANIL 06-25-84 49 FR 25849 8/24/1984 I
ALPHA-ETHYLTRYPTAMINE 03-07-94 09-12-94 59 FR 46757 9/12/1994 I
ALPHA-ETHYLTRYPTAMINE* 03-12-93 58 FR 13533 3/12/1993 I
ALPHA-ETHYLTRYPTAMINE** 03-07-94 59 FR 10720 3/12/1994 I
ALPHA-METHYLFENTANYL 08-05-81 09-22-81 46 FR 46799 9/22/1981 I
ALPHA-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
ALPHA-METHYLTHIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
ALPHA-METHYLTHIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
ALPHA-METHYLTRYPTAMINE (AMT) 09-29-04 69 FR 58050 9/29/2004 I
ALPHA-METHYLTRYPTAMINE (AMT) * 04-04-03 68 FR 16427 4/4/2003 I
ALPHA-METHYLTRYPTAMINE (AMT) ** 04-01-04 69 FR 17034 4/1/2004 I
ALPHA-PYRROLIDINOBUTIOPHENONE (-PBP) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
ALPHA-PYRROLIDINOBUTIOPHENONE (-PBP)* 03-07-14 79 FR 12938 3/7/2014 I
ALPHA-PYRROLIDINOBUTIOPHENONE (-PBP)** 03-04-16 81 FR 11429 3/4/2016 I
ALPHA-PYRROLIDINOPENTIOPHENONE (-PVP) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
ALPHA-PYRROLIDINOPENTIOPHENONE (-PVP)* 03-07-14 79 FR 12938 3/7/2014 I
ALPHA-PYRROLIDINOPENTIOPHENONE (-PVP)** 03-04-16 81 FR 11429 3/4/2016 I
ALPRAZOLAM 04-29-81 11-12-81 46 FR 55688 11/12/1981 IV
AMINOREX 08-20-93 03-18-94 59 FR 12828 3/18/1994 I
AMINOREX* 09-21-92 57 FR 43399 9/21/1992 I
AMINOREX** 08-24-93 58 FR 44611 9/21/1993 I
AMOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
AMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
ANABOLIC STEROIDS PL 108-358 12-16-05 70 FR 74653 1/17/2006 III
ANABOLIC STEROIDS PL 101-647 02-13-91 56 FR 5753 2/27/1991 III
APOMORPHINE 04-08-76 06-28-76 41 FR 26568 6/28/1976 II -> 0
BENZPHETAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
BENZYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I Expired 11/29/86
BETA-HYDROXY-3-METHYLFENTANYL 11-28-86 01-08-88 53 FR 500 1/8/1988 I
BETA-HYDROXY-3-METHYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
BETA-HYDROXY-3-METHYLFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I Expired 5/29/87
BETA-HYDROXYFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
BETA-HYDROXYFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
BETA-HYDROXYFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
BETA-HYDROXYTHIOFENTANYL* 05-12-16 81 FR 29492 5/12/2016 I
BIPHETAMINE & BIPHETAMINE-T 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
BOLDIONE (Androsta-1,4-diene-3,17-dione) 04-25-08 12-04-09 74 FR 63603 1/4/2010 III
BRIVARACETAM (BRV; UCB-34714; BRIVIACT) 05-12-16 81 FR 29487 5/12/2016 V
Scheduling Actions - Alphabetical Order
01-Mar-18 Page 3 of 10
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SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
BROMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
BUPRENORPHINE 03-21-02 10-07-02 67 FR 62354 10/7/2002 V --> III
BUPRENORPHINE 09-20-82 02-28-85 50 FR 8104 4/1/1985 II -> V
BUTORPHANOL 07-10-97 10-01-97 62 FR 51370 10/31/1997 IV
BUTORPHANOL, THEBAINE DERIVED 04-03-92 07-14-92 57 FR 31126 7/14/1992 II->0 Supersede
d 10/97
BUTYLONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
BUTYLONE* 03-07-14 79 FR 12938 3/7/2014 I
BUTYLONE** 03-04-16 81 FR 11429 3/4/2016 I
BUTYRYL FENTANYL* 05-12-16 81 FR 29492 5/12/2016 I
CAMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CARFENTANIL 01-12-88 10-28-88 53 FR 43684 10/28/1988 II
CARISOPRODOL 11-17-09 12-12-11 76 FR 77330 1/11/2012 IV
CATHINE 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
CATHINONE 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
CHLORDIAZEPOXIDE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CHLORPHENTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CLOBAZAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLONAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CLORAZEPATE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CLORTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CLOTIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CONCENTRATE OF POPPY STRAW 12-20-74 02-14-75 40 FR 6779 2/14/1975 II
CP-47,497 * 03-01-11 76 FR 11075 3/1/2011 I
CP-47,497 ** 02-29-12 77 FR 12201 2/29/2012 I
CP-47,497 C8 HOMOLOGUE * 03-01-11 76 FR 11075 3/1/2011 I
CP-47,497 C8 HOMOLOGUE ** 02-29-12 77 FR 12201 2/29/2012 I
CYCLOPROPYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4- 01-04-18 83 FR 469 1/4/2018 I YL)-N-PHENYLCYCLOPROPANECARBOXAMIDE)*
DELORAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
DESOXYMETHYLTESTOSTERONE (17a-methyl-5a-androst-2- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III en-17-ol, madol)
DEXTROPROPOXYPHENE 01-21-80 06-24-80 45 FR 42264 7/24/1980 IV
DEXTROPROPOXYPHENE 09-29-76 02-11-77 42 FR 8636 3/14/1977 IV
DEXTROPROPOXYPHENE (BULK) 07-22-80 45 FR 48881 9/22/1980 IV -> II
DEXTRORPHAN 04-19-76 10-01-76 41 FR 43401 10/1/1976 I -> 0
DIAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
DICHLORALPHENAZONE (chloral hydrate compound) 12-11-00 08-16-01 66 FR 42943 8/16/2001 clarification of CIV control
DIETHYLPROPION 05-10-73 07-06-73 38 FR 18013 7/6/1973 IV
Scheduling Actions - Alphabetical Order
01-Mar-18 Page 4 of 10
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FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
DIFENOXIN 05-07-75 40 FR 19813 6/1/1975 I
DIFENOXIN 1 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> IV
DIFENOXIN 1/2 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> V
DIHYDROETORPHINE (thebaine derivative) 11-17-00 65 FR 69442 11/17/2000 clarification of CII control
DRONABINOL IN ORAL SOLUTION IN DRUG PRODUCT 03-23-17 82 FR 14815 3/23/2017 II APPROVED FOR MARKETING BY U.S. FOOD AND DRUG ADMIN.
DRONABINOL PRODUCT (MARINOL) 11-05-98 07-02-99 64 FR 35928 7/2/1999 II -> III
DRONABINOL PRODUCT (MARINOL) 10-18-85 05-13-86 51 FR 17476 5/13/1986 I -> II
DROTEBANOL 07-03-73 38 FR 17717 8/6/1973 I
ELUXADOLINE 08-11-15 11-12-15 80 FR 69861 12/17/2015 IV
EMBUTRAMIDE 07-29-05 08-29-06 71 FR 51115 9/28/2006 III
ESKATROL 05-26-71 08-18-71 36 FR 15744 8/18/1971 III -> II
ESTAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ETHYL LOFLAZEPATE 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ETORPHINE HYDROCHLORIDE 11-23-73 03-29-74 39 FR 11535 4/19/1974 I -> II
EZOGABINE 10-21-11 12-15-11 76 FR 77895 12/15/2011 V
FENCAMFAMIN 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENETHYLLINE 05-01-81 07-21-81 46 FR 37503 8/20/1981 I
FENFLURAMINE 05-15-03 68 FR 26247 5/15/2003 IV Withdrew
97 proposed
rule
FENFLURAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 IV
FENFLURAMINE 05-06-97 05-06-97 5/6/1997 IV -> 0
FENPROPOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENTANYL-RELATED SUBSTANCES, AS DEFINED IN 21 02-06-18 83 FR 5188 2/6/2018 I CFR 1308.11(h)*
FETAMIN 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
FLUDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLUNITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLURAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
FOSPROPOFOL 07-23-09 10-06-09 74 FR 51234 11/5/2009 IV
FUBAMB, MMB FUBINACA (2-(1-(4-FLUOROBENZYL)- 11-03-17 82 FR 51154 11/3/2017 I 1HINDAZOLE-3-CARBOXAMIDO)-3- METHYLBUTANOATE*
GAMMA HYDROXYBUTYRIC ACID (GHB) PL 106-172 03-13-00 65 FR 13235 3/13/2000 I
GAMMA HYDROXYBUTYRIC ACID (GHB) FDA approved drug PL 106-172 03-13-00 65 FR 13235 3/13/2000 III products
GLUTETHIMIDE 07-26-90 03-21-91 56 FR 11930 3/21/1991 III -> II
HALAZEPAM 04-29-81 10-29-81 46 FR 53407 10/29/1981 IV
HALOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
HYDROCODONE COMBINATION PRODUCTS 02-27-14 08-22-14 79 FR 49661 10/6/2014 III->II
Scheduling Actions - Alphabetical Order
01-Mar-18 Page 5 of 10
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FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
INDIPLON 01-31-08 01-31-08 1/31/2008 IV
JWH-018 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-018 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-073 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-073 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-200 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-200 ** 02-29-12 77 FR 12201 2/29/2012 I
KETAMINE 04-09-99 07-13-99 64 FR 37673 8/12/1999 III
KETAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LACOSAMIDE 03-10-09 05-21-09 74 FR 23789 6/22/2009 V
LEVO-ALPHACETYLMETHADOL (LAAM) 04-28-93 08-18-93 58 FR 43795 8/18/1993 I -> II
LIBRAX 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted RX
LISDEXAMFETAMINE 02-22-07 05-03-07 72 FR 24532 6/4/2007 II
LOPERAMIDE 07-28-82 11-03-82 47 FR 49840 11/3/1982 V -> 0
LOPERAMIDE 07-29-76 05-18-77 42 FR 25498 6/17/1977 V
LOPRAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LORAZEPAM 06-28-77 10-07-77 42 FR 54546 10/3/1977 IV
LORCASERIN 12-19-12 05-08-13 78 FR 26701 6/7/2013 IV
LORMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
MAZINDOL 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
MAZINDOL 04-17-81 10-27-81 46 FR 52333 11/27/1981 III -> IV
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 02-22-88 53 FR 5156 3/23/1988 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 01-27-88 53 FR 2225 1/27/1988 I -> 0
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 07-27-84 10-14-86 51 FR 36552 11/13/1986 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE)* 05-31-85 50 FR 23118 7/1/1985 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE)** 06-17-86 51 FR 21911 7/1/1986 I
MEBUTAMATE 12-13-74 01-30-75 40 FR 4418 1/30/1975 IV
MECLOQUALONE 05-29-75 07-08-75 40 FR 28611 7/10/1975 I
MEDAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
MEFENOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
MENRIUM 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted RX
METHAMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
METHAQUALONE 08-27-84 49 FR 33870 8/27/1984 II -> I
METHAQUALONE 04-11-73 10-04-73 38 FR 27516 10/4/1973 II
METHASTERONE ( 2 ALPHA-17 ALPHA-DIMETHYL-5 ALPHA- 11-23-11 07-30-12 77 FR 44456 8/29/2012 III ANDROSTAN-17BETA-OL-3-ONE)
METHCATHINONE 04-28-93 10-15-93 58 FR 53404 10/15/1993 I
METHCATHINONE* 05-01-92 57 FR 18824 5/1/1992 I
METHCATHINONE** 04-29-93 58 FR 25934 5/1/1993 I
Scheduling Actions - Alphabetical Order
01-Mar-18 Page 6 of 10
-
FINAL ORDER
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FEDERAL
REGISTER
CITATION EFFECTIVE
DATE
CSA
SCHEDULE
METHOXYACETYL FENTANYL (2-METHOXY-N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLACETAMIDE)*
10-26-17 82 FR 49504 10/26/2017 I
METHYL 2-(1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMBFUBINACA)*
04-10-17 82 FR 17119 4/10/2017 I
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3-CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-CHMICA)*
04-10-17 82 FR 17119 4/10/2017 I
METHYL2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-ADB)*
04-10-17 82 FR 17119 4/10/2017 I
METHYL2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3-METHYLBUTANOATE (5F-AMB)*
04-10-17 82 FR 17119 4/10/2017 I
METHYLPHENIDATE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
MIDAZOLAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
MODAFINIL 04-14-98 01-27-99 64 FR 4050 1/27/1999 IV
MPPP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I
MPPP* 07-10-85 50 FR 28098 8/12/1985 I
MPPP** 08-11-86 51 FR 28695 8/12/1986 I
N-(1-ADAMANTYL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (APINACA, AKB48)*
05-16-13 78 FR 28735 5/16/2013 I
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)1H-INDAZOLE-3-CARBOXAMIDE (ADBFUBINACA)*
04-10-17 82 FR 17119 4/10/2017 I
N-(1-AMINO-3,3DIMETHYL-1-OXOBUTAN-2-YL)1-(CYCLOHEXYLMETHYL)-1H-INDAZOLE-3CARBOXAMIDE (MAB-CHMINACA)*
02-05-16 81 FR 6171 2/5/2016 I
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)*
02-10-14 79 FR 7577 2/10/2014 I
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)**
02-05-16 81 FR 6175 2/5/2016 I
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)
09-06-16 81 FR 61130 9/6/2016 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (AB-PINACA)*
01-30-15 80 FR 5042 1/30/2015 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)1-(CYCLOHEXYLMETHYL) 1H-INDAZOLE-3-CARBOXAMIDE (AB-CHMINACA)*
01-30-15 80 FR 5042 1/30/2015 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE FUBINACA)**
(AB-02-05-16 81 FR 6175 2/5/2016 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE FUBINACA)*
(AB-02-10-14 79 FR 7577 2/10/2014 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (AB-FUBINACA)
09-06-16 81 FR 61130 9/6/2016 I
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLCYCLOPENTANECARBOXAMIDE (CYCLOPENTYL FENTANYL)*
02-01-18 83 FR 4580 2/1/2018 I
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLFURAN-2-CARBOXAMIDE (FURANYL FENTANYL) *
11-29-16 81 FR 85873 11/29/2016 I
Scheduling Actions - Alphabetical Order
01-Mar-18 Page 7 of 10
-
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 02-01-18 83 FR 4580 2/1/2018 I PHENYLISOBUTYRAMIDE (ISOBUTYRYL FENTANYL)*
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLPENTANAMIDE 02-01-18 83 FR 4580 2/1/2018 I (VALERYL FENTANYL)*
N-(2-FLUOROPHENYL)-2-METHOXY-N-(1- 02-01-18 83 FR 4580 2/1/2018 I PHENETHYLPIPERIDIN-4-YL)ACETAMIDE (OCFENTANIL)*
N-(4-CHLOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 02-01-18 83 FR 4580 2/1/2018 I YL)ISOBUTYRAMIDE (PARA-CHLOROISOBUTYRYL FENTANYL)*
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 02-01-18 83 FR 4580 2/1/2018 I YL)BUTYRAMIDE (PARA-FLUOROBUTYRYL FENTANYL)*
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 05-03-17 82 FR 20544 5/3/2017 I YL)ISOBUTYRAMIDE (4-FLUOROISOBUTYRYL FENTANYL)*
N-(4-METHOXYPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 02-01-18 83 FR 4580 2/1/2018 I YL)BUTYRAMIDE (PARA-METHOXYBUTYRYL FENTANYL)*
N-(ADAMANTAN-1-YL)-1-(5-FLUOROPENTYL)-1H-INDAZOLE- 04-10-17 82 FR 17119 4/10/2017 I 3-CARBOXAMIDE (5FAPINACA, 5FAKB48)*
N,N-DIMETHYLAMPHETAMINE 08-02-89 02-02-90 55 FR 3586 2/2/1990 I
N,N-DIMETHYLAMPHETAMINE* 08-03-88 53 FR 29232 8/3/1988 I
N,N-DIMETHYLAMPHETAMINE** 08-02-89 54 FR 31815 8/2/1989 I
NABILONE 06-18-86 04-07-87 52 FR 11042 4/7/1987 II
NALBUPHINE 05-11-76 10-01-76 41 FR 43401 10/1/1976 II -> 0
NALMEFENE 05-31-85 11-04-85 50 FR 45815 11/4/1985 II -> 0
NALOXEGEL 10-29-14 01-23-15 80 FR 3468 1/23/2015 II->0
NALOXONE 07-10-74 12-24-74 39 FR 44392 12/24/1974 II -> 0
NALOXONE HYDROCHLORIDE 08-19-71 09-29-71 36 FR 19116 9/29/1971 II -> 0
NALTREXONE 12-09-74 03-06-75 40 FR 10455 3/6/1975 II -> 0
NAPHYRONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
NAPHYRONE* 03-07-14 79 FR 12938 3/7/2014 I
NAPHYRONE** 03-04-16 81 FR 11429 3/4/2016 I
N-BENZYLPIPERAZINE (BZP) 09-08-03 03-18-04 69 FR 12794 3/18/2004 I
N-BENZYLPIPERAZINE (BZP) * 09-20-02 67 FR 59161 9/20/2002 I
N-BENZYLPIPERAZINE (BZP) ** 09-10-03 68 FR 53289 9/20/2003 I
N-ETHYLAMPHETAMINE 09-10-81 12-08-81 46 FR 59969 1/7/1982 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE* 10-15-87 52 FR 38225 10/15/1987 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE** 10-13-88 53 FR 40061 10/13/1988 I
NIMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NORDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ORIPAVINE 09-24-07 72 FR 54208 9/24/2007 II
ORTHO-FLUOROFENTANYL OR 2-FLUOROFENTANYL (N-(2- 10-26-17 82 FR 49504 10/26/2017 I FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4-YL))*
OXAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
OXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
Scheduling Actions - Alphabetical Order
01-Mar-18 Page 8 of 10
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SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
PARA-FLUOROFENTANYL 03-10-87 05-29-87 52 FR 20070 5/29/1987 I
PARA-FLUOROFENTANYL* 02-07-86 51 FR 4722 3/10/1986 I
PARA-FLUOROFENTANYL** 03-10-87 52 FR 7270 3/10/1987 I
PARAHEXYL 08-05-82 11-22-82 47 FR 52432 12/22/1982 I
PCC (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
PCE (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PCH (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
PEMOLINE 11-07-74 01-28-75 40 FR 4150 1/28/1975 IV
PENTAZOCINE 09-13-78 01-10-79 44 FR 2169 2/9/1979 IV
PENTEDRONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
PENTEDRONE* 03-07-14 79 FR 12938 3/7/2014 I
PENTEDRONE** 03-04-16 81 FR 11429 3/4/2016 I
PENTOBARBITAL 05-31-75 11-13-73 38 FR 31310 11/13/1973 III -> II
PENTYLONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
PENTYLONE* 03-07-14 79 FR 12938 3/7/2014 I
PENTYLONE** 03-04-16 81 FR 11429 3/4/2016 I
PEPAP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I
PEPAP* 07-10-85 50 FR 28098 8/12/1985 I
PEPAP** 08-11-86 51 FR 28695 8/12/1986 I
PERAMPANEL [2-(2-OXO-1-PHENYL- 10-22-13 12-02-13 78 FR 72013 1/2/2014 III 5-PYRIDIN-2-YL-l ,2-DIHYDROPYRIDIN-3-YL)BENZONITRILE ]
PHENCYCLIDINE (PCP) 12-19-77 01-25-78 43 FR 3359 2/24/1978 III -> II
PHENDIMETRAZINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
PHENMETRAZINE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
PHENTERMINE 05-09-73 07-06-73 38 FR 18013 7/6/1973 IV
PHENYLACETONE (P2P) 12-12-79 44 FR 71822 2/11/1980 II
PHP (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PINAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
PIPRADROL 09-30-80 45 FR 64570 12/1/1980 IV
PRAZEPAM 07-29-76 12-17-76 41 FR 55176 12/17/1976 IV
PREGABALIN 05-12-05 07-28-05 70 FR 43633 7/28/2005 V
PROPIRAM 01-29-72 37 FR 1468 1/29/1972 I
PROPYLHEXEDRINE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
PROPYLHEXEDRINE 12-03-91 56 FR 61372 12/3/1991 V -> 0
PROSTANOZOL (17 BETA-HYDROXY-5 ALPHA- 11-23-11 07-30-12 77 FR 44456 8/29/2012 III ANDROSTANO[3,2-C]PRYAZOLE
PYROVALERONE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
QUAZEPAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 02-10-14 79 FR 7577 2/10/2014 I CARBOXYLATE ( 5-FLUORO-PB22; 5FPB22)*
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 02-05-16 81 FR 6175 2/5/2016 I CARBOXYLATE ( 5-FLUORO-PB22; 5FPB22)**
Scheduling Actions - Alphabetical Order
01-Mar-18 Page 9 of 10
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SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3-CARBOXYLATE (5-FLUORO-PB-22; 5F-PB-22)
09-06-16 81 FR 61130 9/6/2016 I
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE 02-05-16 81 FR 6175 2/5/2016 I (PB22; QUPIC)**
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE 02-10-14 79 FR 7577 2/10/2014 I (PB22; QUPIC)*
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE (PB- 09-06-16 81 FR 61130 9/6/2016 I 22; QUPIC)
REMIFENTANIL 09-16-96 11-05-96 61 FR 56893 11/5/1996 II
SECOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
SIBUTRAMINE 12-08-97 02-11-98 63 FR 6862 2/11/1998 IV
SPA (LEFETAMINE) 09-30-80 45 FR 64570 12/1/1980 IV
SUFENTANIL 03-20-84 05-25-84 49 FR 22074 5/25/1984 I -> II
SUFENTANIL 09-30-80 45 FR 64571 12/1/1980 I
SUVOREXANT 02-13-14 08-28-14 79 FR 52143 9/29/2014 IV
TAPENTADOL 02-17-09 05-21-09 74 FR 23790 6/22/2009 II
TCP (PCP ANALOG) 05-29-75 07-08-75 40 FR 28611 8/11/1975 I
TEMAZEPAM 01-05-81 04-07-81 45 FR 20671 4/7/1981 IV
TETRAHYDROFURANYL FENTANYL (N-(1- 10-26-17 82 FR 49504 10/26/2017 I PHENETHYLPIPERIDIN-4-YL)-N-PHENYLTETRAHYDROFURAN-2-CARBOXAMIDE)*
TETRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
THENYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I Expired 11/29/86
THIAFENTANIL 08-26-16 81 FR 58834 8/26/2016 II
THIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
THIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
THIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
TILETAMINE/ZOLAZEPAM (TELAZOL) 08-11-86 01-21-87 52 FR 2221 2/20/1987 III
TILIDINE 09-30-80 45 FR 64571 1/12/1980 I
TRAMADOL (2-[(DIMETHYLAMINO)METHYL]-1-(3- 11-04-13 07-02-14 79 FR 37623 8/18/2014 IV METHOXYPHENYL)CYCLOHEXANOL)
TRIAZOLAM 04-29-81 12-28-82 47 FR 57694 12/28/1982 IV
ZALEPLON 05-05-99 09-15-99 64 FR 49982 9/15/1999 IV
ZOLPIDEM 11-24-92 02-05-93 58 FR 7186 2/5/1993 IV
ZOPICLONE 02-14-05 04-04-05 70 FR 16935 4/4/2005 IV
Scheduling Actions - Alphabetical Order
01-Mar-18 Page 10 of 10
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Scheduling Actions C
hronological Order
-
Scheduling Actions
- Chronological Order -
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
AMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
METHAMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
FETAMIN 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
BIPHETAMINE & BIPHETAMINE-T 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
ESKATROL 05-26-71 08-18-71 36 FR 15744 8/18/1971 III -> II
NALOXONE HYDROCHLORIDE 08-19-71 09-29-71 36 FR 19116 9/29/1971 II -> 0
METHYLPHENIDATE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
PHENMETRAZINE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
PROPIRAM 01-29-72 37 FR 1468 1/29/1972 I
MAZINDOL 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
PHENDIMETRAZINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CLORTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CHLORPHENTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
BENZPHETAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
FENFLURAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 IV
PHENTERMINE 05-09-73 07-06-73 38 FR 18013 7/6/1973 IV
DIETHYLPROPION 05-10-73 07-06-73 38 FR 18013 7/6/1973 IV
DROTEBANOL 07-03-73 38 FR 17717 8/6/1973 I
4-METHOXYAMPHETAMINE (PMA) 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
4-BROMO-2,5-DIMETHOXYAMPHETAMINE 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
2,5-DIMETHOXYAMPHETAMINE (DMA) 05-31-73 09-21-73 38 FR 26447 9/21/1973 I
METHAQUALONE 04-11-73 10-04-73 38 FR 27516 10/4/1973 II
PENTOBARBITAL 05-31-75 11-13-73 38 FR 31310 11/13/1973 III -> II
SECOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
AMOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
ETORPHINE HYDROCHLORIDE 11-23-73 03-29-74 39 FR 11535 4/19/1974 I -> II
NALOXONE 07-10-74 12-24-74 39 FR 44392 12/24/1974 II -> 0
PEMOLINE 11-07-74 01-28-75 40 FR 4150 1/28/1975 IV
MEBUTAMATE 12-13-74 01-30-75 40 FR 4418 1/30/1975 IV
CONCENTRATE OF POPPY STRAW 12-20-74 02-14-75 40 FR 6779 2/14/1975 II
NALTREXONE 12-09-74 03-06-75 40 FR 10455 3/6/1975 II -> 0
DIFENOXIN 05-07-75 40 FR 19813 6/1/1975 I
Scheduling Actions - Chronological Order
01-Mar-18 Page 1 of 11
-
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
CLORAZEPATE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
FLURAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
DIAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CHLORDIAZEPOXIDE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
OXAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CLONAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
MECLOQUALONE 05-29-75 07-08-75 40 FR 28611 7/10/1975 I
TCP (PCP ANALOG) 05-29-75 07-08-75 40 FR 28611 8/11/1975 I
MENRIUM 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted RX
LIBRAX 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted RX
APOMORPHINE 04-08-76 06-28-76 41 FR 26568 6/28/1976 II -> 0
NALBUPHINE 05-11-76 10-01-76 41 FR 43401 10/1/1976 II -> 0
DEXTRORPHAN 04-19-76 10-01-76 41 FR 43401 10/1/1976 I -> 0
PRAZEPAM 07-29-76 12-17-76 41 FR 55176 12/17/1976 IV
DEXTROPROPOXYPHENE 09-29-76 02-11-77 42 FR 8636 3/14/1977 IV
LOPERAMIDE 07-29-76 05-18-77 42 FR 25498 6/17/1977 V
LORAZEPAM 06-28-77 10-07-77 42 FR 54546 10/3/1977 IV
PHENCYCLIDINE (PCP) 12-19-77 01-25-78 43 FR 3359 2/24/1978 III -> II
PCC (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
PCH (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
DIFENOXIN 1/2 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> V
DIFENOXIN 1 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> IV
PHP (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PCE (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PENTAZOCINE 09-13-78 01-10-79 44 FR 2169 2/9/1979 IV
TILIDINE 09-30-80 45 FR 64571 1/12/1980 I
PHENYLACETONE (P2P) 12-12-79 44 FR 71822 2/11/1980 II
DEXTROPROPOXYPHENE 01-21-80 06-24-80 45 FR 42264 7/24/1980 IV
DEXTROPROPOXYPHENE (BULK) 07-22-80 45 FR 48881 9/22/1980 IV -> II
PIPRADROL 09-30-80 45 FR 64570 12/1/1980 IV
SPA (LEFETAMINE) 09-30-80 45 FR 64570 12/1/1980 IV
SUFENTANIL 09-30-80 45 FR 64571 12/1/1980 I
TEMAZEPAM 01-05-81 04-07-81 45 FR 20671 4/7/1981 IV
FENETHYLLINE 05-01-81 07-21-81 46 FR 37503 8/20/1981 I
ALPHA-METHYLFENTANYL 08-05-81 09-22-81 46 FR 46799 9/22/1981 I
HALAZEPAM 04-29-81 10-29-81 46 FR 53407 10/29/1981 IV
ALPRAZOLAM 04-29-81 11-12-81 46 FR 55688 11/12/1981 IV
Scheduling Actions - Chronological Order
01-Mar-18 Page 2 of 11
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FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
MAZINDOL 04-17-81 10-27-81 46 FR 52333 11/27/1981 III -> IV
N-ETHYLAMPHETAMINE 09-10-81 12-08-81 46 FR 59969 1/7/1982 I
LOPERAMIDE 07-28-82 11-03-82 47 FR 49840 11/3/1982 V -> 0
PARAHEXYL 08-05-82 11-22-82 47 FR 52432 12/22/1982 I
TRIAZOLAM 04-29-81 12-28-82 47 FR 57694 12/28/1982 IV
SUFENTANIL 03-20-84 05-25-84 49 FR 22074 5/25/1984 I -> II
ALFENTANIL 06-25-84 49 FR 25849 8/24/1984 I
METHAQUALONE 08-27-84 49 FR 33870 8/27/1984 II -> I
ESTAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LORMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
MEDAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
BROMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
HALOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOBAZAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOTIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LOPRAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NORDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
OXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLUNITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
KETAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
PINAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CAMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NIMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ETHYL LOFLAZEPATE 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLUDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
DELORAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
TETRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
BUPRENORPHINE 09-20-82 02-28-85 50 FR 8104 4/1/1985 II -> V
3-METHYLFENTANYL* 03-25-85 50 FR 11690 4/25/1985 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE)* 05-31-85 50 FR 23118 7/1/1985 I
MPPP* 07-10-85 50 FR 28098 8/12/1985 I
PEPAP* 07-10-85 50 FR 28098 8/12/1985 I
NALMEFENE 05-31-85 11-04-85 50 FR 45815 11/4/1985 II -> 0
BETA-HYDROXY-3-METHYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
BETA-HYDROXYFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
THIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
Scheduling Actions - Chronological Order
01-Mar-18 Page 3 of 11
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FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
BENZYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I Expired 11/29/86
3-METHYLTHIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
ALPHA-METHYLTHIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
ACETYL-ALPHA-METHYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
THENYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I Expired 11/29/86
PARA-FLUOROFENTANYL* 02-07-86 51 FR 4722 3/10/1986 I
QUAZEPAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
MIDAZOLAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
3-METHYLFENTANYL** 04-24-86 51 FR 15474 4/25/1986 I
DRONABINOL PRODUCT (MARINOL) 10-18-85 05-13-86 51 FR 17476 5/13/1986 I -> II
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE)** 06-17-86 51 FR 21911 7/1/1986 I
PEPAP** 08-11-86 51 FR 28695 8/12/1986 I
MPPP** 08-11-86 51 FR 28695 8/12/1986 I
3-METHYLFENTANYL 04-24-86 09-22-86 51 FR 33592 9/22/1986 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 07-27-84 10-14-86 51 FR 36552 11/13/1986 I
ACETYL-ALPHA-METHYLFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
3-METHYLTHIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
BETA-HYDROXYFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
BETA-HYDROXY-3-METHYLFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I Expired 5/29/87
ALPHA-METHYLTHIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
THIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
MPPP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I
PEPAP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I
ALFENTANIL 04-17-86 01-23-87 52 FR 2516 1/23/1987 I -> II
TILETAMINE/ZOLAZEPAM (TELAZOL) 08-11-86 01-21-87 52 FR 2221 2/20/1987 III
PARA-FLUOROFENTANYL** 03-10-87 52 FR 7270 3/10/1987 I
NABILONE 06-18-86 04-07-87 52 FR 11042 4/7/1987 II
ALPHA-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
BETA-HYDROXYFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
3-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
ACETYL-ALPHA-METHYLFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
PARA-FLUOROFENTANYL 03-10-87 05-29-87 52 FR 20070 5/29/1987 I
THIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
4-METHYLAMINOREX* 10-15-87 52 FR 38225 10/15/1987 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE* 10-15-87 52 FR 38225 10/15/1987 I
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE* 10-15-87 52 FR 38225 10/15/1987 I
Scheduling Actions - Chronological Order
Page 4 of 11 01-Mar-18
-
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
BETA-HYDROXY-3-METHYLFENTANYL 11-28-86 01-08-88 53 FR 500 1/8/1988 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 01-27-88 53 FR 2225 1/27/1988 I -> 0
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 02-22-88 53 FR 5156 3/23/1988 I
PYROVALERONE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
PROPYLHEXEDRINE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
CATHINE 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENCAMFAMIN 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENPROPOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
MEFENOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
N,N-DIMETHYLAMPHETAMINE* 08-03-88 53 FR 29232 8/3/1988 I
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE** 10-13-88 53 FR 40061 10/13/1988 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE** 10-13-88 53 FR 40061 10/13/1988 I
4-METHYLAMINOREX** 10-13-88 53 FR 40061 10/13/1988 I
CARFENTANIL 01-12-88 10-28-88 53 FR 43684 10/28/1988 II
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
4-METHYLAMINOREX 10-14-88 04-13-89 54 FR 14799 4/13/1989 I
1-[1-(2-THIENYL)CYCLOHEXYL]PYRROLIDINE 03-20-89 07-06-89 54 FR 28414 7/6/1989 I
N,N-DIMETHYLAMPHETAMINE** 08-02-89 54 FR 31815 8/2/1989 I
N,N-DIMETHYLAMPHETAMINE 08-02-89 02-02-90 55 FR 3586 2/2/1990 I
ANABOLIC STEROIDS PL 101-647 02-13-91 56 FR 5753 2/27/1991 III
GLUTETHIMIDE 07-26-90 03-21-91 56 FR 11930 3/21/1991 III -> II
PROPYLHEXEDRINE 12-03-91 56 FR 61372 12/3/1991 V -> 0
METHCATHINONE* 05-01-92 57 FR 18824 5/1/1992 I
BUTORPHANOL, THEBAINE DERIVED 04-03-92 07-14-92 57 FR 31126 7/14/1992 II->0 Supersede
d 10/97
AMINOREX* 09-21-92 57 FR 43399 9/21/1992 I
ZOLPIDEM 11-24-92 02-05-93 58 FR 7186 2/5/1993 IV
CATHINONE 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
2,5-DIMETHOXY-4-ETHYLAMPHETAMINE (DOET) 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
ALPHA-ETHYLTRYPTAMINE* 03-12-93 58 FR 13533 3/12/1993 I
METHCATHINONE** 04-29-93 58 FR 25934 5/1/1993 I
LEVO-ALPHACETYLMETHADOL (LAAM) 04-28-93 08-18-93 58 FR 43795 8/18/1993 I -> II
AMINOREX** 08-24-93 58 FR 44611 9/21/1993 I
METHCATHINONE 04-28-93 10-15-93 58 FR 53404 10/15/1993 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE* 01-06-94 59 FR 00671 1/6/1994 I
ALPHA-ETHYLTRYPTAMINE** 03-07-94 59 FR 10720 3/12/1994 I
Scheduling Actions - Chronological Order
Page 5 of 11 01-Mar-18
-
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
AMINOREX 08-20-93 03-18-94 59 FR 12828 3/18/1994 I
ALPHA-ETHYLTRYPTAMINE 03-07-94 09-12-94 59 FR 46757 9/12/1994 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE** 12-21-94 59 FR 65710 1/6/1995 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE 12-20-94 06-02-95 60 FR 28718 6/2/1995 I
REMIFENTANIL 09-16-96 11-05-96 61 FR 56893 11/5/1996 II
FENFLURAMINE 05-06-97 05-06-97 5/6/1997 IV -> 0
BUTORPHANOL 07-10-97 10-01-97 62 FR 51370 10/31/1997 IV
SIBUTRAMINE 12-08-97 02-11-98 63 FR 6862 2/11/1998 IV
MODAFINIL 04-14-98 01-27-99 64 FR 4050 1/27/1999 IV
DRONABINOL PRODUCT (MARINOL) 11-05-98 07-02-99 64 FR 35928 7/2/1999 II -> III
KETAMINE 04-09-99 07-13-99 64 FR 37673 8/12/1999 III
ZALEPLON 05-05-99 09-15-99 64 FR 49982 9/15/1999 IV
GAMMA HYDROXYBUTYRIC ACID (GHB) PL 106-172 03-13-00 65 FR 13235 3/13/2000 I
GAMMA HYDROXYBUTYRIC ACID (GHB) FDA approved drug PL 106-172 03-13-00 65 FR 13235 3/13/2000 III products
DIHYDROETORPHINE (thebaine derivative) 11-17-00 65 FR 69442 11/17/2000 clarification of CII control
DICHLORALPHENAZONE (chloral hydrate compound) 12-11-00 08-16-01 66 FR 42943 8/16/2001 clarification of CIV control
N-BENZYLPIPERAZINE (BZP) * 09-20-02 67 FR 59161 9/20/2002 I
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) * 09-20-02 67 FR 59161 9/20/2002 I
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-20-02 67 FR 59163 9/20/2002 I T-7) *
BUPRENORPHINE 03-21-02 10-07-02 67 FR 62354 10/7/2002 V --> III
ALPHA-METHYLTRYPTAMINE (AMT) * 04-04-03 68 FR 16427 4/4/2003 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) * 04-04-03 68 FR 16427 4/4/2003 I
FENFLURAMINE 05-15-03 68 FR 26247 5/15/2003 IV Withdrew
97 proposed
rule
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-10-03 68 FR 53289 9/20/2003 I T-7) **
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) ** 09-10-03 68 FR 53289 9/20/2003 I
N-BENZYLPIPERAZINE (BZP) ** 09-10-03 68 FR 53289 9/20/2003 I
N-BENZYLPIPERAZINE (BZP) 09-08-03 03-18-04 69 FR 12794 3/18/2004 I
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-08-03 03-18-04 69 FR 12794 3/18/2004 I T-7)
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) 09-08-03 03-18-04 69 FR 12794 3/19/2004 I --> 0
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) **
04-01-04 69 FR 17034 4/1/2004 I
Scheduling Actions - Chronological Order
Page 6 of 11 01-Mar-18
-
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
ALPHA-METHYLTRYPTAMINE (AMT) ** 04-01-04 69 FR 17034 4/1/2004 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) 09-29-04 69 FR 58050 9/29/2004 I
ALPHA-METHYLTRYPTAMINE (AMT) 09-29-04 69 FR 58050 9/29/2004 I
ZOPICLONE 02-14-05 04-04-05 70 FR 16935 4/4/2005 IV
PREGABALIN 05-12-05 07-28-05 70 FR 43633 7/28/2005 V
ANABOLIC STEROIDS PL 108-358 12-16-05 70 FR 74653 1/17/2006 III
EMBUTRAMIDE 07-29-05 08-29-06 71 FR 51115 9/28/2006 III
LISDEXAMFETAMINE 02-22-07 05-03-07 72 FR 24532 6/4/2007 II
ORIPAVINE 09-24-07 72 FR 54208 9/24/2007 II
INDIPLON 01-31-08 01-31-08 1/31/2008 IV
LACOSAMIDE 03-10-09 05-21-09 74 FR 23789 6/22/2009 V
TAPENTADOL 02-17-09 05-21-09 74 FR 23790 6/22/2009 II
FOSPROPOFOL 07-23-09 10-06-09 74 FR 51234 11/5/2009 IV
19-NOR-4,9(10)-ANDROSTADIENEDIONE (estra-4,9(10)-diene- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III 3,17-dione)
BOLDIONE (Androsta-1,4-diene-3,17-dione) 04-25-08 12-04-09 74 FR 63603 1/4/2010 III
DESOXYMETHYLTESTOSTERONE (17a-methyl-5a-androst-2- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III en-17-ol, madol)
4-ANILINO-N-PHENETHYL-4-PIPERIDINE (ANPP) 04-09-08 06-29-10 75 FR 37296 8/30/2010 II
5-METHOXY-N,N-DIMETHYLTRYPTAMINE 08-21-09 12-20-10 75 FR 79296 1/19/2011 I
CP-47,497 * 03-01-11 76 FR 11075 3/1/2011 I
CP-47,497 C8 HOMOLOGUE * 03-01-11 76 FR 11075 3/1/2011 I
JWH-073 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-018 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-200 * 03-01-11 76 FR 11075 3/1/2011 I
3,4-METHYLENEDIOXYPYROVALERONE (MDPV)* 10-21-11 76 FR 65371 10/21/2011 I
4-METHYL-N-METHYLCATHINONE (MEPHEDRONE)* 10-21-11 76 FR 65371 10/21/2011 I
3,4-METHYLENEDIOXY-N-METHYLCATHINONE 10-21-11 76 FR 65371 10/21/2011 I (METHYLONE)*
EZOGABINE 10-21-11 12-15-11 76 FR 77895 12/15/2011 V
CARISOPRODOL 11-17-09 12-12-11 76 FR 77330 1/11/2012 IV
JWH-018 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-073 ** 02-29-12 77 FR 12201 2/29/2012 I
CP-47,497 C8 HOMOLOGUE ** 02-29-12 77 FR 12201 2/29/2012 I
CP-47,497 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-200 ** 02-29-12 77 FR 12201 2/29/2012 I
METHASTERONE ( 2 ALPHA-17 ALPHA-DIMETHYL-5 ALPHA- 11-23-11 07-30-12 77 FR 44456 8/29/2012 III ANDROSTAN-17BETA-OL-3-ONE)
PROSTANOZOL (17 BETA-HYDROXY-5 ALPHA- 11-23-11 07-30-12 77 FR 44456 8/29/2012 III ANDROSTANO[3,2-C]PRYAZOLE
Scheduling Actions - Chronological Order
Page 7 of 11 01-Mar-18
-
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
3,4-METHYLENEDIOXY-N-METHYLCATHINONE (METHYLONE)
10-21-11 04-12-13 78 FR 21818 4/12/2013 I
(1-PENTYL-1H-INDOL-3-YL)(2,2,3,3-TETRAMETHYLCYCLOPROPYL)METHANONE (UR-144)*
05-16-13 78 FR 28735 5/16/2013 I
[1-(5-FLUORO-PENTYL)1H-INDOL-3-YL](2,2,3,3-TETRAMETHYLCYCLOPROPYL)METHANONE(5-FLUORO-UR-144, XLR11)*
05-16-13 78 FR 28735 5/16/2013 I
N-(1-ADAMANTYL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (APINACA, AKB48)*
05-16-13 78 FR 28735 5/16/2013 I
LORCASERIN 12-19-12 05-08-13 78 FR 26701 6/7/2013 IV
2-(4-IODO-2,5-DIMETHOXYPHENYL)-N-(2-METHOXYBENZYL) ETHANAMINE (25I-NBOMe)*
11-15-13 78 FR 68716 11/15/2013 I
2-(4-CHLORO-2,5-DIMETHOXYPHENYL)-N-(2-METHOXYBENZYL) ETHANAMINE (25C-NBOMe)*
11-15-13 78 FR 68716 11/15/2013 I
2-(4-BROMO-2,5-DIMETHOXYPHENYL)-N-(2-METHOXYBENZYL) ETHANAMINE (25B-NBOMe)*
11-15-13 78 FR 68716 11/15/2013 I
PERAMPANEL [2-(2-OXO-1-PHENYL-5-PYRIDIN-2-YL-l ,2-DIHYDROPYRIDIN-3-YL)BENZONITRILE ]
10-22-13 12-02-13 78 FR 72013 1/2/2014 III
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3-CARBOXYLATE ( 5-FLUORO-PB22; 5FPB22)*
02-10-14 79 FR 7577 2/10/2014 I
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE (PB22; QUPIC)*
02-10-14 79 FR 7577 2/10/2014 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE FUBINACA)*
(AB-02-10-14 79 FR 7577 2/10/2014 I
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)*
02-10-14 79 FR 7577 2/10/2014 I
ALPHA-PYRROLIDINOBUTIOPHENONE (-PBP)* 03-07-14 79 FR 12938 3/7/2014 I
PENTYLONE* 03-07-14 79 FR 12938 3/7/2014 I
PENTEDRONE* 03-07-14 79 FR 12938 3/7/2014 I
NAPHYRONE* 03-07-14 79 FR 12938 3/7/2014 I
ALPHA-PYRROLIDINOPENTIOPHENONE (-PVP)* 03-07-14 79 FR 12938 3/7/2014 I
4-METHYL-N-ETHYLCATHINONE (4-MEC)* 03-07-14 79 FR 12938 3/7/2014 I
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4-MePPP)*
03-07-14 79 FR 12938 3/7/2014 I
4-FLUORO-N-METHYLCATHINONE (4-FMC)* 03-07-14 79 FR 12938 3/7/2014 I
3-FLUORO-N-METHYLCATHINONE (3-FMC)* 03-07-14 79 FR 12938 3/7/2014 I
BUTYLONE* 03-07-14 79 FR 12938 3/7/2014 I
ALFAXALONE (5-PREGNAN-3-OL-11,20-DIONE) 03-25-13 02-27-14 79 FR 10985 3/31/2014 IV
TRAMADOL (2-[(DIMETHYLAMINO)METHYL]-1-(3-METHOXYPHENYL)CYCLOHEXANOL)
11-04-13 07-02-14 79 FR 37623 8/18/2014 IV
SUVOREXANT 02-13-14 08-28-14 79 FR 52143 9/29/2014 IV
HYDROCODONE COMBINATION PRODUCTS 02-27-14 08-22-14 79 FR 49661 10/6/2014 III->II
NALOXEGEL 10-29-14 01-23-15 80 FR 3468 1/23/2015 II->0
Scheduling Actions - Chronological Order
Page 8 of 11 01-Mar-18
-
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
[1-(5-FLUOROPENTYL)-1H-INDAZOL-3-YL](NAPHTHALEN-1-YL)METHANONE (THJ-2201)*
01-30-15 80 FR 5042 1/30/2015 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (AB-PINACA)*
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)1-(CYCLOHEXYLMETHYL) 1H-INDAZOLE-3-CARBOXAMIDE (AB-CHMINACA)*
ACETYL FENTANYL* (N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLACETAMIDE)
ELUXADOLINE
N-(1-AMINO-3,3DIMETHYL-1-OXOBUTAN-2-YL)1-(CYCLOHEXYLMETHYL)-1H-INDAZOLE-3CARBOXAMIDE (MAB-CHMINACA)*
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (AB-FUBINACA)**
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3-CARBOXYLATE ( 5-FLUORO-PB22; 5FPB22)**
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE (PB22; QUPIC)**
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)**
3-FLUORO-N-METHYLCATHINONE (3-FMC)**
PENTYLONE**
PENTEDRONE**
ALPHA-PYRROLIDINOPENTIOPHENONE (-PVP)**
ALPHA-PYRROLIDINOBUTIOPHENONE (-PBP)**
4-METHYL-N-ETHYLCATHINONE (4-MEC)**
4-FLUORO-N-METHYLCATHINONE (4-FMC)**
BUTYLONE**
NAPHYRONE**
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4-MePPP)**
BRIVARACETAM (BRV; UCB-34714; BRIVIACT)
BUTYRYL FENTANYL*
BETA-HYDROXYTHIOFENTANYL*
3,4-DICHLORO-N-[(1-DIMETHYLAMINO)CYCLOHEXYLMETHYL]BENZAMIDE) (AH-7921)
THIAFENTANIL
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE (PB-22; QUPIC)
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3-CARBOXYLATE (5-FLUORO-PB-22; 5F-PB-22)
08-11-15
01-30-15
01-30-15
07-17-15
11-12-15
02-05-16
02-05-16
02-05-16
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05-12-16
04-14-16
08-26-16
09-06-16
09-06-16
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80 FR 5042
80 FR 42381
80 FR 69861
81 FR 6171
81 FR 6175
81 FR 6175
81 FR 6175
81 FR 6175
81 FR 11429
81 FR 11429
81 FR 11429
81 FR 11429
81 FR 11429
81 FR 11429
81 FR 11429
81 FR 11429
81 FR 11429
81 FR 11429
81 FR 29487
81 FR 29492
81 FR 29492
81 FR 22023
81 FR 58834
81 FR 61130
81 FR 61130
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1/30/2015
7/17/2015
12/17/2015
2/5/2016
2/5/2016
2/5/2016
2/5/2016
2/5/2016
3/4/2016
3/4/2016
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3/4/2016
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3/4/2016
3/4/2016
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Scheduling Actions - Chronological Order
01-Mar-18 Page 9 of 11
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FINAL ORDER
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FEDERAL
REGISTER
CITATION EFFECTIVE
DATE
CSA
SCHEDULE
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (AB-FUBINACA)
09-06-16 81 FR 61130 9/6/2016 I
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)
09-06-16 81 FR 61130 9/6/2016 I
3,4-DICHLORO-N-[2-(DIMETHYLAMINO)CYCLOHEXYL]-N-METHYLBENZAMIDE (U-47700)*
11-14-16 81 FR 79389 11/14/2016 I
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLFURAN-2-CARBOXAMIDE (FURANYL FENTANYL) *
11-29-16 81 FR 85873 11/29/2016 I
3-FLUORO-N-METHYLCATHINONE (3-FMC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
NAPHYRONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
4-FLUORO-N-METHYLCATHINONE (4-FMC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4-MePPP)
03-04-16 03-01-17 82 FR 12171 3/1/2017 I
BUTYLONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
PENTEDRONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
PENTYLONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
ALPHA-PYRROLIDINOPENTIOPHENONE (-PVP) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
4-METHYL-N-ETHYLCATHINONE (4-MEC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
ALPHA-PYRROLIDINOBUTIOPHENONE (-PBP) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
DRONABINOL IN ORAL SOLUTION IN DRUG PRODUCT APPROVED FOR MARKETING BY U.S. FOOD AND DRUG ADMIN.
03-23-17 82 FR 14815 3/23/2017 II
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)1H-INDAZOLE-3-CARBOXAMIDE (ADBFUBINACA)*
04-10-17 82 FR 17119 4/10/2017 I
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3-CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-CHMICA)*
04-10-17 82 FR 17119 4/10/2017 I
N-(ADAMANTAN-1-YL)-1-(5-FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDE (5FAPINACA, 5FAKB48)*
04-10-17 82 FR 17119 4/10/2017 I
METHYL2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3-METHYLBUTANOATE (5F-AMB)*
04-10-17 82 FR 17119 4/10/2017 I
METHYL2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-ADB)*
04-10-17 82 FR 17119 4/10/2017 I
METHYL 2-(1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMBFUBINACA)*
04-10-17 82 FR 17119 4/10/2017 I
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4-YL)ISOBUTYRAMIDE (4-FLUOROISOBUTYRYL FENTANYL)*
05-03-17 82 FR 20544 5/3/2017 I
ACETYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLACETAMIDE)
06-07-17 82 FR 26349 6/7/2017 I
ACRYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLACRYLAMIDE)*
07-14-17 82 FR 32453 7/14/2017 I
ORTHO-FLUOROFENTANYL OR 2-FLUOROFENTANYL (N-(2-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4-YL))*
10-26-17 82 FR 49504 10/26/2017 I
Scheduling Actions - Chronological Order
Page 10 of 11 01-Mar-18
-
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
TETRAHYDROFURANYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLTETRAHYDROFURAN-2-CARBOXAMIDE)*
10-26-17 82 FR 49504 10/26/2017 I
METHOXYACETYL FENTANYL (2-METHOXY-N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLACETAMIDE)*
10-26-17 82 FR 49504 10/26/2017 I
FUBAMB, MMB FUBINACA (2-(1-(4-FLUOROBENZYL)-1HINDAZOLE-3-CARBOXAMIDO)-3- METHYLBUTANOATE*
11-03-17 82 FR 51154 11/3/2017 I
CYCLOPROPYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLCYCLOPROPANECARBOXAMIDE)*
01-04-18 83 FR 469 1/4/2018 I
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLPENTANAMIDE (VALERYL FENTANYL)*
02-01-18 83 FR 4580 2/1/2018 I
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4-YL)BUTYRAMIDE (PARA-FLUOROBUTYRYL FENTANYL)*
02-01-18 83 FR 4580 2/1/2018 I
N-(4-METHOXYPHENYL)-N-(1-PHENETHYLPIPERIDIN-4-YL)BUTYRAMIDE (PARA-METHOXYBUTYRYL FENTANYL)*
02-01-18 83 FR 4580 2/1/2018 I
N-(4-CHLOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4-YL)ISOBUTYRAMIDE (PARA-CHLOROISOBUTYRYL FENTANYL)*
02-01-18 83 FR 4580 2/1/2018 I
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLISOBUTYRAMIDE (ISOBUTYRYL FENTANYL)*
02-01-18 83 FR 4580 2/1/2018 I
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLCYCLOPENTANECARBOXAMIDE (CYCLOPENTYL FENTANYL)*
02-01-18 83 FR 4580 2/1/2018 I
N-(2-FLUOROPHENYL)-2-METHOXY-N-(1-PHENETHYLPIPERIDIN-4-YL)ACETAMIDE (OCFENTANIL)*
02-01-18 83 FR 4580 2/1/2018 I
FENTANYL-RELATED SUBSTANCES, AS DEFINED IN 21 CFR 1308.11(h)*
02-06-18 83 FR 5188 2/6/2018 I
Scheduling Actions - Chronological Order
Page 11 of 11 01-Mar-18
-
Controlled Substances
Alphabetical O
rder
-
Controlled Substances
- Alphabetical Order -
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
-6-bromo-androsta-1,4-diene-3,17-dione 4000 III N
[3,2-c]-furazan-5-androstan-17-ol 4000 III N
[3,2-c]pyrazole-androst-4-en-17-ol 4000 III N
1-(1-Phenylcyclohexyl)pyrrolidine 7458 I N PCPy, PHP, rolicyclidine
1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine 9663 I Y PEPAP, synthetic heroin
1-[1-(2-Thienyl)cyclohexyl]piperidine 7470 I N TCP, tenocyclidine
1-[1-(2-Thienyl)cyclohexyl]pyrrolidine 7473 I N TCPy
13Beta-ethyl-17beta-hydroxygon-4-en-3-one 4000 III N
17Alpha-methyl-3alpha,17beta-dihydroxy-5alpha- 4000 III N
androstane
17Alpha-methyl-3beta,17beta-dihydroxy-5alpha- 4000 III N
androstane
17Alpha-methyl-3beta,17beta-dihydroxyandrost-4-ene 4000 III N
17Alpha-methyl-4-hydroxynandrolone (17alpha-methyl- 4000 III N
4-hydroxy-17beta-hydroxyestr-4-en-3-one)
17Alpha-methyl-delta1-dihydrotestosterone (17beta- 4000 III N 17-Alpha-methyl-1-testosterone hydroxy-17alpha-methyl-5alpha-androst-1-en-3-one)
17-Methyl-5-androstan-17-ol 4000 III N
17-methyl-androst-2-ene-3,17-diol 4000 III N
17-methyl-androsta-1,4-diene-3,17-diol 4000 III N
17-Methyl-androstan-3-hydroxyimine-17-ol 4000 III N
17-Hydroxy-androstano[2,3-d]isoxazole 4000 III N
17-Hydroxy-androstano[3,2-c]isoxazole 4000 III N
18a-Homo-3-hydroxy-estra-2,5(10)-dien-17-one 4000 III N
19-Nor-4,9(10)-androstadienedione 4000 III N
19-Nor-4-androstenediol (3beta,17beta-dihydroxyestr-4- 4000 III N
ene; 3alpha,17beta-dihydroxyestr-4-ene)
19-Nor-4-androstenedione (estr-4-en-3,17-dione) 4000 III N
19-Nor-5-androstenediol (3beta,17beta-dihydroxyestr-5- 4000 III N
ene; 3alpha,17beta-dihydroxyestr-5-ene)
19-Nor-5-androstenedione (estr-5-en-3,17-dione) 4000 III N
1-Androstenediol (3beta,17beta-dihydroxy-5alpha- 4000 III N
androst-1-ene; 3alpha,17beta-dihydroxy-5alpha-androst-1-ene)
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
01-Mar-18 Page 1 of 16
-
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
1-Androstenedione (5alpha-androst-1-en-3,17-dione) 4000 III N
1-Methyl-4-phenyl-4-propionoxypiperidine 9661 I Y MPPP, synthetic heroin
1-Phenylcyclohexylamine 7460 II N PCP precursor
1-Piperidinocyclohexanecarbonitrile 8603 II N PCC, PCP precursor
2-(1-(4-fluorobenzyl)-1Hindazole-3-carboxamido)-3- 7021 I N FUBAMB, MMB FUBINACA, AMBFUBINACA methylbutanoate
2-(2,5-Dimethoxy-4-(n)-propylphenyl) ethanamine (2C- 7524 I N 2C-P P)
2-(2,5-Dimethoxy-4-ethylphenyl) ethanamine (2C-E ) 7509 I N 2C-E (Positional Isomer: 2,5-Dimethoxy-3,4-dimethylphenethylamine (2C-G))
2-(2,5-Dimethoxy-4-methylphenyl) ethanamine (2C-D) 7508 I N 2C-D
2-(2,5-Dimethoxy-4-nitro-phenyl) ethanamine (2C-N) 7521 I N 2C-N
2-(2,5-Dimethoxyphenyl) ethanamine (2C-H) 7517 I N 2C-H
2-(4-bromo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7536 I N 25B-NBOMe, 2C-B-NBOMe, 25B, Cimbi-36 ethanamine (25B-NBOMe)
2-(4-Chloro-2,5-dimethoxyphenyl) ethanamine (2C-C) 7519 I N 2C-C
2-(4-chloro-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7537 I N 25C-NBOMe, 2C-C-NBOMe, 25C, Cimbi-82 ethanamine (25C-NBOMe)
2-(4-Ethylthio-2,5-dimethoxyphenyl) ethanamine (2C- 7385 I N 2C-T-2 T-2 )
2-(4-iodo-2,5-dimethoxyphenyl) ethanamine (2C-I) 7518 I N 2C-I
2-(4-iodo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7538 I N 25I-NBOMe, 2C-I-NBOMe, 25I, Cimbi-5 ethanamine (25I-NBOMe)
2-(4-Isopropylthio)-2,5-dimethoxyphenyl) ethanamine 7532 I N 2C-T-4 (Positional Isomer: 2,5-Dimethoxy-4-(2C-T-4 ) ethylthioamphetamine (Aleph-2))
2,5-Dimethoxy-4-(n)-propylthiophenethylamine (2C-T- 7348 I N 2C-T-7 (Positional Isomer: 2,5-Dimethoxy-4-7) ethylthioamphetamine (Aleph-2))
2,5-Dimethoxy-4-ethylamphetamine 7399 I N DOET
2,5-Dimethoxyamphetamine 7396 I N DMA, 2,5-DMA
2-methoxy-N-(1-phenethylpiperidin-4-yl)-N- 9825 I Y Methoxyacetyl fentanyl phenylacetamide
2,17-dimethyl-17-hydroxy-5-androstan-3-one 4000 III N
2,3-epithio-17-methyl-5-androstan-17-ol 4000 III N
3,4,5-Trimethoxyamphetamine 7390 I N TMA (Positional Isomers: 2,4,5-Trimethoxy-amphetamine (TMA-5), 2,4,6-Trimethoxy-amphetamine (TMA-6), Escaline)
3,4-Methylenedioxyamphetamine 7400 I N MDA, Love Drug
3,4-Methylenedioxymethamphetamine 7405 I N MDMA, Ecstasy, XTC
3,4-Methylenedioxy-N-ethylamphetamine 7404 I N N-ethyl MDA, MDE, MDEA
3Alpha,17beta-dihydroxy-5alpha-androstane 4000 III N
3Beta,17beta-dihydroxy-5alpha-androstane 4000 III N
3-Fluoro-N-methylcathinone (3-FMC) 1233 I N 1-(3-fluorophenyl)-2-(methylamino)propan-1-one) (Positional isomer: 2-FMC)
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
01-Mar-18 Page 2 of 16
-
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
3-Methylfentanyl 9813 I Y China White, fentanyl
3-Methylthiofentanyl 9833 I Y China White, fentanyl
3-hydroxy-estra-4,9,11-trien-17-one 4000 III N
4-Androstenediol (3beta,17beta-dihydroxy-androst-4- 4000 III N 4-AD ene)
4-Androstenedione (androst-4-en-3,17-dione) 4000 III N
4-Anilino-N-phenethyl-4-piperidine (ANPP) 8333 II N ANPP, Despropionyl fentanyl
4-Bromo-2,5-dimethoxyamphetamine 7391 I N DOB, 4-bromo-DMA
4-Bromo-2,5-dimethoxyphenethylamine 7392 I N 2C-B, Nexus, has been sold as Ecstasy, i.e. MDMA
4-chloro-17-methyl-17-hydroxy-androst-4-en-3-one 4000 III N
4-chloro-17-methyl-17-hydroxy-androst-4-ene-3,11- 4000 III N
dione
4-chloro-17-methyl-androst-4-ene-3,17-diol 4000 III N
4-chloro-17-methyl-androsta-1,4-diene-3,17-diol 4000 III N
4-Dihydrotestosterone (17beta-hydroxyandrostan-3- 4000 III N Anabolex, Andractim, Pesomax, Stanolone one)
4-Fluoroisobutyryl fentanyl (N-(4-fluorophenyl)-N-(1- 9824 I Y Para-fluoroisobutyryl fentanyl phenethylpiperidin-4-yl)isobutyramide)
4-Fluoro-N-methylcathinone (4-FMC) 1238 I N flephedrone; 1-(4-fluorophenyl)-2-(methylamino)propan-1-one) (Positional isomer: 2-FMC)
4-Hydroxy-19-nortestosterone (4,17beta-dihydroxyestr- 4000 III N
4-en-3-one)
4-Hydroxy-androst-4-ene-3,17-dione 4000 III N Listed as 4-Hydroxy-androst-4-ene-3,17-dione[3,2-c]pyrazole-5-androstan-17-ol
4-Hydroxytestosterone (4,17beta-dihydroxyandrost-4- 4000 III N
en-3-one)
4-Methoxyamphetamine 7411 I N PMA
4-Methyl-2,5-dimethoxyamphetamine 7395 I N DOM, STP (Positional Isomer: 2,5-Dimethoxy-3,4-dimethylphenethylamine (2C-G))
4-Methyl-alphapyrrolidinopropiophenone (4-MePPP) 7498 I N MePPP, 4-methyl--pyrrolidinopropiophenone, 1-(4-methylphenyl)-2-(pyrrolidin-1-yl)-propan-1-one)
4-Methylaminorex (cis isomer) 1590 I N U4Euh, McN-422
4-Methyl-N-ethylcathinone (4-MEC) 1249 I N 2-(ethylamino)-1-(4-methylphenyl)propan-1-one)(Positional Isomers:3-methylethcathinone (3-MEC), 4-ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-MeMABP;4-MeBP), 3,4-dimethylmethcathinone(3,4-DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-methylcathinone(EMC))
5-Androstenediol (3beta,17beta-dihydroxy-androst-5- 4000 III N
ene)
5-Androstenedione (androst-5-en-3,17-dione) 4000 III N
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
01-Mar-18 Page 3 of 16
-
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
5FADB; 5FMDMBPINACA (Methyl 2-(1-(5-fluoropentyl)-1H-indazole-3-carboxamido)-3,3-dimethylbutanoate)
7034 I N 5F-ADB, 5F-MDMB-PINACA
5FAMB (Methyl 2-(1-(5-fluoropentyl)-1H-indazole-3- 7033 I N 5F-AMB carboxamido)-3-methylbutanoate)
5FAPINACA, 5FAKB48 (N-(adamantan-1-yl)-1-(5- 7049 I N 5F-APINACA, 5F-AKB48 fluoropentyl)-1H-indazole-3-carboxamide)
5-Fluoro-UR-144 and XLR11 [1-(5-Fluoro-pentyl)1H- 7011 I N 5-Fluoro-UR-144, XLR-11 and XLR11 indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone
5F-PB-22 (Quinolin-8-yl 1-(5-fluoropentyl)-1H-indole-3- 7225 I N 5-Fluoro-PB-22; 5F-PB-22 carboxylate)
5-Methoxy-3,4-methylenedioxyamphetamine 7401 I N MMDA
5-Methoxy-N,N-diisopropyltryptamine 7439 I N 5-MeO-DIPT (Positional Isomer: 5-Methoxy-N,N-dipropyltryptamine (5-MeO-DPT))
5-Methoxy-N-N-dimethyltryptamine 7431 I N 5-MeO-DMT (Positional Isomer: 4-Methoxy-N,N-dimethyltryptamine (4-MeO-DMT))
5-Androstan-3,6,17-trione 4000 III N
6-bromo-androstan-3,17-dione 4000 III N
6-Methyl-androst-4-ene-3,17-dione 4000 III N
AB-CHMINACA (N-(1-amino-3-methyl-1- 7031 I N AB-CHMINACA oxobutan-2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide
AB-FUBINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)- 7012 I N AB-FUBINACA 1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)
AB-PINACA (N-(1-amino-3-methyl- 7023 I N AB-PINACA 1-oxobutan-2-yl)-1-pentyl-1H-indazole-3-carboxamide)
Acetorphine 9319 I Y
Acetyl Fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9821 I Y
phenylacetamide)
Acetyl-alpha-methylfentanyl 9815 I Y
Acetyldihydrocodeine 9051 I Y Acetylcodone
Acetylmethadol 9601 I Y Methadyl acetate
Acryl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9811 I Y Acryloylfentanyl phenylacrylamide)
ADBFUBINACA (N-(1-amino-3,3-dimethyl-1-oxobutan- 7010 I N ADB-FUBINACA 2-yl)-1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)
ADB-PINACA (N-(1-amino-3,3-dimethyl-1-oxobutan-2- 7035 I N ADB-PINACA yl)-1-pentyl-1H-indazole-3-carboxamide)
AH-7921 (3,4-dichloro-N-[(1- 9551 I Y AH-7921 dimethylamino)cyclohexylmethyl]benzamide))
Alfaxalone 2731 IV N Alfaxan, 5-pregnan-3-ol-11,20-dione
Alfentanil 9737 II Y Alfenta
Allylprodine 9602 I Y
Alphacetylmethadol except levo-alphacetylmethadol 9603 I Y
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
01-Mar-18 Page 4 of 16
-
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Alpha-ethyltryptamine 7249 I N ET, Trip
Alphameprodine 9604 I Y
Alphamethadol 9605 I Y
Alpha-methylfentanyl 9814 I Y China White, fentanyl
Alpha-methylthiofentanyl 9832 I Y China White, fentanyl
Alpha-methyltryptamine 7432 I N AMT (Positional Isomer: N-Methyltryptamine)
Alphaprodine 9010 II Y Nisentil
alpha-pyrrolidinobutiophenone (-PBP) 7546 I N 1-phenyl-2-(pyrrolidin-1-yl)butan-1-one)
alpha-pyrrolidinopentiophenone (-PVP) 7545 I N -pyrrolidinovalerophenone, 1-phenyl-2- (pyrrolidin-1-yl)pentan-1-one)(Positional isomers: 4-methyl--pyrrolidinobutiophenone (4-MePBP), 1-phenyl-2-(piperidin-1-yl)butan-1-one)
Alprazolam 2882 IV N Xanax
AM2201 (1-(5-Fluoropentyl)-3-(1-naphthoyl) indole) 7201 I N AM2201
AM-694 (1-(5-Fluoropentyl)-3-(2-iodobenzoyl) indole) 7694 I N AM-694
Aminorex 1585 I N has been sold as methamphetamine
Amobarbital 2125 II N Amytal, Tuinal
Amobarbital & noncontrolled active ingred. 2126 III N
Amobarbital suppository dosage form 2126 III N
Amphetamine 1100 II N Dexedrine, Adderall, Obetrol
Anabolic steroids 4000 III N "Body Building" drugs
Androstanedione (5alpha-androstan-3,17-dione) 4000 III N
Anileridine 9020 II Y Leritine
APINACA and AKB48 N-(1-Adamantyl)-1-pentyl-1H- 7048 I N APINACA and AKB48 indazole-3-carboxamide
Aprobarbital 2100 III N Alurate
Barbital 2145 IV N Veronal, Plexonal, barbitone
Barbituric acid derivative 2100 III N Barbiturates not specifically listed
Benzethidine 9606 I Y
Benzphetamine 1228 III N Didrex, Inapetyl
Benzylmorphine 9052 I Y
Betacetylmethadol 9607 I Y
Beta-hydroxy-3-methylfentanyl 9831 I Y China White, fentanyl
Beta-hydroxyfentanyl 9830 I Y China White, fentanyl
Beta-hydroxythiofentanyl 9836 I Y N-[1-[2-hydroxy-2-(thiophen-2-yl)ethyl]piperidin-4-yl]-N-phenylpropionamide, N-[1-[2-hydroxy-2-(2-thienyl)ethyl]-4-piperidinyl]-N-phenylpropanamide
Betameprodine 9608 I Y
Betamethadol 9609 I Y
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
01-Mar-18 Page 5 of 16
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SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Betaprodine 9611 I Y
Bezitramide 9800 II Y Burgodin
Bolasterone (7alpha,17alpha-dimethyl-17beta- 4000 III N
hydroxyandrost-4-en-3-one)
Boldenone (17beta-hydroxyandrost-1,4-diene-3-one) 4000 III N Equipoise, Parenabol, Vebonol, dehydrotestosterone
Boldione 4000 III N
Brivaracetam 2710 V N BRV, UCB-34714, Briviact, ((2S)-2-[(4R)-2-oxo-4-propylpyrrolidin-1-yl] butanamide)
Bromazepam 2748 IV N Lexotan, Lexatin, Lexotanil
Bufotenine 7433 I N Mappine, N,N-dimethylserotonin
Buprenorphine 9064 III Y Buprenex, Temgesic, Subutex, Suboxone
Butabarbital (secbutabarbital) 2100 III N Butisol, Butibel
Butalbital 2100 III N Fiorinal, Butalbital with aspirin
Butobarbital (butethal) 2100 III N Soneryl (UK)
Butorphanol 9720 IV N Stadol, Stadol NS, Torbugesic, Torbutrol
Butylone 7541 I N bk-MBDB; 1-(1,3-benzodioxol-5-yl)-2-(methylamino)butan-1-one) (Positional Isomers: -ethylone (bk-MDEA; MDEC), dimethylone (bk-MDDMA; MDDMC))
Butyryl Fentanyl 9822 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylbutyramide, N-(1-phenethylpiperidin-4-yl)-N-phenylbutanamide
Calusterone (7beta,17alpha-dimethyl-17beta- 4000 III N Methosarb hydroxyandrost-4-en-3-one)
Camazepam 2749 IV N Albego, Limpidon, Paxor
Carfentanil 9743 II Y Wildnil
Carisoprodol 8192 IV N Soma
Cathine 1230 IV N Constituent of "Khat" plant, (+)-norpseudoephedrine
Cathinone 1235 I N Constituent of "Khat" plant
Chloral betaine 2460 IV N Beta Chlor
Chloral hydrate 2465 IV N Noctec
Chlordiazepoxide 2744 IV N Librium, Libritabs, Limbitrol, SK-Lygen
Chlorhexadol 2510 III N Mechloral, Mecoral, Medodorm, Chloralodol
Chlorphentermine 1645 III N Pre-Sate, Lucofen, Apsedon, Desopimon
Clobazam 2751 IV N Urbadan, Urbanyl
Clonazepam 2737 IV N Klonopin, Clonopin
Clonitazene 9612 I Y
Clorazepate 2768 IV N Tranxene
Clortermine 1647 III N Voranil
Clostebol (4-chloro-17beta-hydroxyandrost-4-en-3-one) 4000 III N Alfa-Trofodermin, Clostene, 4-chlorotestosterone
Clotiazepam 2752 IV N Trecalmo, Rize, Clozan, Veratran
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
01-Mar-18 Page 6 of 16
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DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Cloxazolam 2753 IV N Akton, Lubalix, Olcadil, Sepazon
Coca Leaves 9040 II Y
Cocaine 9041 II Y Methyl benzoylecgonine, Crack
Codeine 9050 II Y Morphine methyl ester, methyl morphine
Codeine & isoquinoline alkaloid 90 mg/du 9803 III Y Codeine with papaverine or noscapine
Codeine combination product 90 mg/du 9804 III Y Empirin,Fiorinal,Tylenol,ASA or APAP w/codeine
Codeine methylbromide 9070 I Y
Codeine preparations - 200 mg/(100 ml or 100 gm) V Y Cosanyl,Robitussin A-C,Cheracol,Cerose,Pediacof
Codeine-N-oxide 9053 I Y
CP-47,497 (5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3- 7297 I N CP-47,497 hydroxycyclohexyl-phenol)
CP-47,497 C8 Homologue (5-(1,1-Dimethyloctyl)-2- 7298 I N CP-47,497 C8 Homologue [(1R,3S)3-hydroxycyclohexyl-phenol)
Cyclopentyl fentanyl 9847 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylcyclopentanecarboxamide
Cyclopropyl Fentanyl 9845 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylcyclopropanecarboxamide
Cyprenorphine 9054 I Y
Dehydrochloromethyltestosterone (4-chloro-17beta- 4000 III N Oral-Turinabol hydroxy-17alpha-methylandrost-1,4-dien-3-one)
Delorazepam 2754 IV N
Delta1-dihydrotestosterone (17beta-hydroxy-5alpha- 4000 III N 1-Testosterone androst-1-en-3-one)
Desomorphine 9055 I Y
Desoxymethyltestosterone 4000 III N
Dexfenfluramine 1670 IV N Redux
Dextromoramide 9613 I Y Palfium, Jetrium, Narcolo
Dextropropoxyphene dosage forms 9278 IV Y Darvon, propoxyphene, Darvocet, Propacet
Dextropropoxyphene, bulk (non-dosage forms) 9273 II Y Propoxyphene
Diampromide 9615 I Y
Diazepam 2765 IV N Valium, Diastat
Dichloralphenazone 2467 IV N Midrin, dichloralantipyrine
Diethylpropion 1610 IV N Tenuate, Tepanil
Diethylthiambutene 9616 I Y
Diethyltryptamine 7434 I N DET, N,N-Diethyltryptamine (Positional Isomer: N-Methyl-N-isopropyltryptamine (MiPT))
Difenoxin 9168 I Y Lyspafen
Difenoxin 1 mg/25 ug AtSO4/du 9167 IV Y Motofen
Difenoxin preparations - 0.5 mg/25 ug AtSO4/du V Y Motofen
Dihydrocodeine 9120 II Y Didrate, Parzone
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
01-Mar-18 Page 7 of 16
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SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Dihydrocodeine combination product 90 mg/du 9807 III Y Synalgos-DC, Compal
Dihydrocodeine preparations 100mg/(100 ml or 100 V Y Cophene-S, various others gm)
Dihydroetorphine 9334 II Y DHE
Dihydromorphine 9145 I Y
Dimenoxadol 9617 I Y
Dimepheptanol 9618 I Y
Dimethylthiambutene 9619 I Y
Dimethyltryptamine 7435 I N DMT
Dioxaphetyl butyrate 9621 I Y
Diphenoxylate 9170 II Y
Diphenoxylate preparations 2.5 mg/25 ug AtSO4 V Y Lomotil, Logen
Dipipanone 9622 I Y Dipipan, phenylpiperone HCl, Diconal, Wellconal
Dronabinol (synthetic) in sesame oil in soft gelatin 7369 III N Marinol, synthetic THC in sesame oil/soft gelatin as capsule as approved by FDA approved by FDA
Dronabinol in an oral solution in a drug product 7365 II N Syndros approved for marketing by the U.S. Food and Drug Administration
Drostanolone (17beta-hydroxy-2alpha-methyl-5alpha- 4000 III N Drolban, Masterid, Permastril androstan-3-one)
Drotebanol 9335 I Y Metebanyl, oxymethebanol
Ecgonine 9180 II Y Cocaine precursor, in Coca leaves
Eluxadoline 9725 IV N VIBERZI
Embutramide 2020 III N Tributane
Estazolam 2756 IV N ProSom, Domnamid, Eurodin, Nuctalon
Estra-4,9,11-triene-3,17-dione 4000 III N
Ethchlorvynol 2540 IV N Placidyl
Ethinamate 2545 IV N Valmid, Valamin
Ethyl loflazepate 2758 IV N
Ethylestrenol (17alpha-ethyl-17beta-hydroxyestr-4-ene) 4000 III N Maxibolin, Orabolin, Durabolin-O, Duraboral
Ethylmethylthiambutene 9623 I Y
Ethylmorphine 9190 II Y Dionin
Ethylmorphine combination product 15 mg/du 9808 III Y
Ethylmorphine preparations 100 mg/(100 ml or 100 gm) V Y
Etonitazene 9624 I Y
Etorphine (except HCl) 9056 I Y
Etorphine HCl 9059 II Y M 99
Etoxeridine 9625 I Y
Ezogabine 2779 V N Potiga
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
01-Mar-18 Page 8 of 16
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SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Fencamfamin 1760 IV N Reactivan
Fenethylline 1503 I N Captagon,amfetyline,ethyltheophylline amphetamine
Fenfluramine 1670 IV N Pondimin, Ponderal
Fenproporex 1575 IV N Gacilin, Solvolip
Fentanyl 9801 II Y Duragesic, Oralet, Actiq, Sublimaze, Innovar
Fentanyl related-compounds as defined in 21 CFR 9850 I Y
1308.11(h)
Fludiazepam 2759 IV N
Flunitrazepam 2763 IV N Rohypnol, Narcozep, Darkene, Roipnol
Fluoxymesterone (9-fluoro-17alpha-methyl- 4000 III N Anadroid-F, Halotestin, Ora-Testryl 11beta,17beta-dihydroxyandrost-4-en-3-one)
Flurazepam 2767 IV N Dalmane
Formebolone (2-formyl-17alpha-methyl- 4000 III N Esiclene, Hubernol 11alpha,17beta-dihydroxyandrost-1,4-dien-3-one)
Fospropofol 2138 IV N Lusedra
Furanyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9834 I Y
phenylfuran-2-carboxamide)
Furazabol (17alpha-methyl-17beta- 4000 III N Frazalon, Miotolon, Qu Zhi Shu hydroxyandrostano[2,3-c]-furazan)
Furethidine 9626 I Y
Gamma Hydroxybutyric Acid 2010 I N GHB, gamma hydroxybutyrate, sodium oxybate
Gamma Hydroxybutyric Acid preparations 2012 III N Xyrem
Glutethimide 2550 II N Doriden, Dorimide
Halazepam 2762 IV N Paxipam
Haloxazolam 2771 IV N
Heroin 9200 I Y Diacetylmorphine, diamorphine
Hydrocodone 9193 II Y dihydrocodeinone
Hydromorphinol 9301 I Y
Hydromorphone 9150 II Y Dilaudid, dihydromorphinone
Hydroxypethidine 9627 I Y
Ibogaine 7260 I N Constituent of "Tabernanthe iboga" plant
Isobutyryl fentanyl 9827 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylisobutyramide
Isomethadone 9226 II Y Isoamidone
JWH-018 (also known as AM678) (1-Pentyl-3-(1- 7118 I N JWH-018 and AM-678 naphthoyl)indole)
JWH-019 (1-Hexyl-3-(1-naphthoyl)indole) 7019 I N JWH-019
JWH-073 (1-Butyl-3-(1-naphthoyl)indole) 7173 I N JWH-073
JWH-081 (1-Pentyl-3-(1-(4-methoxynaphthoyl) indole) 7081 I N JWH-081
JWH-122 (1-Pentyl-3-(4-methyl-1-naphthoyl) indole) 7122 I N JWH-122
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
01-Mar-18 Page 9 of 16
-
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
JWH-200 (1-[2-(4-Morpholinyl)ethyl]-3-(1- 7200 I N JWH-200 naphthoyl)indole)
JWH-203 (1-Pentyl-3-(2-chlorophenylacetyl) indole) 7203 I N JWH-203
JWH-250 (1-Pentyl-3-(2-methoxyphenylacetyl) indole) 6250 I N JWH-250
JWH-398 (1-Pentyl-3-(4-chloro-1-naphthoyl) indole) 7398 I N JWH-398
Ketamine 7285 III N Ketaset, Ketalar, Special K, K
Ketazolam 2772 IV N Anxon, Loftran, Solatran, Contamex
Ketobemidone 9628 I Y Cliradon
Lacosamide 2746 V N Vimpat
Levo-alphacetylmethadol 9648 II Y LAAM, long acting methadone, levomethadyl acetate
Levomethorphan 9210 II Y
Levomoramide 9629 I Y
Levophenacylmorphan 9631 I Y
Levorphanol 9220 II Y Levo-Dromoran
Lisdexamfetamine 1205 II N Vyvanse
Loprazolam 2773 IV N
Lorazepam 2885 IV N Ativan
Lorcaserin 1625 IV N Belviq
Lormetazepam 2774 IV N Noctamid
Lysergic acid 7300 III N LSD precursor
Lysergic acid amide 7310 III N LSD precursor
Lysergic acid diethylamide 7315 I N LSD, lysergide
MAB-CHMINACA (N-(1-amino-3,3dimethyl-1- 7032 I N MAB-CHMINACA and ADB-CHMINACA oxobutan-2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide)
Marihuana 7360 I N Cannabis, marijuana
Marihuana Extract 7350 I N
Mazindol 1605 IV N Sanorex, Mazanor
MDMBCHMICA, MMBCHMINACA (Methyl 2-(1- 7042 I N MDMB-CHMICA, MMB-CHMINACA (cyclohexylmethyl)-1H-indole-3-carboxamido)-3,3-dimethylbutanoate)
MDMBFUBINACA (Methyl 2-(1-(4-fluorobenzyl)-1H- 7020 I N MDMB-FUBINACA indazole-3-carboxamido)-3,3-dimethylbutanoate)
MDPV (3,4-Methylenedioxypyrovalerone) 7535 I N MDPV
Mebutamate 2800 IV N Capla
Mecloqualone 2572 I N Nubarene
Medazepam 2836 IV N Nobrium
Mefenorex 1580 IV N Anorexic, Amexate, Doracil, Pondinil
Meperidine 9230 II Y Demerol, Mepergan, pethidine
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
01-Mar-18 Page 10 of 16
-
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Meperidine intermediate-A 9232 II Y Meperidine precursor
Meperidine intermediate-B 9233 II Y Meperidine precursor, normeperidine
Meperidine intermediate-C 9234 II Y Meperidine precursor
Mephedrone